DK1254159T3 - Fremgangsmåde til fremstilling af acetylamidiniophenylalanylcyclohexylglycylpyridylalaninamider - Google Patents
Fremgangsmåde til fremstilling af acetylamidiniophenylalanylcyclohexylglycylpyridylalaninamiderInfo
- Publication number
- DK1254159T3 DK1254159T3 DK01911497T DK01911497T DK1254159T3 DK 1254159 T3 DK1254159 T3 DK 1254159T3 DK 01911497 T DK01911497 T DK 01911497T DK 01911497 T DK01911497 T DK 01911497T DK 1254159 T3 DK1254159 T3 DK 1254159T3
- Authority
- DK
- Denmark
- Prior art keywords
- cyclohexylglycylpyridylalanine
- acetylamidiniophenylalanyl
- amides
- preparation
- cyclohexylglycylpyridylalanine amides
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10003586 | 2000-01-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1254159T3 true DK1254159T3 (da) | 2006-09-11 |
Family
ID=7628946
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK01911497T DK1254159T3 (da) | 2000-01-28 | 2001-01-18 | Fremgangsmåde til fremstilling af acetylamidiniophenylalanylcyclohexylglycylpyridylalaninamider |
Country Status (30)
| Country | Link |
|---|---|
| US (2) | US20010031858A1 (da) |
| EP (1) | EP1254159B9 (da) |
| JP (1) | JP4778181B2 (da) |
| KR (1) | KR100758141B1 (da) |
| CN (1) | CN1176104C (da) |
| AR (1) | AR027246A1 (da) |
| AT (1) | ATE325810T1 (da) |
| AU (1) | AU779722B2 (da) |
| BR (1) | BR0107804A (da) |
| CA (1) | CA2398497C (da) |
| CZ (1) | CZ20022583A3 (da) |
| DE (1) | DE60119491T2 (da) |
| DK (1) | DK1254159T3 (da) |
| EE (1) | EE200200410A (da) |
| ES (1) | ES2262632T3 (da) |
| HK (1) | HK1051866A1 (da) |
| HR (1) | HRP20020631A2 (da) |
| HU (1) | HUP0301986A2 (da) |
| IL (2) | IL150897A0 (da) |
| MX (1) | MXPA02006762A (da) |
| NO (1) | NO20023577L (da) |
| NZ (1) | NZ520427A (da) |
| PL (1) | PL356801A1 (da) |
| PT (1) | PT1254159E (da) |
| RU (1) | RU2250212C2 (da) |
| SK (1) | SK10842002A3 (da) |
| TW (1) | TWI236481B (da) |
| WO (1) | WO2001055175A2 (da) |
| YU (1) | YU51202A (da) |
| ZA (1) | ZA200205990B (da) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH695999A5 (de) | 2002-02-28 | 2006-11-15 | Wilex Ag | Verfahren zur Herstellung von 3- Amidinophenylalanin-Derivaten. |
| JP2009518345A (ja) * | 2005-12-07 | 2009-05-07 | テフニーシェ ウニヴェルジテート ミュンヘン | 因子ｖｉｉｉおよび因子ｖｉｉｉ様タンパク質に対する小型ペプチドおよびペプチド模倣物の親和性リガンド |
| CN101774942B (zh) * | 2010-01-27 | 2012-08-22 | 宁波武盛化学有限公司 | 制备n-乙酰基-dl-环己基甘氨酸的方法 |
| ES2686298T3 (es) * | 2010-04-20 | 2018-10-17 | Chiral Quest, Inc. | Procedimiento enantioselectivo para alaninas beta sustituidas con cicloalquenilo |
| EP2646150A4 (en) * | 2010-11-29 | 2014-10-08 | Takasago Perfumery Co Ltd | CATALYST FOR ASYMMETRIC HYDROGENATION AND METHOD FOR PRODUCING AN OPTICALLY ACTIVE CARBONYL COMPOUND THEREWITH |
| CN115068469B (zh) * | 2022-07-08 | 2024-02-27 | 深圳市小分子新药创新中心有限公司 | Tigit抑制剂及其应用 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2916711A1 (de) * | 1979-04-25 | 1980-11-06 | Behringwerke Ag | Blutgerinnungsfaktoren und verfahren zu ihrer herstellung |
| US4623717A (en) * | 1980-03-05 | 1986-11-18 | Miles Laboratories, Inc. | Pasteurized therapeutically active protein compositions |
