JP2006509004A5 - - Google Patents
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- Publication number
- JP2006509004A5 JP2006509004A5 JP2004556131A JP2004556131A JP2006509004A5 JP 2006509004 A5 JP2006509004 A5 JP 2006509004A5 JP 2004556131 A JP2004556131 A JP 2004556131A JP 2004556131 A JP2004556131 A JP 2004556131A JP 2006509004 A5 JP2006509004 A5 JP 2006509004A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- group
- haloalkyl
- compound
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims description 21
- 229910052736 halogen Inorganic materials 0.000 claims description 18
- 150000002367 halogens Chemical class 0.000 claims description 18
- 229910052739 hydrogen Inorganic materials 0.000 claims description 7
- 239000001257 hydrogen Substances 0.000 claims description 7
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims description 6
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 claims 25
- 150000003839 salts Chemical class 0.000 claims 14
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims 11
- 125000006526 (C1-C2) alkyl group Chemical group 0.000 claims 10
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 claims 10
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 7
- 125000006272 (C3-C7) cycloalkyl group Chemical group 0.000 claims 6
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 claims 5
- 229910052760 oxygen Inorganic materials 0.000 claims 5
- 229910052717 sulfur Inorganic materials 0.000 claims 5
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims 4
- 125000002947 alkylene group Chemical group 0.000 claims 4
- 125000000623 heterocyclic group Chemical group 0.000 claims 4
- 125000006536 (C1-C2)alkoxy group Chemical group 0.000 claims 3
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 claims 3
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims 3
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims 3
- 125000006644 (C2-C6) haloalkynyl group Chemical group 0.000 claims 3
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 3
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims 3
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims 3
- 229910052799 carbon Inorganic materials 0.000 claims 3
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 claims 3
- 125000005842 heteroatom Chemical group 0.000 claims 3
- 229910052757 nitrogen Inorganic materials 0.000 claims 3
- 125000006583 (C1-C3) haloalkyl group Chemical group 0.000 claims 2
- 125000006274 (C1-C3)alkoxy group Chemical group 0.000 claims 2
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 claims 2
- 241000607479 Yersinia pestis Species 0.000 claims 2
- 125000003545 alkoxy group Chemical group 0.000 claims 2
- 239000003814 drug Substances 0.000 claims 2
- 238000000034 method Methods 0.000 claims 2
- 125000000896 monocarboxylic acid group Chemical group 0.000 claims 2
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 2
- 229920006395 saturated elastomer Polymers 0.000 claims 2
- 125000006677 (C1-C3) haloalkoxy group Chemical group 0.000 claims 1
- 125000006590 (C2-C6) alkenylene group Chemical group 0.000 claims 1
- 239000012872 agrochemical composition Substances 0.000 claims 1
