KR101288753B1 - 살충성 5-(아실아미노)피라졸 유도체 - Google Patents

살충성 5-(아실아미노)피라졸 유도체 Download PDF

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Publication number
KR101288753B1
KR101288753B1 KR1020057009951A KR20057009951A KR101288753B1 KR 101288753 B1 KR101288753 B1 KR 101288753B1 KR 1020057009951 A KR1020057009951 A KR 1020057009951A KR 20057009951 A KR20057009951 A KR 20057009951A KR 101288753 B1 KR101288753 B1 KR 101288753B1
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South Korea
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alkyl
formula
compound
haloalkyl
group
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KR1020057009951A
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English (en)
Korean (ko)
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KR20050084103A (ko
Inventor
스테판 쉬나테러
데이비드 윌리암 호킨스
다니엘라 얀
마이클 마이어
안케 쿨만
에리크 프리에드리히 산왈드
마리아-테레샤 토네센
칼 시거
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바이엘 에스.에이.에스
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020057009951A 2002-12-03 2003-11-12 살충성 5-(아실아미노)피라졸 유도체 Expired - Fee Related KR101288753B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP02027062.5 2002-12-03
EP02027062 2002-12-03
PCT/EP2003/012619 WO2004049803A1 (en) 2002-12-03 2003-11-12 Pesticidal 5- (acylamino) pyrazole derivatives

Publications (2)

Publication Number Publication Date
KR20050084103A KR20050084103A (ko) 2005-08-26
KR101288753B1 true KR101288753B1 (ko) 2013-07-23

Family

ID=32405692

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020057009951A Expired - Fee Related KR101288753B1 (ko) 2002-12-03 2003-11-12 살충성 5-(아실아미노)피라졸 유도체

Country Status (16)

Country Link
US (1) US7514561B2 (https=)
EP (1) EP1569517B1 (https=)
JP (1) JP4759682B2 (https=)
KR (1) KR101288753B1 (https=)
CN (2) CN1719974A (https=)
AR (1) AR042255A1 (https=)
AU (1) AU2003288038B2 (https=)
BR (1) BRPI0316993B1 (https=)
CA (1) CA2508412C (https=)
CO (1) CO5690506A2 (https=)
EA (1) EA011505B1 (https=)
ES (1) ES2436746T3 (https=)
MX (1) MXPA05005899A (https=)
NZ (1) NZ540462A (https=)
WO (1) WO2004049803A1 (https=)
ZA (1) ZA200503743B (https=)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006082952A1 (ja) * 2005-02-01 2006-08-10 Takeda Pharmaceutical Company Limited アミド化合物
JP2008542224A (ja) * 2005-05-25 2008-11-27 ビーエーエスエフ ソシエタス・ヨーロピア 節足動物害虫および線虫を防除するためのピリジン化合物
ES2781828T3 (es) 2008-11-19 2020-09-08 Boehringer Ingelheim Animal Health Usa Inc Composiciones que comprenden un aril pirazol y/o una formamidina, procedimientos y usos de las mismas
UA108641C2 (uk) 2010-04-02 2015-05-25 Паразитицидна композиція, яка містить чотири активних агенти, та спосіб її застосування
JP6027128B2 (ja) * 2011-10-26 2016-11-16 ダウ アグロサイエンシィズ エルエルシー 有害生物防除組成物およびそれに関連した方法
CN104023720B (zh) 2011-11-17 2016-10-26 梅里亚有限公司 包含芳基吡唑和取代咪唑的组合物，其方法和用途
JP2016536295A (ja) 2013-10-17 2016-11-24 ダウ アグロサイエンシィズ エルエルシー 有害生物防除性化合物の製造方法
WO2015058024A1 (en) 2013-10-17 2015-04-23 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
WO2015058022A1 (en) 2013-10-17 2015-04-23 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
CN105636440A (zh) 2013-10-17 2016-06-01 美国陶氏益农公司 制备杀虫化合物的方法
WO2015058028A1 (en) 2013-10-17 2015-04-23 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
US9174962B2 (en) 2013-10-17 2015-11-03 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
US9085564B2 (en) 2013-10-17 2015-07-21 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
GB201322334D0 (en) 2013-12-17 2014-01-29 Agency Science Tech & Res Maleimide derivatives as modulators of WNT pathway
EP3174856A4 (en) 2014-07-31 2018-01-10 Dow AgroSciences LLC Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine
JP2017523168A (ja) 2014-07-31 2017-08-17 ダウ アグロサイエンシィズ エルエルシー ３−（３−クロロ−１ｈ−ピラゾール−１−イル）ピリジンの製造方法
BR112017000565A2 (pt) 2014-07-31 2017-11-07 Dow Agrosciences Llc processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina
EP3183238A4 (en) 2014-08-19 2018-01-10 Dow AgroSciences LLC Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine
BR112017004613A2 (pt) 2014-09-12 2017-12-05 Dow Agrosciences Llc processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina
WO2016069983A1 (en) 2014-10-31 2016-05-06 Merial, Inc. Parasiticidal composition comprising fipronil
WO2016163379A1 (ja) * 2015-04-09 2016-10-13 住友化学株式会社 オキサリルアミド化合物及びその有害節足動物防除用途
WO2016163383A1 (ja) * 2015-04-09 2016-10-13 住友化学株式会社 オキサリルアミド化合物及びその有害節足動物防除用途
CN105712933B (zh) * 2016-01-28 2019-01-11 中南民族大学 甲酰化芳基吡唑衍生物及其醚热合成方法和应用
CN105732505B (zh) * 2016-01-28 2018-10-12 中南民族大学 丙烯酰胺化芳基吡唑型化合物及其溶剂热一锅合成法与应用
CN106417329B (zh) * 2016-09-27 2019-08-27 辽宁省蚕业科学研究所 一类柞蚕饰腹寄蝇病防治化合物及使用方法
CN110325036B (zh) 2016-12-29 2021-10-26 美国陶氏益农公司 用于制备杀虫化合物的方法
WO2018125815A1 (en) 2016-12-29 2018-07-05 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
CN107629005A (zh) * 2017-08-22 2018-01-26 王泊理 多取代苯基吡唑衍生物及其制备方法和用途

