JP2003523364A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2003523364A5 JP2003523364A5 JP2001561027A JP2001561027A JP2003523364A5 JP 2003523364 A5 JP2003523364 A5 JP 2003523364A5 JP 2001561027 A JP2001561027 A JP 2001561027A JP 2001561027 A JP2001561027 A JP 2001561027A JP 2003523364 A5 JP2003523364 A5 JP 2003523364A5
- Authority
- JP
- Japan
- Prior art keywords
- mol
- hydrogenation
- isomer
- hplc
- hours
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10003586 | 2000-01-28 | ||
| DE10003586.8 | 2000-01-28 | ||
| PCT/EP2001/000523 WO2001055175A2 (en) | 2000-01-28 | 2001-01-18 | Process for the preparation of acetyl-amidiniophenylalanyl-cyclohexylglycyl-pyridinioalaninamides |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2003523364A JP2003523364A (ja) | 2003-08-05 |
| JP2003523364A5 true JP2003523364A5 (enExample) | 2008-02-28 |
| JP4778181B2 JP4778181B2 (ja) | 2011-09-21 |
Family
ID=7628946
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001561027A Expired - Fee Related JP4778181B2 (ja) | 2000-01-28 | 2001-01-18 | アセチル−アミジニオフェニルアラニル−シクロヘキシルグリシル−ピリジニオアラニンアミドの製造方法 |
Country Status (29)
| Country | Link |
|---|---|
| US (2) | US20010031858A1 (enExample) |
| EP (1) | EP1254159B9 (enExample) |
| JP (1) | JP4778181B2 (enExample) |
| KR (1) | KR100758141B1 (enExample) |
| CN (1) | CN1176104C (enExample) |
| AR (1) | AR027246A1 (enExample) |
| AT (1) | ATE325810T1 (enExample) |
| AU (1) | AU779722B2 (enExample) |
| BR (1) | BR0107804A (enExample) |
| CA (1) | CA2398497C (enExample) |
| CZ (1) | CZ20022583A3 (enExample) |
| DE (1) | DE60119491T2 (enExample) |
| DK (1) | DK1254159T3 (enExample) |
| EE (1) | EE200200410A (enExample) |
| ES (1) | ES2262632T3 (enExample) |
| HR (1) | HRP20020631A2 (enExample) |
| HU (1) | HUP0301986A2 (enExample) |
| IL (2) | IL150897A0 (enExample) |
| MX (1) | MXPA02006762A (enExample) |
| NO (1) | NO20023577L (enExample) |
| NZ (1) | NZ520427A (enExample) |
| PL (1) | PL356801A1 (enExample) |
| PT (1) | PT1254159E (enExample) |
| RU (1) | RU2250212C2 (enExample) |
| SK (1) | SK10842002A3 (enExample) |
| TW (1) | TWI236481B (enExample) |
| WO (1) | WO2001055175A2 (enExample) |
| YU (1) | YU51202A (enExample) |
| ZA (1) | ZA200205990B (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH695999A5 (de) | 2002-02-28 | 2006-11-15 | Wilex Ag | Verfahren zur Herstellung von 3- Amidinophenylalanin-Derivaten. |
| WO2007065691A2 (en) * | 2005-12-07 | 2007-06-14 | Technische Universität München | Small peptidic and peptido-mimetic affinity ligands for factor viii and factor viii-like proteins |
| CN101774942B (zh) * | 2010-01-27 | 2012-08-22 | 宁波武盛化学有限公司 | 制备n-乙酰基-dl-环己基甘氨酸的方法 |
| US8558023B2 (en) * | 2010-04-20 | 2013-10-15 | Chiral Quest, Inc. | Enantioselective process for cycloalkenyl β-substituted alanines |
| EP2646150A4 (en) * | 2010-11-29 | 2014-10-08 | Takasago Perfumery Co Ltd | CATALYST FOR ASYMMETRIC HYDROGENATION AND METHOD FOR PRODUCING AN OPTICALLY ACTIVE CARBONYL COMPOUND THEREWITH |
