IT1066857B - Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione - Google Patents

Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione

Info

Publication number
IT1066857B
IT1066857B IT27806/65A IT2780665A IT1066857B IT 1066857 B IT1066857 B IT 1066857B IT 27806/65 A IT27806/65 A IT 27806/65A IT 2780665 A IT2780665 A IT 2780665A IT 1066857 B IT1066857 B IT 1066857B
Authority
IT
Italy
Prior art keywords
ipiazole
pyridin
derivatives
processes
preparation
Prior art date
Application number
IT27806/65A
Other languages
English (en)
Inventor
Giuseppe Palazzo
Bruno Silvestrini
Original Assignee
Acraf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Acraf filed Critical Acraf
Priority to IT27806/65A priority Critical patent/IT1066857B/it
Priority to US590226A priority patent/US3381009A/en
Priority to GB5073866A priority patent/GB1117068A/en
Priority to BE743313D priority patent/BE743313A/fr
Application granted granted Critical
Publication of IT1066857B publication Critical patent/IT1066857B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
IT27806/65A 1965-12-15 1965-12-15 Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione IT1066857B (it)

Priority Applications (4)

Application Number Priority Date Filing Date Title
IT27806/65A IT1066857B (it) 1965-12-15 1965-12-15 Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione
US590226A US3381009A (en) 1965-12-15 1966-10-28 Triazole-(4,3-a)-pyridines
GB5073866A GB1117068A (en) 1965-12-15 1966-11-11 S-triazole-[4,3-a]-pyridine derivatives and processes for their preparation
BE743313D BE743313A (en) 1965-12-15 1969-12-17 (A) s-Triazolo-(4,3a)pyridines (I) where R = H or Me R' = H, (1-4C) alkyl, (1-4C) alkoxy, halogen (B) Non-toxic salts of (I) with organic and

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT27806/65A IT1066857B (it) 1965-12-15 1965-12-15 Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione

Publications (1)

Publication Number Publication Date
IT1066857B true IT1066857B (it) 1985-03-12

Family

ID=11222366

Family Applications (1)

Application Number Title Priority Date Filing Date
IT27806/65A IT1066857B (it) 1965-12-15 1965-12-15 Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione

Country Status (2)

Country Link
US (1) US3381009A (it)
IT (1) IT1066857B (it)