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5556873A (en) * 1993-02-24 1996-09-17 Rhone-Poulenc Inc. Pesticidal 1-aryl-5-(substituted alkyl (thio) amido)pyrazoles
EP0811615A1 (en) * 1996-06-03 1997-12-10 Rhone-Poulenc Agrochimie 1-Aryl-5-(substituted alkyl (thio) amido) pyrazoles and their use as pesticides
JPH107509A (ja) * 1996-06-17 1998-01-13 Rhone Poulenc Agrochim 新規な農薬
JP2002532477A (ja) * 1998-12-11 2002-10-02 アベンティス・クロップサイエンス・エス・アー 動物における節足動物の制御

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3602728A1 (de) 1985-05-17 1986-11-20 Bayer Ag, 51373 Leverkusen Schaedlingsbekaempfungsmittel auf basis von pyrazolderivaten
GB8531485D0 (en) 1985-12-20 1986-02-05 May & Baker Ltd Compositions of matter
US5232940A (en) 1985-12-20 1993-08-03 Hatton Leslie R Derivatives of N-phenylpyrazoles
GB8713768D0 (en) 1987-06-12 1987-07-15 May & Baker Ltd Compositions of matter
GB9120641D0 (en) 1991-09-27 1991-11-06 Ici Plc Heterocyclic compounds
GB9306184D0 (en) 1993-03-25 1993-05-19 Zeneca Ltd Heteroaromatic compounds
DE4343832A1 (de) 1993-12-22 1995-06-29 Bayer Ag Substituierte 1-Arylpyrazole
DE4414333A1 (de) 1994-04-25 1995-10-26 Bayer Ag Substituierte Pyridylpyrazole
JPH10152476A (ja) 1996-01-30 1998-06-09 Takeda Chem Ind Ltd １−アリールピラゾール誘導体、その製造法および用途
GB9625045D0 (en) 1996-11-30 1997-01-22 Pfizer Ltd Parasiticidal compounds
DE19650197A1 (de) 1996-12-04 1998-06-10 Bayer Ag 3-Thiocarbamoylpyrazol-Derivate

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5556873A (en) * 1993-02-24 1996-09-17 Rhone-Poulenc Inc. Pesticidal 1-aryl-5-(substituted alkyl (thio) amido)pyrazoles
EP0811615A1 (en) * 1996-06-03 1997-12-10 Rhone-Poulenc Agrochimie 1-Aryl-5-(substituted alkyl (thio) amido) pyrazoles and their use as pesticides
JPH107509A (ja) * 1996-06-17 1998-01-13 Rhone Poulenc Agrochim 新規な農薬
JP2002532477A (ja) * 1998-12-11 2002-10-02 アベンティス・クロップサイエンス・エス・アー 動物における節足動物の制御

Also Published As

Publication number Publication date
JP2006509004A (ja) 2006-03-16
US20060135778A1 (en) 2006-06-22
EA011505B1 (ru) 2009-04-28
CO5690506A2 (es) 2006-10-31
CN1944413A (zh) 2007-04-11
CA2508412A1 (en) 2004-06-17
WO2004049803A1 (en) 2004-06-17
EA200500930A1 (ru) 2006-10-27
EP1569517B1 (en) 2013-10-02
AU2003288038A1 (en) 2004-06-23
ES2436746T3 (es) 2014-01-07
CA2508412C (en) 2011-07-26
EP1569517A1 (en) 2005-09-07
US7514561B2 (en) 2009-04-07
KR20050084103A (ko) 2005-08-26
AR042255A1 (es) 2005-06-15
MXPA05005899A (es) 2005-08-29
ZA200503743B (en) 2006-11-29
AU2003288038B2 (en) 2009-04-23
NZ540462A (en) 2008-03-28
BRPI0316993B1 (pt) 2016-07-05
BR0316993A (pt) 2005-10-25
JP4759682B2 (ja) 2011-08-31
CN1719974A (zh) 2006-01-11

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