AU2003288038B2 - Pesticidal 5- (acylamino) pyrazole derivatives - Google Patents

Pesticidal 5- (acylamino) pyrazole derivatives Download PDF

Info

Publication number
AU2003288038B2
AU2003288038B2 AU2003288038A AU2003288038A AU2003288038B2 AU 2003288038 B2 AU2003288038 B2 AU 2003288038B2 AU 2003288038 A AU2003288038 A AU 2003288038A AU 2003288038 A AU2003288038 A AU 2003288038A AU 2003288038 B2 AU2003288038 B2 AU 2003288038B2
Authority
AU
Australia
Prior art keywords
alkyl
compound
haloalkyl
group
alkoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU2003288038A
Other languages
English (en)
Other versions
AU2003288038A1 (en
Inventor
David William Hawkins
Daniela Jans
Anke Kuhlmann
Michael Maier
Erich Friedrich Sanwald
Stefan Schnatterer
Karl Seeger
Maria-Theresia Thonessen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Animal Health USA Inc
Original Assignee
Boehringer Ingelheim Animal Health USA Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Animal Health USA Inc filed Critical Boehringer Ingelheim Animal Health USA Inc
Publication of AU2003288038A1 publication Critical patent/AU2003288038A1/en
Assigned to MERIAL LTD reassignment MERIAL LTD Request for Assignment Assignors: BAYER CROPSCIENCE S.A.
Application granted granted Critical
Publication of AU2003288038B2 publication Critical patent/AU2003288038B2/en
Assigned to MERIAL, INC. reassignment MERIAL, INC. Request for Assignment Assignors: MERIAL LTD
Assigned to Boehringer Ingelheim Animal Health USA Inc. reassignment Boehringer Ingelheim Animal Health USA Inc. Request for Assignment Assignors: MERIAL, INC.
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/561,2-Diazoles; Hydrogenated 1,2-diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/44Oxygen and nitrogen or sulfur and nitrogen atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2003288038A 2002-12-03 2003-11-12 Pesticidal 5- (acylamino) pyrazole derivatives Ceased AU2003288038B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP02027062.5 2002-12-03
EP02027062 2002-12-03
PCT/EP2003/012619 WO2004049803A1 (en) 2002-12-03 2003-11-12 Pesticidal 5- (acylamino) pyrazole derivatives

Publications (2)

Publication Number Publication Date
AU2003288038A1 AU2003288038A1 (en) 2004-06-23
AU2003288038B2 true AU2003288038B2 (en) 2009-04-23

Family

ID=32405692

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003288038A Ceased AU2003288038B2 (en) 2002-12-03 2003-11-12 Pesticidal 5- (acylamino) pyrazole derivatives

Country Status (16)

