EE200200410A - Meetod atsetüülamidiniofenüülalanüültsükloheksüülglütsüülpüridinioalaniinamiidide valmistamiseks ning selleks vajalikud lähte- ja vaheühendid - Google Patents
Meetod atsetüülamidiniofenüülalanüültsükloheksüülglütsüülpüridinioalaniinamiidide valmistamiseks ning selleks vajalikud lähte- ja vaheühendidInfo
- Publication number
- EE200200410A EE200200410A EEP200200410A EEP200200410A EE200200410A EE 200200410 A EE200200410 A EE 200200410A EE P200200410 A EEP200200410 A EE P200200410A EE P200200410 A EEP200200410 A EE P200200410A EE 200200410 A EE200200410 A EE 200200410A
- Authority
- EE
- Estonia
- Prior art keywords
- starting
- preparation
- intermediate compounds
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Diabetes (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Hematology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Investigating Or Analysing Biological Materials (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10003586 | 2000-01-28 | ||
| PCT/EP2001/000523 WO2001055175A2 (en) | 2000-01-28 | 2001-01-18 | Process for the preparation of acetyl-amidiniophenylalanyl-cyclohexylglycyl-pyridinioalaninamides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| EE200200410A true EE200200410A (et) | 2003-12-15 |
Family
ID=7628946
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EEP200200410A EE200200410A (et) | 2000-01-28 | 2001-01-18 | Meetod atsetüülamidiniofenüülalanüültsükloheksüülglütsüülpüridinioalaniinamiidide valmistamiseks ning selleks vajalikud lähte- ja vaheühendid |
Country Status (30)
| Country | Link |
|---|---|
| US (2) | US20010031858A1 (et) |
| EP (1) | EP1254159B9 (et) |
| JP (1) | JP4778181B2 (et) |
| KR (1) | KR100758141B1 (et) |
| CN (1) | CN1176104C (et) |
| AR (1) | AR027246A1 (et) |
| AT (1) | ATE325810T1 (et) |
| AU (1) | AU779722B2 (et) |
| BR (1) | BR0107804A (et) |
| CA (1) | CA2398497C (et) |
| CZ (1) | CZ20022583A3 (et) |
| DE (1) | DE60119491T2 (et) |
| DK (1) | DK1254159T3 (et) |
| EE (1) | EE200200410A (et) |
| ES (1) | ES2262632T3 (et) |
| HK (1) | HK1051866A1 (et) |
| HR (1) | HRP20020631A2 (et) |
| HU (1) | HUP0301986A2 (et) |
| IL (2) | IL150897A0 (et) |
| MX (1) | MXPA02006762A (et) |
| NO (1) | NO20023577L (et) |
| NZ (1) | NZ520427A (et) |
| PL (1) | PL356801A1 (et) |
| PT (1) | PT1254159E (et) |
| RU (1) | RU2250212C2 (et) |
| SK (1) | SK10842002A3 (et) |
| TW (1) | TWI236481B (et) |
| WO (1) | WO2001055175A2 (et) |
| YU (1) | YU51202A (et) |
| ZA (1) | ZA200205990B (et) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH695999A5 (de) | 2002-02-28 | 2006-11-15 | Wilex Ag | Verfahren zur Herstellung von 3- Amidinophenylalanin-Derivaten. |
| JP2009518345A (ja) * | 2005-12-07 | 2009-05-07 | テフニーシェ ウニヴェルジテート ミュンヘン | 因子ｖｉｉｉおよび因子ｖｉｉｉ様タンパク質に対する小型ペプチドおよびペプチド模倣物の親和性リガンド |
| CN101774942B (zh) * | 2010-01-27 | 2012-08-22 | 宁波武盛化学有限公司 | 制备n-乙酰基-dl-环己基甘氨酸的方法 |