| US4440679A (en) * | 1980-03-05 | 1984-04-03 | Cutter Laboratories, Inc. | Pasteurized therapeutically active protein compositions |
| US5849510A (en) | 1994-04-26 | 1998-12-15 | Selectide Corporation | Factor Xa inhibitors |
| CN1181091C (zh) * | 1994-04-26 | 2004-12-22 | 西莱克泰德公司 | 因子Xa抑制剂 |
| EP0868526B1 (en) * | 1995-12-20 | 2002-08-14 | Aventis Pharmaceuticals Inc. | PROCESS FOR PREPARING N-ACETYL(L)-4-CYANOPHENYLALANINE Ac-(L)-Phe(4-CN)-OH AND N-ACETYL-(L)-p-AMIDINOPHENYLALANINE-CYCLOHEXYLGLYCINE-BETA-(3-N-METHYLPYRIDINIUM)-ALANINE Ac-(L)-pAph-Chg-PalMe(3)-NH2 |
| DE19856443A1 (de) | 1998-12-08 | 2000-06-21 | Centeon Pharma Gmbh | Stabilisiertes Antithrombin III-Präparat |
-
2001
- 2001-01-18 DE DE60119491T patent/DE60119491T2/de not_active Expired - Lifetime
- 2001-01-18 CZ CZ20022583A patent/CZ20022583A3/cs unknown
- 2001-01-18 HU HU0301986A patent/HUP0301986A2/hu unknown
- 2001-01-18 RU RU2002123046/04A patent/RU2250212C2/ru not_active IP Right Cessation
- 2001-01-18 YU YU51202A patent/YU51202A/sh unknown
- 2001-01-18 EP EP01911497A patent/EP1254159B9/en not_active Expired - Lifetime
- 2001-01-18 NZ NZ520427A patent/NZ520427A/en unknown
- 2001-01-18 IL IL15089701A patent/IL150897A0/xx active IP Right Grant
- 2001-01-18 BR BR0107804-6A patent/BR0107804A/pt not_active Application Discontinuation
- 2001-01-18 CN CNB018041523A patent/CN1176104C/zh not_active Expired - Fee Related
- 2001-01-18 AR ARP010100225A patent/AR027246A1/es unknown
- 2001-01-18 KR KR1020027009583A patent/KR100758141B1/ko not_active IP Right Cessation
- 2001-01-18 PL PL01356801A patent/PL356801A1/xx unknown
- 2001-01-18 SK SK1084-2002A patent/SK10842002A3/sk unknown
- 2001-01-18 WO PCT/EP2001/000523 patent/WO2001055175A2/en not_active Application Discontinuation
- 2001-01-18 JP JP2001561027A patent/JP4778181B2/ja not_active Expired - Fee Related
- 2001-01-18 EE EEP200200410A patent/EE200200410A/xx unknown
- 2001-01-18 PT PT01911497T patent/PT1254159E/pt unknown
- 2001-01-18 ES ES01911497T patent/ES2262632T3/es not_active Expired - Lifetime
- 2001-01-18 DK DK01911497T patent/DK1254159T3/da active
- 2001-01-18 MX MXPA02006762A patent/MXPA02006762A/es active IP Right Grant
- 2001-01-18 AT AT01911497T patent/ATE325810T1/de active
- 2001-01-18 AU AU40516/01A patent/AU779722B2/en not_active Ceased
- 2001-01-18 CA CA2398497A patent/CA2398497C/en not_active Expired - Fee Related
- 2001-01-26 US US09/769,487 patent/US20010031858A1/en not_active Abandoned
- 2001-03-07 TW TW090101207A patent/TWI236481B/zh not_active IP Right Cessation
-
2002
- 2002-07-24 IL IL150897A patent/IL150897A/en not_active IP Right Cessation
- 2002-07-25 HR HRP20020631 patent/HRP20020631A2/hr not_active Application Discontinuation
- 2002-07-26 ZA ZA200205990A patent/ZA200205990B/en unknown
- 2002-07-26 NO NO20023577A patent/NO20023577L/no unknown
-
2003
- 2003-06-11 HK HK03104146A patent/HK1051866A1/xx not_active IP Right Cessation
-
2004
- 2004-06-17 US US10/869,076 patent/US7084250B2/en not_active Expired - Lifetime
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