IL98482A - 1,6-dihydro-5- (2,5-disubstituted phenyl)-7h-pyrazolo-[4,3-d] pyrimidin-7-ones and pharmaceutical compositions containing them - Google Patents

1,6-dihydro-5- (2,5-disubstituted phenyl)-7h-pyrazolo-[4,3-d] pyrimidin-7-ones and pharmaceutical compositions containing them

Info

Publication number
IL98482A
IL98482A IL9848291A IL9848291A IL98482A IL 98482 A IL98482 A IL 98482A IL 9848291 A IL9848291 A IL 9848291A IL 9848291 A IL9848291 A IL 9848291A IL 98482 A IL98482 A IL 98482A
Authority
IL
Israel
Prior art keywords
alkyl
methyl
dihydro
pyrazolo
propyl
Prior art date
Application number
IL9848291A
Other languages
English (en)
Other versions
IL98482A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10677918&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL98482(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of IL98482A0 publication Critical patent/IL98482A0/xx
Publication of IL98482A publication Critical patent/IL98482A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • G—PHYSICS
    • G05—CONTROLLING; REGULATING
    • G05B—CONTROL OR REGULATING SYSTEMS IN GENERAL; FUNCTIONAL ELEMENTS OF SUCH SYSTEMS; MONITORING OR TESTING ARRANGEMENTS FOR SUCH SYSTEMS OR ELEMENTS
    • G05B2219/00—Program-control systems
    • G05B2219/30—Nc systems
    • G05B2219/36—Nc in input of data, input key till input tape
    • G05B2219/36395—Load local computer program from host, data transfer ram to rom, BTR

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Cardiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
IL9848291A 1990-06-20 1991-06-13 1,6-dihydro-5- (2,5-disubstituted phenyl)-7h-pyrazolo-[4,3-d] pyrimidin-7-ones and pharmaceutical compositions containing them IL98482A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB909013750A GB9013750D0 (en) 1990-06-20 1990-06-20 Therapeutic agents

Publications (2)

Publication Number Publication Date
IL98482A0 IL98482A0 (en) 1992-07-15
IL98482A true IL98482A (en) 1995-11-27

Family

ID=10677918

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9848291A IL98482A (en) 1990-06-20 1991-06-13 1,6-dihydro-5- (2,5-disubstituted phenyl)-7h-pyrazolo-[4,3-d] pyrimidin-7-ones and pharmaceutical compositions containing them

Country Status (31)

Country Link
EP (1) EP0463756B1 (pt)
JP (1) JPH07121945B2 (pt)
KR (1) KR940006628B1 (pt)
CN (1) CN1028758C (pt)
AT (1) ATE121403T1 (pt)
AU (1) AU626757B2 (pt)
BR (1) BR9102560A (pt)
CA (1) CA2044748C (pt)
CY (2) CY1971A (pt)
CZ (1) CZ279289B6 (pt)
DE (2) DE19975015I2 (pt)
DK (1) DK0463756T3 (pt)
EG (1) EG19651A (pt)
ES (1) ES2071919T4 (pt)
FI (1) FI95132C (pt)
GB (1) GB9013750D0 (pt)
HK (1) HK219496A (pt)
HU (1) HU218945B (pt)
IE (1) IE66040B1 (pt)
IL (1) IL98482A (pt)
LU (1) LU90360I2 (pt)
MY (1) MY107176A (pt)
NL (1) NL990005I2 (pt)
NO (2) NO178029C (pt)
NZ (1) NZ238586A (pt)
PL (1) PL166490B1 (pt)
PT (1) PT98011B (pt)
RU (2) RU2114114C1 (pt)
TW (1) TW222633B (pt)
YU (1) YU47962B (pt)
ZA (1) ZA914707B (pt)

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