| CN115068469B (zh) * | 2022-07-08 | 2024-02-27 | 深圳市小分子新药创新中心有限公司 | Tigit抑制剂及其应用 |
| CN115612702A (zh) * | 2022-10-09 | 2023-01-17 | 深圳市茵诺圣生物科技有限公司 | L-丙氨酸类非天然氨基酸3-(3-吡啶基)-l-丙氨酸的合成方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2916711A1 (de) | 1979-04-25 | 1980-11-06 | Behringwerke Ag | Blutgerinnungsfaktoren und verfahren zu ihrer herstellung |
| US4440679A (en) * | 1980-03-05 | 1984-04-03 | Cutter Laboratories, Inc. | Pasteurized therapeutically active protein compositions |
| US4623717A (en) * | 1980-03-05 | 1986-11-18 | Miles Laboratories, Inc. | Pasteurized therapeutically active protein compositions |
| SE9301916D0 (sv) * | 1993-06-03 | 1993-06-03 | Ab Astra | New peptides derivatives |
| US5866685A (en) * | 1993-10-15 | 1999-02-02 | Rhone-Poulenc Rorer Pharmaceuticals Inc. | Antithrombotic azacycloalkylalkanoyl peptides and pseudopeptides |
| ZA953361B (en) * | 1994-04-26 | 1996-01-12 | Selectide Corp | Factor Xa inhibitors |
| US5849510A (en) | 1994-04-26 | 1998-12-15 | Selectide Corporation | Factor Xa inhibitors |
| SK281432B6 (sk) * | 1995-12-20 | 2001-03-12 | Hoechst Marion Roussel, Inc. | Spôsob prípravy n-acetyl-(l)-4-kyanofenylalanínu ac-(l)-phe(4- -cn)-oh a n-acetyl-(l)-p-amidinofenylalanín-cyklohexylglycín- -beta-(3-n-metylpyridínium)-alanínu ac-(l)-paph-chg-palme(3)-nh2 |
| DE19856443A1 (de) | 1998-12-08 | 2000-06-21 | Centeon Pharma Gmbh | Stabilisiertes Antithrombin III-Präparat |
-
2001
- 2001-01-18 HU HU0301986A patent/HUP0301986A2/hu unknown
- 2001-01-18 DE DE60119491T patent/DE60119491T2/de not_active Expired - Lifetime
- 2001-01-18 NZ NZ520427A patent/NZ520427A/en unknown
- 2001-01-18 RU RU2002123046/04A patent/RU2250212C2/ru not_active IP Right Cessation
- 2001-01-18 CN CNB018041523A patent/CN1176104C/zh not_active Expired - Fee Related
- 2001-01-18 EP EP01911497A patent/EP1254159B9/en not_active Expired - Lifetime
- 2001-01-18 KR KR1020027009583A patent/KR100758141B1/ko not_active Expired - Fee Related
- 2001-01-18 AT AT01911497T patent/ATE325810T1/de active
- 2001-01-18 EE EEP200200410A patent/EE200200410A/xx unknown
- 2001-01-18 MX MXPA02006762A patent/MXPA02006762A/es active IP Right Grant
- 2001-01-18 PL PL01356801A patent/PL356801A1/xx unknown
- 2001-01-18 SK SK1084-2002A patent/SK10842002A3/sk unknown
- 2001-01-18 AU AU40516/01A patent/AU779722B2/en not_active Ceased
- 2001-01-18 CA CA2398497A patent/CA2398497C/en not_active Expired - Fee Related
- 2001-01-18 ES ES01911497T patent/ES2262632T3/es not_active Expired - Lifetime
- 2001-01-18 JP JP2001561027A patent/JP4778181B2/ja not_active Expired - Fee Related
- 2001-01-18 AR ARP010100225A patent/AR027246A1/es unknown
- 2001-01-18 HR HRP20020631 patent/HRP20020631A2/hr not_active Application Discontinuation
- 2001-01-18 BR BR0107804-6A patent/BR0107804A/pt not_active Application Discontinuation
- 2001-01-18 WO PCT/EP2001/000523 patent/WO2001055175A2/en not_active Ceased