Country Link
US (1) US7514561B2 (https=)
EP (1) EP1569517B1 (https=)
JP (1) JP4759682B2 (https=)
KR (1) KR101288753B1 (https=)
CN (2) CN1944413A (https=)
AR (1) AR042255A1 (https=)
AU (1) AU2003288038B2 (https=)
BR (1) BRPI0316993B1 (https=)
CA (1) CA2508412C (https=)
CO (1) CO5690506A2 (https=)
EA (1) EA011505B1 (https=)
ES (1) ES2436746T3 (https=)
MX (1) MXPA05005899A (https=)
NZ (1) NZ540462A (https=)
WO (1) WO2004049803A1 (https=)
ZA (1) ZA200503743B (https=)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20090048258A1 (en) * 2005-02-01 2009-02-19 Masaki Ogino Amide Compound
US20080176826A1 (en) * 2005-05-25 2008-07-24 Michael Puhl Pyridine Compounds For Combating Arthropod Pests and Nematodes
MY155497A (en) 2008-11-19 2015-10-30 Merial Inc Compositions comprising an aryl pyrazole and/or a formamidine, methods and use thereof
UA108641C2 (uk) 2010-04-02 2015-05-25 Паразитицидна композиція, яка містить чотири активних агенти, та спосіб її застосування
JP6027128B2 (ja) * 2011-10-26 2016-11-16 ダウ アグロサイエンシィズ エルエルシー 有害生物防除組成物およびそれに関連した方法
AU2012340351B2 (en) 2011-11-17 2017-06-15 Boehringer Ingelheim Animal Health USA Inc. Compositions comprising an aryl pyrazole and a substituted imidazole, methods and uses thereof
CA2926095A1 (en) 2013-10-17 2015-04-23 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
JP2016539092A (ja) 2013-10-17 2016-12-15 ダウ アグロサイエンシィズ エルエルシー 有害生物防除性化合物の製造方法
US9029554B1 (en) 2013-10-17 2015-05-12 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
EP3057429A4 (en) 2013-10-17 2017-08-09 Dow AgroSciences LLC Processes for the preparation of pesticidal compounds
CA2925953C (en) 2013-10-17 2021-11-02 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
CA2925952A1 (en) 2013-10-17 2015-04-23 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
MX2016004941A (es) * 2013-10-17 2016-06-28 Dow Agrosciences Llc Proceso para la preparacion de compuestos plaguicidas.
GB201322334D0 (en) 2013-12-17 2014-01-29 Agency Science Tech & Res Maleimide derivatives as modulators of WNT pathway
BR112017000293A2 (pt) 2014-07-31 2017-10-31 Dow Agrosciences Llc processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina
JP2017523168A (ja) 2014-07-31 2017-08-17 ダウ アグロサイエンシィズ エルエルシー 3−(3−クロロ−1h−ピラゾール−1−イル)ピリジンの製造方法
US9249122B1 (en) 2014-07-31 2016-02-02 Dow Agrosciences Llc Process for the preparation of 3-(3-chloro-1H-pyrazol-1-yl)pyridine
JP2017525703A (ja) 2014-08-19 2017-09-07 ダウ アグロサイエンシィズ エルエルシー 3−(3−クロロ−1h−ピラゾール−1−イル)ピリジンの調製方法
AR098113A1 (es) 2014-09-12 2016-05-04 Dow Agrosciences Llc Proceso para la preparación de 3-(3-cloro-1h-pirazol-1-il)piridina
US10864193B2 (en) 2014-10-31 2020-12-15 Boehringer Ingelheim Animal Health USA Inc. Parasiticidal compositions comprising fipronil at high concentrations
WO2016163379A1 (ja) * 2015-04-09 2016-10-13 住友化学株式会社 オキサリルアミド化合物及びその有害節足動物防除用途
WO2016163383A1 (ja) * 2015-04-09 2016-10-13 住友化学株式会社 オキサリルアミド化合物及びその有害節足動物防除用途
CN105732505B (zh) * 2016-01-28 2018-10-12 中南民族大学 丙烯酰胺化芳基吡唑型化合物及其溶剂热一锅合成法与应用
CN105712933B (zh) * 2016-01-28 2019-01-11 中南民族大学 甲酰化芳基吡唑衍生物及其醚热合成方法和应用
CN106417329B (zh) * 2016-09-27 2019-08-27 辽宁省蚕业科学研究所 一类柞蚕饰腹寄蝇病防治化合物及使用方法
JP2020503336A (ja) 2016-12-29 2020-01-30 ダウ アグロサイエンシィズ エルエルシー 殺有害生物化合物の調製方法
CN110325036B (zh) 2016-12-29 2021-10-26 美国陶氏益农公司 用于制备杀虫化合物的方法
CN107629005A (zh) * 2017-08-22 2018-01-26 王泊理 多取代苯基吡唑衍生物及其制备方法和用途

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5556873A (en) * 1993-02-24 1996-09-17 Rhone-Poulenc Inc. Pesticidal 1-aryl-5-(substituted alkyl (thio) amido)pyrazoles
EP0811615A1 (en) * 1996-06-03 1997-12-10 Rhone-Poulenc Agrochimie 1-Aryl-5-(substituted alkyl (thio) amido) pyrazoles and their use as pesticides

