JP2007529433A5 - - Google Patents
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- Publication number
- JP2007529433A5 JP2007529433A5 JP2007503195A JP2007503195A JP2007529433A5 JP 2007529433 A5 JP2007529433 A5 JP 2007529433A5 JP 2007503195 A JP2007503195 A JP 2007503195A JP 2007503195 A JP2007503195 A JP 2007503195A JP 2007529433 A5 JP2007529433 A5 JP 2007529433A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- compounds
- calcipotriol
- protecting group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 C[C@@]([C@@](CC1)[C@@](C)(CCC2)[C@@]1C2=C[C@@](C(C1)=C(C2)[C@](*)C[C@@]1O*)S2(=O)=O)C=C[C@](C1CC1)O Chemical compound C[C@@]([C@@](CC1)[C@@](C)(CCC2)[C@@]1C2=C[C@@](C(C1)=C(C2)[C@](*)C[C@@]1O*)S2(=O)=O)C=C[C@](C1CC1)O 0.000 description 3
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US55396204P | 2004-03-18 | 2004-03-18 | |
| DKPA200400454 | 2004-03-22 | ||
| PCT/DK2005/000161 WO2005087719A1 (en) | 2004-03-18 | 2005-03-10 | Stereoselective synthesis of vitamin d analogues |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2007529433A JP2007529433A (ja) | 2007-10-25 |
| JP2007529433A5 true JP2007529433A5 (enExample) | 2008-05-01 |
| JP4667450B2 JP4667450B2 (ja) | 2011-04-13 |
Family
ID=34961016
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007503195A Expired - Fee Related JP4667450B2 (ja) | 2004-03-18 | 2005-03-10 | ビタミンｄ類似体の立体選択的合成 |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP1730108B1 (enExample) |
| JP (1) | JP4667450B2 (enExample) |
| KR (1) | KR100859277B1 (enExample) |
| CN (1) | CN1934078B (enExample) |
| AR (1) | AR048274A1 (enExample) |
| AT (1) | ATE390411T1 (enExample) |
| BR (1) | BRPI0507318A (enExample) |
| CA (1) | CA2555260C (enExample) |
| CY (1) | CY1108156T1 (enExample) |
| DE (2) | DE602005005645T2 (enExample) |
| ES (1) | ES2304686T3 (enExample) |
| IL (1) | IL176718A (enExample) |
| PL (1) | PL1730108T3 (enExample) |
| RU (1) | RU2380359C2 (enExample) |
| SI (1) | SI1730108T1 (enExample) |
| TW (1) | TWI324063B (enExample) |
| WO (1) | WO2005087719A1 (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2378252C2 (ru) * | 2004-04-02 | 2010-01-10 | Лео Фарма А/С | Новый способ получения промежуточных соединений, применяемых для синтеза аналогов витамина d |
| BRPI0621471A2 (pt) | 2006-03-17 | 2012-09-11 | Leo Pharma As | métodos de isomerização de uma solução de um derivado de vitamina d, para produzir e preparar calcipotriol ou monoidrato de calcipotriol, e para a fabricação de uma formulação farmacêutica ou medicamento, e, uso de um reator foto-reator de fluxo direto ou foto-reator de fluxo contìnuo |
| US8013189B2 (en) | 2007-09-21 | 2011-09-06 | Basf Se | Accelerated amide and ester reductions with amine boranes and additives |
| WO2009153782A1 (en) * | 2008-06-17 | 2009-12-23 | Ben Gurion University Of The Negev R&D Authority | Substituted cyclohexylidene-ethylidene-octahydro-indene compounds |
| CN103265528B (zh) * | 2013-05-10 | 2015-05-06 | 湖南千金湘江药业股份有限公司 | 埃索美拉唑镁的制备方法 |
