JP2006522041A - インドロンアセトアミド誘導体、その調製方法及びその使用 - Google Patents
インドロンアセトアミド誘導体、その調製方法及びその使用 Download PDFInfo
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- JP2006522041A JP2006522041A JP2006504696A JP2006504696A JP2006522041A JP 2006522041 A JP2006522041 A JP 2006522041A JP 2006504696 A JP2006504696 A JP 2006504696A JP 2006504696 A JP2006504696 A JP 2006504696A JP 2006522041 A JP2006522041 A JP 2006522041A
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- dihydro
- indol
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Classifications
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/32—Oxygen atoms
- C07D209/34—Oxygen atoms in position 2
Landscapes
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
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- Pulmonology (AREA)
- Psychiatry (AREA)
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- Cardiology (AREA)
- Psychology (AREA)
- Immunology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP03007214 | 2003-03-31 | ||
| PCT/EP2004/002691 WO2004087658A1 (fr) | 2003-03-31 | 2004-03-16 | Derives d'indolone-acetamide, leurs procedes de preparation et leurs utilisations |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JP2006522041A true JP2006522041A (ja) | 2006-09-28 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006504696A Pending JP2006522041A (ja) | 2003-03-31 | 2004-03-16 | インドロンアセトアミド誘導体、その調製方法及びその使用 |
Country Status (19)
| Country | Link |
|---|---|
| US (2) | US7645887B2 (fr) |
| EP (1) | EP1620399B1 (fr) |
| JP (1) | JP2006522041A (fr) |
| KR (1) | KR20050119186A (fr) |
| CN (1) | CN100364973C (fr) |
| AR (1) | AR043959A1 (fr) |
| AT (1) | ATE482193T1 (fr) |
| AU (1) | AU2004226288A1 (fr) |
| BR (1) | BRPI0408863A (fr) |
| CA (1) | CA2520568A1 (fr) |
| DE (1) | DE602004029245D1 (fr) |
| ES (1) | ES2353461T3 (fr) |
| HK (1) | HK1089768A1 (fr) |
| MX (1) | MXPA05009089A (fr) |
| NO (1) | NO20055026L (fr) |
| RU (1) | RU2005131317A (fr) |
| TW (1) | TW200508197A (fr) |
| WO (1) | WO2004087658A1 (fr) |
| ZA (1) | ZA200507231B (fr) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
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| TW200508197A (en) | 2003-03-31 | 2005-03-01 | Ucb Sa | Indolone-acetamide derivatives, processes for preparing them and their uses |
| WO2005080334A1 (fr) * | 2004-02-23 | 2005-09-01 | Dainippon Sumitomo Pharma Co., Ltd. | Nouveau compose heterocyclique |
| ATE482194T1 (de) * | 2004-07-22 | 2010-10-15 | Ucb Pharma Sa | Indolonderivate, verfahren zu deren herstellung und deren anwendungen |
| US20090023778A1 (en) | 2005-04-28 | 2009-01-22 | Eisai R&D Management Co., Ltd. | Composition Containing Anti-Dementia Drug |
| ES2441178T3 (es) | 2005-06-01 | 2014-02-03 | Ucb Pharma, S.A. | Derivados de 2-oxo-1-pirrolidina, procedimientos para prepararlos y el uso terapéutico de los mismos sobre el sistema nervioso central |
| US7790726B2 (en) * | 2005-08-16 | 2010-09-07 | Chemocentryx, Inc. | Monocyclic and bicyclic compounds and methods of use |
| TW200801011A (en) | 2006-02-07 | 2008-01-01 | Astrazeneca Ab | New compounds II |
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| CN114874127B (zh) * | 2022-05-23 | 2023-06-09 | 中国药科大学 | 一种二氟羰基化吲哚酮类化合物的制备方法 |
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- 2004-03-16 KR KR1020057018789A patent/KR20050119186A/ko not_active Application Discontinuation
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- 2004-03-16 RU RU2005131317/04A patent/RU2005131317A/ru not_active Application Discontinuation
- 2004-03-16 EP EP04720863A patent/EP1620399B1/fr not_active Expired - Lifetime
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- 2004-03-16 DE DE602004029245T patent/DE602004029245D1/de not_active Expired - Lifetime
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Also Published As
| Publication number | Publication date |
|---|---|
| NO20055026D0 (no) | 2005-10-28 |
| CA2520568A1 (fr) | 2004-10-14 |
| CN100364973C (zh) | 2008-01-30 |
| US7964593B2 (en) | 2011-06-21 |
| WO2004087658A1 (fr) | 2004-10-14 |
| AU2004226288A1 (en) | 2004-10-14 |
| ES2353461T3 (es) | 2011-03-02 |
| ZA200507231B (en) | 2006-11-29 |
| BRPI0408863A (pt) | 2006-04-11 |
| MXPA05009089A (es) | 2005-11-17 |
| US20070043038A1 (en) | 2007-02-22 |
| DE602004029245D1 (de) | 2010-11-04 |
| NO20055026L (no) | 2005-12-22 |
| CN1768036A (zh) | 2006-05-03 |
| RU2005131317A (ru) | 2006-02-27 |
| HK1089768A1 (en) | 2006-12-08 |
| AR043959A1 (es) | 2005-08-17 |
| US20100069375A1 (en) | 2010-03-18 |
| US7645887B2 (en) | 2010-01-12 |
| KR20050119186A (ko) | 2005-12-20 |
| ATE482193T1 (de) | 2010-10-15 |
| TW200508197A (en) | 2005-03-01 |
| EP1620399A1 (fr) | 2006-02-01 |
| EP1620399B1 (fr) | 2010-09-22 |
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