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IT1051559B (it) * 1972-02-29 1981-05-20 Acraf Procedimento per la peparazione di derivati della s.triazolo 4.3.a piridina
JPS5070389A (it) * 1973-10-30 1975-06-11
US4154832A (en) * 1974-08-26 1979-05-15 Bruno Silvestrini Novel treatment for acute organic cerebral syndromes (strokes)
IT1073639B (it) * 1976-05-05 1985-04-17 Acraf Impiego del trazodone e etoperidone nel morbo di parikinson ed in altre sindromi extrapiramidali caratterizzate da tremori
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IT1094076B (it) * 1978-04-18 1985-07-26 Acraf Cicloalchiltriazoli
US4465683A (en) * 1979-09-14 1984-08-14 Mead Johnson & Company Anti-psychotic agents
US4252806A (en) * 1979-09-24 1981-02-24 Mead Johnson & Company Triazoloquinolones
US4254124A (en) * 1979-09-24 1981-03-03 Mead Johnson & Company Antidepressant agent
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US4338317A (en) * 1981-03-16 1982-07-06 Mead Johnson & Company Phenoxyethyl-1,2,4,-triazol-3-one antidepressants
US4487773A (en) * 1981-03-16 1984-12-11 Mead Johnson & Company 1,2,4-Triazol-3-one antidepressants
US4340597A (en) * 1981-04-13 1982-07-20 Schering Corporation 1-Substituted-4-aryl-1,2,5,6-tetrahydro and hexahydropyridines
US4386091A (en) * 1982-02-24 1983-05-31 Mead Johnson & Company 2-Phenoxyalkyl-1,2,4-triazol-3-one antidepressants
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US4613600A (en) * 1983-09-30 1986-09-23 Mead Johnson & Company Antidepressant 1,2,4-triazolone compounds
US4596807A (en) * 1985-03-26 1986-06-24 Serotonin Industries Of Charleston Method and compositions for controlling pain, depression and sedation
FR2580648B1 (fr) * 1985-04-17 1987-05-15 Adir Nouveaux derives du triazole, leur procede de preparation et les compositions pharmaceutiques les renfermant
US4840952A (en) * 1985-11-01 1989-06-20 Bristol-Myers Company Method for treatment of male impotence
US4687771A (en) * 1985-11-01 1987-08-18 Bristol-Myers Company Method for treatment of male impotence
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IT1268414B1 (it) * 1993-07-01 1997-02-27 Angelini Francesco Ist Ricerca Enantiomeri farmacologicamente attivi
CA2144669A1 (en) * 1994-03-29 1995-09-30 Kozo Akasaka Biphenyl derivatives
CA2160423A1 (en) * 1994-11-02 1996-05-03 Hemant N. Joshi Salts of nefazodone having improved dissolution rates
JPH11500123A (ja) * 1995-02-15 1999-01-06 ファルマシア・アンド・アップジョン・カンパニー ＣＮＳおよび心臓病の治療のためのイミダゾ［１，２−ａ］ピリジン類
DE19734516A1 (de) * 1997-08-08 1999-02-11 Bayer Ag Verfahren zur Herstellung von N-Aryl-N'-alkyl-piperazinen
US6013654A (en) * 1997-08-14 2000-01-11 Pharmacia & Upjohn Company Imidazo[1,2-A]pyridines for the treatment of CNS and cardiac diseases
IL141235A (en) * 2000-02-09 2012-04-30 Novartis Int Pharm Ltd Combined use of an alpha-adrenoceptor antagonist and a muscarinic antagonist in the preparation of a drug for the treatment of non-malignant prostatic hyperplasia
US20020065286A1 (en) * 2000-08-21 2002-05-30 Davies Michael John Treatment of wounds
US20020091129A1 (en) * 2000-11-20 2002-07-11 Mitradev Boolell Treatment of premature ejaculation
GB0130219D0 (en) * 2001-12-18 2002-02-06 Pfizer Ltd Compounds for the treatment of sexual dysfunction
US20030229001A1 (en) * 2002-01-31 2003-12-11 Pfizer Inc. Treatment of male sexual dysfunction
GB0219961D0 (en) 2002-08-28 2002-10-02 Pfizer Ltd Oxytocin inhibitors
TWI319713B (en) * 2002-10-25 2010-01-21 Sustained-release tramadol formulations with 24-hour efficacy
US8487002B2 (en) * 2002-10-25 2013-07-16 Paladin Labs Inc. Controlled-release compositions
US7323462B2 (en) * 2002-12-10 2008-01-29 Pfizer Inc. Morpholine dopamine agonists
CA2451267A1 (en) * 2002-12-13 2004-06-13 Warner-Lambert Company Llc Pharmaceutical uses for alpha2delta ligands
PA8597401A1 (es) * 2003-03-14 2005-05-24 Pfizer Derivados del acido 3-(1-[3-(1,3-benzotiazol-6-il) propilcarbamoil] cicloalquil) propanoico como inhibidores de nep
US20040220186A1 (en) * 2003-04-30 2004-11-04 Pfizer Inc. PDE9 inhibitors for treating type 2 diabetes,metabolic syndrome, and cardiovascular disease
US20050065158A1 (en) * 2003-07-16 2005-03-24 Pfizer Inc. Treatment of sexual dysfunction
US7291640B2 (en) * 2003-09-22 2007-11-06 Pfizer Inc. Substituted triazole derivatives as oxytocin antagonists
US20060172006A1 (en) * 2003-10-10 2006-08-03 Vincent Lenaerts Sustained-release tramadol formulations with 24-hour clinical efficacy
US20050267096A1 (en) * 2004-05-26 2005-12-01 Pfizer Inc New indazole and indolone derivatives and their use pharmaceuticals
US20050288270A1 (en) * 2004-05-27 2005-12-29 Pfizer Inc New aminopyridine derivatives and their use as pharmaceuticals
JP2008533193A (ja) * 2005-03-21 2008-08-21 ファイザー・リミテッド オキシトシン拮抗薬としての置換トリアゾール誘導体
JP2008533192A (ja) * 2005-03-21 2008-08-21 ファイザー・リミテッド オキシトシンアンタゴニストとしての置換されたトリアゾール誘導体
EP1917257A1 (en) * 2005-08-10 2008-05-07 Pfizer Limited Substituted triazole derivatives as oxytocin antagonists
DK1931346T3 (da) * 2005-09-09 2012-10-22 Angelini Labopharm Llc Trazodonsammensætning til indgivelse en gang om dagen
ITMI20071603A1 (it) * 2007-08-03 2009-02-04 Acraf Trazodone e trazodone cloridrato in forma purificata
US8461389B2 (en) 2008-04-18 2013-06-11 University College Dublin, National University Of Ireland, Dublin Psycho-pharmaceuticals
TWI368512B (en) * 2009-04-30 2012-07-21 Univ Kaohsiung Medical Pharmaceutical compositions comprising chlorophenyl piperazine derived compounds and use of the compounds in producing medicaments
WO2012072665A1 (en) 2010-11-30 2012-06-07 Pharmaneuroboost N.V. Compositions comprising pipamperone and serotonin antagonist reuptake inhibitors
EP2785183B1 (en) * 2011-11-14 2018-12-19 Merck Sharp & Dohme Corp. Triazolopyridinone pde10 inhibitors
CA2937417C (en) * 2014-01-21 2022-04-12 Piramal Enterprises Limited An improved process for the preparation of trazodone and hydrochloride salt thereof
WO2016192657A1 (en) 2015-06-03 2016-12-08 Sunshine Lake Pharma Co., Ltd. Substituted piperazine compounds and methods of use and use thereof
PL234822B1 (pl) 2017-03-14 2020-04-30 Politechnika Krakowska Im Tadeusza Kosciuszki Sposób otrzymywania trazodonu
RS63323B1 (sr) 2018-02-07 2022-07-29 Acraf Kontinualni postupak za dobijanje trazodona
RU2706700C1 (ru) 2019-09-24 2019-11-20 Общество с ограниченной ответственностью "Научно-производственная компания "СКиФФ" Фармацевтическая композиция для коррекции поведения кошек и собак в стрессовых ситуациях

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DE1235930B (de) * 1963-10-15 1967-03-09 Acraf Verfahren zur Herstellung von als Heilmittel geeignetem 1-Phenyl-3-butyl-4-methyl-triazolon-(5)

Also Published As

Publication number Publication date
US3381009A (en) 1968-04-30

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