JP2006511527A - 種々の薬学的用途のためのα2δリガンド - Google Patents
種々の薬学的用途のためのα2δリガンド Download PDFInfo
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- JP2006511527A JP2006511527A JP2004560036A JP2004560036A JP2006511527A JP 2006511527 A JP2006511527 A JP 2006511527A JP 2004560036 A JP2004560036 A JP 2004560036A JP 2004560036 A JP2004560036 A JP 2004560036A JP 2006511527 A JP2006511527 A JP 2006511527A
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- Prior art keywords
- aminomethyl
- pain
- acetic acid
- disorders
- disease
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/66—Phosphorus compounds
- A61K31/662—Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
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- A61K31/18—Sulfonamides
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- A61K31/19—Carboxylic acids, e.g. valproic acid
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- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
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- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
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- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
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- Dermatology (AREA)
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- Immunology (AREA)
- Pulmonology (AREA)
- Diabetes (AREA)
- Anesthesiology (AREA)
- Oncology (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
- AIDS & HIV (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US43349102P | 2002-12-13 | 2002-12-13 | |
| PCT/IB2003/005669 WO2004054559A1 (en) | 2002-12-13 | 2003-12-03 | Alpha2delta ligands for different pharmaceutical uses |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JP2006511527A true JP2006511527A (ja) | 2006-04-06 |
Family
ID=32595199
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004560041A Withdrawn JP2006515587A (ja) | 2002-12-13 | 2003-12-03 | 性的不能を治療する方法 |
| JP2004560036A Pending JP2006511527A (ja) | 2002-12-13 | 2003-12-03 | 種々の薬学的用途のためのα2δリガンド |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004560041A Withdrawn JP2006515587A (ja) | 2002-12-13 | 2003-12-03 | 性的不能を治療する方法 |
Country Status (15)
| Country | Link |
|---|---|
| US (8) | US7432299B2 (enExample) |
| EP (2) | EP1572172A1 (enExample) |
| JP (2) | JP2006515587A (enExample) |
| KR (2) | KR20050085537A (enExample) |
| CN (8) | CN100430048C (enExample) |
| AU (3) | AU2003303037A1 (enExample) |
| BR (2) | BR0317273A (enExample) |
| CA (3) | CA2451267A1 (enExample) |
| MX (2) | MXPA05006318A (enExample) |
| MY (1) | MY140525A (enExample) |
| NZ (2) | NZ566452A (enExample) |
| PL (2) | PL377729A1 (enExample) |
| TW (2) | TW200412241A (enExample) |
| WO (3) | WO2004054559A1 (enExample) |
| ZA (6) | ZA200503863B (enExample) |
Families Citing this family (38)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3693258B2 (ja) | 1996-07-24 | 2005-09-07 | ワーナー―ランバート・コンパニー | イソブチルgabaまたはその誘導体を含有する鎮静剤 |
| US20050043345A1 (en) * | 2003-08-22 | 2005-02-24 | Pfizer Inc | Pharmaceutical composition for the prevention and treatment of addiction in a mammal |
| US20050043407A1 (en) * | 2003-08-22 | 2005-02-24 | Pfizer Inc | Pharmaceutical composition for the prevention and treatment of addiction in a mammal |
| US20050043406A1 (en) * | 2003-08-22 | 2005-02-24 | Pfizer Inc | Pharmaceutical composition for the treatment of obesity or to facilitate or promote weight loss |
| EP1670452A2 (en) * | 2003-09-25 | 2006-06-21 | Warner-Lambert Company LLC | Method of use of aminoacids having affinity for the a2d protein |
| AR049384A1 (es) | 2004-05-24 | 2006-07-26 | Glaxo Group Ltd | Derivados de purina |
| EP1766077B1 (en) | 2004-06-21 | 2012-03-28 | The Board Of Trustees Of The Leland Stanford Junior University | Genes and pathways differentially expressed in bipolar disorder and/or major depressive disorder |
| JP4820819B2 (ja) * | 2004-08-02 | 2011-11-24 | 株式会社サビンサジャパンコーポレーション | 過剰増殖性皮膚疾患を治療するための組成物および方法 |
| ES2393768T3 (es) | 2005-05-26 | 2012-12-27 | Neuron Systems, Inc | Derivado de quinolina para el tratamiento de enfermedades retinianas |
| GB0514809D0 (en) | 2005-07-19 | 2005-08-24 | Glaxo Group Ltd | Compounds |
| EP1928450A2 (en) * | 2005-08-26 | 2008-06-11 | Xenoport, Inc. | Treating premature ejaculation using gabapentin and pregabalin prodrugs |
| DE102005050377A1 (de) * | 2005-10-21 | 2007-04-26 | Bayer Healthcare Ag | Heterocyclische Verbindungen und ihre Verwendung |
| EP2101752A1 (en) * | 2006-12-08 | 2009-09-23 | Xenoport, Inc. | Use of prodrugs of gaba analogs for treating diseases |
| DE102007001804A1 (de) * | 2007-01-12 | 2008-07-17 | Johann Wolfgang Goethe-Universität Frankfurt am Main | Verwendung von GABAB-Rezeptor selektiven Agonisten zur Behandlung entzündlicher Hauterkrankungen |
| WO2009055059A1 (en) * | 2007-10-26 | 2009-04-30 | The Scripps Research Institute | Methods for treating substance dependence |
| AU2008318311B2 (en) * | 2007-11-02 | 2014-05-15 | The Board Of Trustees Of The Leland Stanford Junior University | FGF9-related methods for treating anxiety |
| ES2601852T3 (es) * | 2008-01-25 | 2017-02-16 | Xenoport, Inc. | Forma cristalina de sales de calcio de ácidos (3S)-aminometil-5-metil-hexanoicos y métodos de uso |
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