TW200412241A - Pharmaceutical uses for alpha2delta ligands - Google Patents

Pharmaceutical uses for alpha2delta ligands Download PDF

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Publication number
TW200412241A
TW200412241A TW092135260A TW92135260A TW200412241A TW 200412241 A TW200412241 A TW 200412241A TW 092135260 A TW092135260 A TW 092135260A TW 92135260 A TW92135260 A TW 92135260A TW 200412241 A TW200412241 A TW 200412241A
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TW
Taiwan
Prior art keywords
pain
aminomethyl
disorders
disease
methyl
Prior art date
Application number
TW092135260A
Other languages
English (en)
Chinese (zh)
Inventor
David James Dooley
Charles Price Taylor Jr
Andrew John Thorpe
Fong Wang
David Juergen Wustrow
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of TW200412241A publication Critical patent/TW200412241A/zh

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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/662Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
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    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/18Sulfonamides
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    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
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    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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TW092135260A 2002-12-13 2003-12-12 Pharmaceutical uses for alpha2delta ligands TW200412241A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US43349102P 2002-12-13 2002-12-13

Publications (1)

Publication Number Publication Date
TW200412241A true TW200412241A (en) 2004-07-16

Family

ID=32595199

Family Applications (2)

Application Number Title Priority Date Filing Date
TW092135260A TW200412241A (en) 2002-12-13 2003-12-12 Pharmaceutical uses for alpha2delta ligands
TW092135262A TWI286934B (en) 2002-12-13 2003-12-12 Method of treatment for sexual dysfunction

Family Applications After (1)

Application Number Title Priority Date Filing Date
TW092135262A TWI286934B (en) 2002-12-13 2003-12-12 Method of treatment for sexual dysfunction

Country Status (15)

Country Link
US (8) US7432299B2 (enExample)
EP (2) EP1572172A1 (enExample)
JP (2) JP2006515587A (enExample)
KR (2) KR20050085537A (enExample)
CN (8) CN100430048C (enExample)
AU (3) AU2003283708A1 (enExample)
BR (2) BR0317273A (enExample)
CA (3) CA2451267A1 (enExample)
MX (2) MXPA05005665A (enExample)
MY (1) MY140525A (enExample)
NZ (2) NZ539971A (enExample)
PL (2) PL377729A1 (enExample)
TW (2) TW200412241A (enExample)
WO (3) WO2004054559A1 (enExample)
ZA (6) ZA200503861B (enExample)

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WO2006002262A2 (en) 2004-06-21 2006-01-05 The Board Of Trustees Of The Leland Stanford Junior University Genes and pathways differentially expressed in bipolar disorder and/or major depressive disorder
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WO2007027476A2 (en) * 2005-08-26 2007-03-08 Xenoport, Inc. Treating premature ejaculation using gabapentin and pregabalin prodrugs
DE102005050377A1 (de) * 2005-10-21 2007-04-26 Bayer Healthcare Ag Heterocyclische Verbindungen und ihre Verwendung
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DE102007001804A1 (de) * 2007-01-12 2008-07-17 Johann Wolfgang Goethe-Universität Frankfurt am Main Verwendung von GABAB-Rezeptor selektiven Agonisten zur Behandlung entzündlicher Hauterkrankungen
AU2008317336A1 (en) * 2007-10-26 2009-04-30 The Scripps Research Institute Methods for treating substance dependence
WO2009059316A1 (en) * 2007-11-02 2009-05-07 The Board Of Trustees Of The Leland Stanford Junior University Fgf9-related methods for treating anxiety
US7868043B2 (en) 2008-01-25 2011-01-11 Xenoport, Inc. Mesophasic forms of (3S)-aminomethyl-5-methyl-hexanoic acid prodrugs and methods of use
EP2250148B1 (en) * 2008-01-25 2016-08-17 XenoPort, Inc. Crystalline form of calcium-salts of (3s)-aminomethyl-5-methyl-hexanoic acids and methods of use
CA2706575C (en) * 2008-01-25 2015-07-14 Xenoport, Inc. Enantiomerically resolving acyloxyalkyl thiocarbonates used in synthesizing acyloxyalkyl carbamate prodrugs
SG157299A1 (en) 2008-05-09 2009-12-29 Agency Science Tech & Res Diagnosis and treatment of kawasaki disease
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