| CN102984945B (zh) * | 2010-04-20 | 2014-08-20 | 凯瑞斯德生化(苏州)有限公司 | 一种环烯基在β位取代的丙氨酸的不对称合成方法 |
| EP2646150A4 (en) * | 2010-11-29 | 2014-10-08 | Takasago Perfumery Co Ltd | CATALYST FOR ASYMMETRIC HYDROGENATION AND METHOD FOR PRODUCING AN OPTICALLY ACTIVE CARBONYL COMPOUND THEREWITH |
| CN115068469B (zh) * | 2022-07-08 | 2024-02-27 | 深圳市小分子新药创新中心有限公司 | Tigit抑制剂及其应用 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2916711A1 (de) | 1979-04-25 | 1980-11-06 | Behringwerke Ag | Blutgerinnungsfaktoren und verfahren zu ihrer herstellung |
| US4440679A (en) | 1980-03-05 | 1984-04-03 | Cutter Laboratories, Inc. | Pasteurized therapeutically active protein compositions |
| US4623717A (en) | 1980-03-05 | 1986-11-18 | Miles Laboratories, Inc. | Pasteurized therapeutically active protein compositions |
| ZA953361B (en) * | 1994-04-26 | 1996-01-12 | Selectide Corp | Factor Xa inhibitors |
| US5849510A (en) | 1994-04-26 | 1998-12-15 | Selectide Corporation | Factor Xa inhibitors |
| RU2170764C2 (ru) * | 1995-12-20 | 2001-07-20 | Авентис Фармасьютикалз Инк. | НОВЫЙ СПОСОБ ПОЛУЧЕНИЯ N-АЦЕТИЛ-(L)-4-ЦИАНОФЕНИЛАЛАНИНА АС-(L)-PHE(4-CN)-OH И N-АЦЕТИЛ-(L)-N-АМИДИНОФЕНИЛАЛАНИН-ЦИКЛОГЕКСИЛ-ГЛИЦИН-β-(3-N-МЕТИЛПИРИДИН ИЯ)-АЛАНИНА АС-(L)-PАPH-СHG-РAL МE(3)-NH2 |
| DE19856443A1 (de) | 1998-12-08 | 2000-06-21 | Centeon Pharma Gmbh | Stabilisiertes Antithrombin III-Präparat |
-
2001
- 2001-01-18 DK DK01911497T patent/DK1254159T3/da active
- 2001-01-18 MX MXPA02006762A patent/MXPA02006762A/es active IP Right Grant
- 2001-01-18 SK SK1084-2002A patent/SK10842002A3/sk unknown
- 2001-01-18 EE EEP200200410A patent/EE200200410A/et unknown
- 2001-01-18 PL PL01356801A patent/PL356801A1/xx unknown
- 2001-01-18 CA CA2398497A patent/CA2398497C/en not_active Expired - Fee Related
- 2001-01-18 AT AT01911497T patent/ATE325810T1/de active
- 2001-01-18 PT PT01911497T patent/PT1254159E/pt unknown
- 2001-01-18 JP JP2001561027A patent/JP4778181B2/ja not_active Expired - Fee Related
- 2001-01-18 YU YU51202A patent/YU51202A/sh unknown
- 2001-01-18 AU AU40516/01A patent/AU779722B2/en not_active Ceased
- 2001-01-18 ES ES01911497T patent/ES2262632T3/es not_active Expired - Lifetime
- 2001-01-18 IL IL15089701A patent/IL150897A0/xx active IP Right Grant
- 2001-01-18 RU RU2002123046/04A patent/RU2250212C2/ru not_active IP Right Cessation
- 2001-01-18 NZ NZ520427A patent/NZ520427A/en unknown
- 2001-01-18 CZ CZ20022583A patent/CZ20022583A3/cs unknown
- 2001-01-18 CN CNB018041523A patent/CN1176104C/zh not_active Expired - Fee Related
- 2001-01-18 WO PCT/EP2001/000523 patent/WO2001055175A2/en not_active Application Discontinuation
- 2001-01-18 HU HU0301986A patent/HUP0301986A2/hu unknown
- 2001-01-18 BR BR0107804-6A patent/BR0107804A/pt not_active Application Discontinuation
- 2001-01-18 AR ARP010100225A patent/AR027246A1/es unknown
- 2001-01-18 KR KR1020027009583A patent/KR100758141B1/ko not_active IP Right Cessation