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3602728A1 (de) 1985-05-17 1986-11-20 Bayer Ag, 51373 Leverkusen Schaedlingsbekaempfungsmittel auf basis von pyrazolderivaten
GB8713768D0 (en) 1987-06-12 1987-07-15 May & Baker Ltd Compositions of matter
US5232940A (en) 1985-12-20 1993-08-03 Hatton Leslie R Derivatives of N-phenylpyrazoles
GB8531485D0 (en) 1985-12-20 1986-02-05 May & Baker Ltd Compositions of matter
GB9120641D0 (en) 1991-09-27 1991-11-06 Ici Plc Heterocyclic compounds
GB9306184D0 (en) 1993-03-25 1993-05-19 Zeneca Ltd Heteroaromatic compounds
DE4343832A1 (de) 1993-12-22 1995-06-29 Bayer Ag Substituierte 1-Arylpyrazole
DE4414333A1 (de) 1994-04-25 1995-10-26 Bayer Ag Substituierte Pyridylpyrazole
US6316477B1 (en) 1996-01-30 2001-11-13 Takeda Chemical Industries, Ltd. Arylpyrazole insecticides
JP3735159B2 (ja) * 1996-06-17 2006-01-18 ローヌ−プーラン・アグロシミ 新規な農薬
GB9625045D0 (en) 1996-11-30 1997-01-22 Pfizer Ltd Parasiticidal compounds
DE19650197A1 (de) 1996-12-04 1998-06-10 Bayer Ag 3-Thiocarbamoylpyrazol-Derivate
AR021608A1 (es) 1998-12-11 2002-07-31 Merial Ltd Represion de artropodos en animales

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5556873A (en) * 1993-02-24 1996-09-17 Rhone-Poulenc Inc. Pesticidal 1-aryl-5-(substituted alkyl (thio) amido)pyrazoles
EP0811615A1 (en) * 1996-06-03 1997-12-10 Rhone-Poulenc Agrochimie 1-Aryl-5-(substituted alkyl (thio) amido) pyrazoles and their use as pesticides

Also Published As

Publication number Publication date
EP1569517A1 (en) 2005-09-07
JP4759682B2 (ja) 2011-08-31
EA011505B1 (ru) 2009-04-28
BRPI0316993B1 (pt) 2016-07-05
MXPA05005899A (es) 2005-08-29
KR20050084103A (ko) 2005-08-26
ES2436746T3 (es) 2014-01-07
BR0316993A (pt) 2005-10-25
CA2508412C (en) 2011-07-26
EP1569517B1 (en) 2013-10-02
US20060135778A1 (en) 2006-06-22
CA2508412A1 (en) 2004-06-17
AU2003288038A1 (en) 2004-06-23
US7514561B2 (en) 2009-04-07
WO2004049803A1 (en) 2004-06-17
CO5690506A2 (es) 2006-10-31
EA200500930A1 (ru) 2006-10-27
AR042255A1 (es) 2005-06-15
CN1944413A (zh) 2007-04-11
ZA200503743B (en) 2006-11-29
KR101288753B1 (ko) 2013-07-23
NZ540462A (en) 2008-03-28
CN1719974A (zh) 2006-01-11
JP2006509004A (ja) 2006-03-16

Similar Documents

Publication Publication Date Title
AU2003288038B2 (en) Pesticidal 5- (acylamino) pyrazole derivatives
AU2003221298B2 (en) 5-substituted-alkylaminopyrazole derivatives as pesticides
US7872038B2 (en) 1-phenyl and 1-pyridylpyrazole derivatives and their use as pesticides
AU2003296246B2 (en) Pesticidal sulphonylaminopyrazoles
US7517877B2 (en) 5-substituted-alkylaminopyrazole derivatives as pesticides
US7514428B2 (en) Pesticidal 1-aryl-3-amidoxime-pyrazole derivatives
EP1730115B1 (en) 5-aminoalkylpyrazole derivatives as pesticidal agents
AU2004270341B9 (en) Pesticides
EP1671967A1 (en) 1-Arylpyrazoles and their use as pesticides
AU2004270342A1 (en) Pesticidal 5-substituted-oxyalkylamino-1-arylpyrazole derivatives
HK1099746B (en) Pesticides

Legal Events

Date Code Title Description
PC1 Assignment before grant (sect. 113)

Owner name: MERIAL LTD

Free format text: FORMER APPLICANT(S): BAYER CROPSCIENCE S.A.

FGA Letters patent sealed or granted (standard patent)
PC Assignment registered

Owner name: MERIAL, INC.

Free format text: FORMER OWNER WAS: MERIAL LTD

PC Assignment registered

Owner name: BOEHRINGER INGELHEIM ANIMAL HEALTH USA INC.

Free format text: FORMER OWNER(S): MERIAL, INC.

MK14 Patent ceased section 143(a) (annual fees not paid) or expired