| CN106908524B (zh) * | 2015-12-23 | 2021-05-04 | 重庆华邦胜凯制药有限公司 | 卡泊三醇中间体l及其潜在基因毒性杂质的分离与测定方法 |
| CN107643354B (zh) * | 2016-07-22 | 2022-02-01 | 重庆华邦胜凯制药有限公司 | 卡泊三醇起始原料a及相关杂质的分离与测定方法 |
| ES2945426B2 (es) * | 2021-12-30 | 2024-01-22 | Laboratorios Vinas S A | Procedimiento para obtener epímeros 24S a partir de derivados de vitaminas D y procedimiento de obtención de vitaminas D relacionado |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH07100685B2 (ja) * | 1985-08-02 | 1995-11-01 | レオ・ファ−マシュ−ティカル・プロダクツ・リミテッド・エイ／エス（レ−ベンス・ケミスケ・ファブリック・プロデュクチオンスアクチ−セルスカブ） | 新規ビタミンｄ類似体 |
| JPH075542B2 (ja) * | 1988-09-14 | 1995-01-25 | 呉羽化学工業株式会社 | ビタミンｄ▲下３▼誘導体及びその製造方法 |
| US5247104A (en) * | 1992-11-04 | 1993-09-21 | Wisconsin Alumni Research Foundation | Preparation of 1α, 24-dihydroxyvitamin D analogs |
| US5763426A (en) * | 1993-01-15 | 1998-06-09 | Leo Pharmaceutical Products Ltd. | Crystalline form of a vitamin D analogue |
| US5449668A (en) * | 1993-06-04 | 1995-09-12 | Duphar International Research B.V. | Vitamin D compounds and method of preparing these compounds |
| GB9524812D0 (en) * | 1995-12-05 | 1996-02-07 | Leo Pharm Prod Ltd | Chemical compounds |
| GB9622590D0 (en) * | 1996-10-30 | 1997-01-08 | Leo Pharm Prod Ltd | Chemical compounds |
| US6262283B1 (en) * | 1996-12-06 | 2001-07-17 | Magainin Pharmaceuticals Inc. | Stereoselective synthesis of 24-hydroxylated compounds useful for the preparation of aminosterols, vitamin D analogs, and other compounds |
| WO2000024712A1 (en) * | 1998-10-23 | 2000-05-04 | Teijin Limited | Vitamin d3 derivatives and remedies for inflammatory respiratory diseases containing the same |
-
2005
- 2005-03-10 JP JP2007503195A patent/JP4667450B2/ja not_active Expired - Fee Related
- 2005-03-10 CA CA2555260A patent/CA2555260C/en not_active Expired - Fee Related
- 2005-03-10 EP EP05706821A patent/EP1730108B1/en not_active Expired - Lifetime
- 2005-03-10 PL PL05706821T patent/PL1730108T3/pl unknown
- 2005-03-10 CN CN2005800086209A patent/CN1934078B/zh not_active Expired - Fee Related
- 2005-03-10 DE DE602005005645T patent/DE602005005645T2/de not_active Expired - Lifetime
- 2005-03-10 WO PCT/DK2005/000161 patent/WO2005087719A1/en not_active Ceased
- 2005-03-10 KR KR1020067015590A patent/KR100859277B1/ko not_active Expired - Fee Related
- 2005-03-10 AT AT05706821T patent/ATE390411T1/de active
- 2005-03-10 ES ES05706821T patent/ES2304686T3/es not_active Expired - Lifetime
- 2005-03-10 SI SI200530248T patent/SI1730108T1/sl unknown
- 2005-03-10 BR BRPI0507318-9A patent/BRPI0507318A/pt not_active IP Right Cessation
- 2005-03-10 RU RU2006129922/04A patent/RU2380359C2/ru active
- 2005-03-10 DE DE05706821T patent/DE05706821T1/de active Pending
- 2005-03-16 TW TW094108053A patent/TWI324063B/zh not_active IP Right Cessation
- 2005-03-17 AR ARP050101046A patent/AR048274A1/es unknown
-
2006
- 2006-07-05 IL IL176718A patent/IL176718A/en active IP Right Grant
-
2008
- 2008-06-26 CY CY20081100667T patent/CY1108156T1/el unknown
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