- 125000000217 alkyl group Chemical group 0.000 claims 1
- 230000002152 alkylating effect Effects 0.000 claims 1
- 125000003118 aryl group Chemical group 0.000 claims 1
- 125000000392 cycloalkenyl group Chemical group 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 claims 1
- 238000003795 desorption Methods 0.000 claims 1
- 239000003085 diluting agent Substances 0.000 claims 1
- 150000002431 hydrogen Chemical class 0.000 claims 1
- 238000004519 manufacturing process Methods 0.000 claims 1
- 238000010534 nucleophilic substitution reaction Methods 0.000 claims 1
- 238000002360 preparation method Methods 0.000 claims 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims 1
- 125000004076 pyridyl group Chemical group 0.000 claims 1
- 125000006413 ring segment Chemical group 0.000 claims 1
- 239000004094 surface-active agent Substances 0.000 claims 1
- ZMXDDKWLCZADIW-UHFFFAOYSA-N N,N-Dimethylformamide Chemical compound CN(C)C=O ZMXDDKWLCZADIW-UHFFFAOYSA-N 0.000 description 3
- WYURNTSHIVDZCO-UHFFFAOYSA-N Tetrahydrofuran Chemical compound C1CCOC1 WYURNTSHIVDZCO-UHFFFAOYSA-N 0.000 description 2
- 0 **N(*)c1c(*)c(*)n[n]1C1=C(*)C=C(*)C=*CCC1 Chemical compound **N(*)c1c(*)c(*)n[n]1C1=C(*)C=C(*)C=*CCC1 0.000 description 1
- RYHBNJHYFVUHQT-UHFFFAOYSA-N 1,4-Dioxane Chemical compound C1COCCO1 RYHBNJHYFVUHQT-UHFFFAOYSA-N 0.000 description 1
- ZCYVEMRRCGMTRW-UHFFFAOYSA-N 7553-56-2 Chemical compound [I] ZCYVEMRRCGMTRW-UHFFFAOYSA-N 0.000 description 1
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 description 1
- KEAYESYHFKHZAL-UHFFFAOYSA-N Sodium Chemical compound [Na] KEAYESYHFKHZAL-UHFFFAOYSA-N 0.000 description 1
- 229910052801 chlorine Inorganic materials 0.000 description 1
- 239000000460 chlorine Substances 0.000 description 1
- 239000011630 iodine Substances 0.000 description 1
- 229910052740 iodine Inorganic materials 0.000 description 1
- 229910000104 sodium hydride Inorganic materials 0.000 description 1
- 239000012312 sodium hydride Substances 0.000 description 1
- 239000002904 solvent Substances 0.000 description 1
- YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02027062.5 | 2002-12-03 | ||
| EP02027062 | 2002-12-03 | ||
| PCT/EP2003/012619 WO2004049803A1 (en) | 2002-12-03 | 2003-11-12 | Pesticidal 5- (acylamino) pyrazole derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2006509004A JP2006509004A (ja) | 2006-03-16 |
| JP2006509004A5 true JP2006509004A5 (https=) | 2006-12-28 |
| JP4759682B2 JP4759682B2 (ja) | 2011-08-31 |
Family
ID=32405692
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004556131A Expired - Fee Related JP4759682B2 (ja) | 2002-12-03 | 2003-11-12 | 農薬としての５−（アシルアミノ）ピラゾール誘導体 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US7514561B2 (https=) |
| EP (1) | EP1569517B1 (https=) |
| JP (1) | JP4759682B2 (https=) |
| KR (1) | KR101288753B1 (https=) |
| CN (2) | CN1944413A (https=) |
| AR (1) | AR042255A1 (https=) |
| AU (1) | AU2003288038B2 (https=) |
| BR (1) | BRPI0316993B1 (https=) |
| CA (1) | CA2508412C (https=) |
| CO (1) | CO5690506A2 (https=) |
| EA (1) | EA011505B1 (https=) |
| ES (1) | ES2436746T3 (https=) |
| MX (1) | MXPA05005899A (https=) |