- 2001-01-18 IL IL15089701A patent/IL150897A0/xx active IP Right Grant
- 2001-01-18 YU YU51202A patent/YU51202A/sh unknown
- 2001-01-18 PT PT01911497T patent/PT1254159E/pt unknown
- 2001-01-18 CZ CZ20022583A patent/CZ20022583A3/cs unknown
- 2001-01-18 DK DK01911497T patent/DK1254159T3/da active
- 2001-01-26 US US09/769,487 patent/US20010031858A1/en not_active Abandoned
- 2001-03-07 TW TW090101207A patent/TWI236481B/zh not_active IP Right Cessation
-
2002
- 2002-07-24 IL IL150897A patent/IL150897A/en not_active IP Right Cessation
- 2002-07-26 ZA ZA200205990A patent/ZA200205990B/en unknown
- 2002-07-26 NO NO20023577A patent/NO20023577L/no unknown
-
2004
- 2004-06-17 US US10/869,076 patent/US7084250B2/en not_active Expired - Lifetime
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| TWI225476B (en) | Novel process of preparing tolterodine and analogues thereof, and novel intermediates prepared therein | |
| HK1079790A1 (zh) | 10，11-二氢-10-羟基-5h-二苯并b，f氮杂卓-5-羧酰胺的对映体及其新晶形两者制备的对映选择性方法 | |
| JP2005500987A5 (enExample) | ||
| MXPA03011972A (es) | Arilaminas para tratamiento de condiciones asociadas con gsk-3. | |
| JP2006521826A5 (enExample) | ||
| SI8310672A8 (en) | Process for the production of cis-4-fenil-1,2,3,4-tetrahydro-1-naphthylamine derivates. | |
| MXPA04000756A (es) | Nuevos compuestos. | |
| CN1531551A (zh) | 一种生产促胰岛素分泌肽glp-1(7-36)及glp-1类似物的方法 | |
| DE60202958D1 (de) | Stabiles polymorph von flibanserin, industrielles verfahren zu dessen herstellung und dessen verwendung zur herstellung von medikamenten | |
| WO2002065979A3 (en) | (diazolo-pyridinyl)-pyrimidines for use in treatment of cns disorders and diabetes | |
| HU228815B1 (en) | Asymmetric synthesis of pregabalin | |
| WO2004060277A3 (en) | Process for purification of plasmid dna | |
| JP2004532624A5 (enExample) | ||
| WO2004063185A8 (en) | Thiophene carboxamides as inhibitors of the enzyme ikk-2 | |
| WO2005014608A3 (en) | Process for preparing maltitol enriched products | |
| JP2000351758A (ja) | キラルテトラロンからのセルトラリンの製造法 | |
| IL162171A0 (en) | Crystalline venlafaxine base and novel polymorphs of venlafaxine hydrochloride, processes for preparing thereof | |
| NO20042681L (no) | Ny krystallinsk polymorf av venlafaxine-hydroklorid og fremgangsmater for fremstilling derav | |
| NO20061310L (no) | Nye forbindelser og deres anvendelse i medisin; fremgangsmate for deres fremstilling og farmasoytiske sammensetninger som inneholder dem | |
| WO2005023791A3 (en) | Process for the production of mycophenolate mofetil | |
| NO20061404L (no) | Renseprosess | |
| PL372933A1 (en) | Methylthiophene carboxanilides | |
| MXPA02012053A (es) | Procedimiento para la obtencion de 3,3,5-trimetilciclohexanol. | |
| CA2534194A1 (en) | Indoline-sulfanilic acid amides used as ppar delta modulators | |
| Yu et al. | Mono-chlorination of electron-rich arylalkyl-and heteroarylalkyl-amines and amino acids using sulfuryl chloride |