- 2001-01-18 DE DE60119491T patent/DE60119491T2/de not_active Expired - Lifetime
- 2001-01-18 EP EP01911497A patent/EP1254159B9/en not_active Expired - Lifetime
- 2001-01-26 US US09/769,487 patent/US20010031858A1/en not_active Abandoned
- 2001-03-07 TW TW090101207A patent/TWI236481B/zh not_active IP Right Cessation
-
2002
- 2002-07-24 IL IL150897A patent/IL150897A/en not_active IP Right Cessation
- 2002-07-25 HR HRP20020631 patent/HRP20020631A2/hr not_active Application Discontinuation
- 2002-07-26 ZA ZA200205990A patent/ZA200205990B/en unknown
- 2002-07-26 NO NO20023577A patent/NO20023577L/no unknown
-
2003
- 2003-06-11 HK HK03104146A patent/HK1051866A1/xx not_active IP Right Cessation
-
2004
- 2004-06-17 US US10/869,076 patent/US7084250B2/en not_active Expired - Lifetime
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NO20030012L (no) | Fremgangsmåte for fremstilling av substituerte oktanoylamider | |
| EE200200704A (et) | Uued ühendid, meetod nende valmistamiseks ning nende kasutamine | |
| EE200200470A (et) | Uued ühendid, meetod nende valmistamiseks ning nende kasutamine | |
| CY2007029I2 (el) | Μεθοδος για την παρασκευη υποκατεστημενων οκτανοϋλ-αμιδιων | |
| EE05223B1 (et) | Triasoloprimidiini hendid, meetod nende valmistamiseks ning nende kasutamine | |
| FI20011578A0 (fi) | Menetelmä puhtaan sitalopraamin valmistamiseksi | |
| FI20011621A (fi) | Menetelmä sitalopraamin valmistamiseksi | |
| NO20023928L (no) | Fremgangsmåte ved fremstillingen av citalopram | |
| NO20024007L (no) | Fremgangsmåte ved fremstillingen av citalopram | |
| EE200100574A (et) | Uued ühendid, nende valmistamise meetod ning kasutamine | |
| DE60121150D1 (de) | Verfahren zur herstellung von ansamitocin | |
| EE05308B1 (et) | Sulfoonamiid-asendatud imidasotriasinoonide valmistamismeetod | |
| FI20011889A (fi) | Menetelmä ksylitolin valmistamiseksi | |
| NO20024180L (no) | Fremgangsmåte ved fremstillingen av citalopram | |
| EE200200697A (et) | Uued ühendid, meetod nende valmistamiseks ning nende kasutamine | |
| NO20025423L (no) | Fremgangsmate for fremstilling av Citalopram | |
| NO20024213L (no) | FremgangsmÕte ved fremstilling av citalopram | |
| AU8311901A (en) | Polymorphs of zaleplon and methods for the preparation thereof | |
| EE200100573A (et) | Uued ühendid, nende valmistamise meetod ning kasutamine | |
| EE200200410A (et) | Meetod atsetüülamidiniofenüülalanüültsükloheksüülglütsüülpüridinioalaniinamiidide valmistamiseks ning selleks vajalikud lähte- ja vaheühendid | |
| NO20021118D0 (no) | Fremgangsmåte for fremstilling av citalopram | |
| NO20031927L (no) | Forbedret fremgangsmåte for fremstilling av gabapentinmellomprodukt | |
| NO20030515L (no) | Fremgangsmåte for fremstilling av dinapsolin | |
| NO20024214D0 (no) | Fremgangsmåte ved fremstilling av citalopram | |
| NO20023702L (no) | Fremgangsmåte for fremstilling av 5-arylnikotinaldehyder |