| NZ (1) | NZ540462A (https=) |
| WO (1) | WO2004049803A1 (https=) |
| ZA (1) | ZA200503743B (https=) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090048258A1 (en) * | 2005-02-01 | 2009-02-19 | Masaki Ogino | Amide Compound |
| US20080176826A1 (en) * | 2005-05-25 | 2008-07-24 | Michael Puhl | Pyridine Compounds For Combating Arthropod Pests and Nematodes |
| MY155497A (en) | 2008-11-19 | 2015-10-30 | Merial Inc | Compositions comprising an aryl pyrazole and/or a formamidine, methods and use thereof |
| UA108641C2 (uk) | 2010-04-02 | 2015-05-25 | Паразитицидна композиція, яка містить чотири активних агенти, та спосіб її застосування | |
| JP6027128B2 (ja) * | 2011-10-26 | 2016-11-16 | ダウ アグロサイエンシィズ エルエルシー | 有害生物防除組成物およびそれに関連した方法 |
| AU2012340351B2 (en) | 2011-11-17 | 2017-06-15 | Boehringer Ingelheim Animal Health USA Inc. | Compositions comprising an aryl pyrazole and a substituted imidazole, methods and uses thereof |
| CA2926095A1 (en) | 2013-10-17 | 2015-04-23 | Dow Agrosciences Llc | Processes for the preparation of pesticidal compounds |
| JP2016539092A (ja) | 2013-10-17 | 2016-12-15 | ダウ アグロサイエンシィズ エルエルシー | 有害生物防除性化合物の製造方法 |
| US9029554B1 (en) | 2013-10-17 | 2015-05-12 | Dow Agrosciences Llc | Processes for the preparation of pesticidal compounds |
| EP3057429A4 (en) | 2013-10-17 | 2017-08-09 | Dow AgroSciences LLC | Processes for the preparation of pesticidal compounds |
| CA2925953C (en) | 2013-10-17 | 2021-11-02 | Dow Agrosciences Llc | Processes for the preparation of pesticidal compounds |
| CA2925952A1 (en) | 2013-10-17 | 2015-04-23 | Dow Agrosciences Llc | Processes for the preparation of pesticidal compounds |
| MX2016004941A (es) * | 2013-10-17 | 2016-06-28 | Dow Agrosciences Llc | Proceso para la preparacion de compuestos plaguicidas. |
| GB201322334D0 (en) | 2013-12-17 | 2014-01-29 | Agency Science Tech & Res | Maleimide derivatives as modulators of WNT pathway |
| BR112017000293A2 (pt) | 2014-07-31 | 2017-10-31 | Dow Agrosciences Llc | processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina |
| JP2017523168A (ja) | 2014-07-31 | 2017-08-17 | ダウ アグロサイエンシィズ エルエルシー | ３−（３−クロロ−１ｈ−ピラゾール−１−イル）ピリジンの製造方法 |
| US9249122B1 (en) | 2014-07-31 | 2016-02-02 | Dow Agrosciences Llc | Process for the preparation of 3-(3-chloro-1H-pyrazol-1-yl)pyridine |
| JP2017525703A (ja) | 2014-08-19 | 2017-09-07 | ダウ アグロサイエンシィズ エルエルシー | ３−（３−クロロ−１ｈ−ピラゾール−１−イル）ピリジンの調製方法 |
| AR098113A1 (es) | 2014-09-12 | 2016-05-04 | Dow Agrosciences Llc | Proceso para la preparación de 3-(3-cloro-1h-pirazol-1-il)piridina |
| US10864193B2 (en) | 2014-10-31 | 2020-12-15 | Boehringer Ingelheim Animal Health USA Inc. | Parasiticidal compositions comprising fipronil at high concentrations |
| WO2016163379A1 (ja) * | 2015-04-09 | 2016-10-13 | 住友化学株式会社 | オキサリルアミド化合物及びその有害節足動物防除用途 |
| WO2016163383A1 (ja) * | 2015-04-09 | 2016-10-13 | 住友化学株式会社 | オキサリルアミド化合物及びその有害節足動物防除用途 |
| CN105732505B (zh) * | 2016-01-28 | 2018-10-12 | 中南民族大学 | 丙烯酰胺化芳基吡唑型化合物及其溶剂热一锅合成法与应用 |
| CN105712933B (zh) * | 2016-01-28 | 2019-01-11 | 中南民族大学 | 甲酰化芳基吡唑衍生物及其醚热合成方法和应用 |
| CN106417329B (zh) * | 2016-09-27 | 2019-08-27 | 辽宁省蚕业科学研究所 | 一类柞蚕饰腹寄蝇病防治化合物及使用方法 |
| JP2020503336A (ja) | 2016-12-29 | 2020-01-30 | ダウ アグロサイエンシィズ エルエルシー | 殺有害生物化合物の調製方法 |
| CN110325036B (zh) | 2016-12-29 | 2021-10-26 | 美国陶氏益农公司 | 用于制备杀虫化合物的方法 |
| CN107629005A (zh) * | 2017-08-22 | 2018-01-26 | 王泊理 | 多取代苯基吡唑衍生物及其制备方法和用途 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3602728A1 (de) | 1985-05-17 | 1986-11-20 | Bayer Ag, 51373 Leverkusen | Schaedlingsbekaempfungsmittel auf basis von pyrazolderivaten |
| GB8713768D0 (en) | 1987-06-12 | 1987-07-15 | May & Baker Ltd | Compositions of matter |
| US5232940A (en) | 1985-12-20 | 1993-08-03 | Hatton Leslie R | Derivatives of N-phenylpyrazoles |
| GB8531485D0 (en) | 1985-12-20 | 1986-02-05 | May & Baker Ltd | Compositions of matter |
| GB9120641D0 (en) | 1991-09-27 | 1991-11-06 | Ici Plc | Heterocyclic compounds |
| US5556873A (en) | 1993-02-24 | 1996-09-17 | Rhone-Poulenc Inc. | Pesticidal 1-aryl-5-(substituted alkyl (thio) amido)pyrazoles |
| GB9306184D0 (en) | 1993-03-25 | 1993-05-19 | Zeneca Ltd | Heteroaromatic compounds |
| DE4343832A1 (de) | 1993-12-22 | 1995-06-29 | Bayer Ag | Substituierte 1-Arylpyrazole |
| DE4414333A1 (de) | 1994-04-25 | 1995-10-26 | Bayer Ag | Substituierte Pyridylpyrazole |
| US6316477B1 (en) | 1996-01-30 | 2001-11-13 | Takeda Chemical Industries, Ltd. | Arylpyrazole insecticides |
| EP0811615A1 (en) * | 1996-06-03 | 1997-12-10 | Rhone-Poulenc Agrochimie | 1-Aryl-5-(substituted alkyl (thio) amido) pyrazoles and their use as pesticides |
| JP3735159B2 (ja) * | 1996-06-17 | 2006-01-18 | ローヌ−プーラン・アグロシミ | 新規な農薬 |
| GB9625045D0 (en) | 1996-11-30 | 1997-01-22 | Pfizer Ltd | Parasiticidal compounds |
| DE19650197A1 (de) | 1996-12-04 | 1998-06-10 | Bayer Ag | 3-Thiocarbamoylpyrazol-Derivate |
| AR021608A1 (es) | 1998-12-11 | 2002-07-31 | Merial Ltd | Represion de artropodos en animales |
-
2003
- 2003-11-12 US US10/537,547 patent/US7514561B2/en not_active Expired - Lifetime
- 2003-11-12 JP JP2004556131A patent/JP4759682B2/ja not_active Expired - Fee Related
- 2003-11-12 WO PCT/EP2003/012619 patent/WO2004049803A1/en not_active Ceased
- 2003-11-12 MX MXPA05005899A patent/MXPA05005899A/es active IP Right Grant
- 2003-11-12 CA CA2508412A patent/CA2508412C/en not_active Expired - Fee Related
- 2003-11-12 CN CNA2006101492437A patent/CN1944413A/zh active Pending
- 2003-11-12 NZ NZ540462A patent/NZ540462A/en not_active IP Right Cessation
- 2003-11-12 BR BRPI0316993A patent/BRPI0316993B1/pt not_active IP Right Cessation
- 2003-11-12 AU AU2003288038A patent/AU2003288038B2/en not_active Ceased
- 2003-11-12 EP EP03779895.6A patent/EP1569517B1/en not_active Expired - Lifetime
- 2003-11-12 CN CNA2003801048559A patent/CN1719974A/zh active Pending
- 2003-11-12 KR KR1020057009951A patent/KR101288753B1/ko not_active Expired - Fee Related
- 2003-11-12 EA EA200500930A patent/EA011505B1/ru not_active IP Right Cessation
- 2003-11-12 ES ES03779895.6T patent/ES2436746T3/es not_active Expired - Lifetime
- 2003-12-01 AR ARP030104421A patent/AR042255A1/es active IP Right Grant
-
2005
- 2005-05-10 ZA ZA200503743A patent/ZA200503743B/en unknown
- 2005-05-31 CO CO05052700A patent/CO5690506A2/es active IP Right Grant
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