IL156306A0 - Pyrimidineamines as angiogenesis modulators - Google Patents

Pyrimidineamines as angiogenesis modulators

Info

Publication number
IL156306A0
IL156306A0 IL15630601A IL15630601A IL156306A0 IL 156306 A0 IL156306 A0 IL 156306A0 IL 15630601 A IL15630601 A IL 15630601A IL 15630601 A IL15630601 A IL 15630601A IL 156306 A0 IL156306 A0 IL 156306A0
Authority
IL
Israel
Prior art keywords
pyrimidineamines
angiogenesis modulators
pyrimidine derivatives
angiogenesis
modulators
Prior art date
Application number
IL15630601A
Other languages
English (en)
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26946028&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL156306(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of IL156306A0 publication Critical patent/IL156306A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/10—Ophthalmic agents for accommodation disorders, e.g. myopia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08—Radicals containing only hydrogen and carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
IL15630601A 2000-12-21 2001-12-19 Pyrimidineamines as angiogenesis modulators IL156306A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25752600P 2000-12-21 2000-12-21
US26240301P 2001-01-16 2001-01-16
PCT/US2001/049367 WO2002059110A1 (fr) 2000-12-21 2001-12-19 Composes chimiques

Publications (1)

Publication Number Publication Date
IL156306A0 true IL156306A0 (en) 2004-01-04

Family

ID=26946028

Family Applications (2)

Application Number Title Priority Date Filing Date
IL15630601A IL156306A0 (en) 2000-12-21 2001-12-19 Pyrimidineamines as angiogenesis modulators
IL156306A IL156306A (en) 2000-12-21 2003-06-04 5 - ({4 - [(2,3 - DIMETHYL l - 2H - INDAZOL - 6 - YL)(METHYL) AMINO] PYRIMIDIN - 2 - YL} AMINO) - 2 -

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL156306A IL156306A (en) 2000-12-21 2003-06-04 5 - ({4 - [(2,3 - DIMETHYL l - 2H - INDAZOL - 6 - YL)(METHYL) AMINO] PYRIMIDIN - 2 - YL} AMINO) - 2 -

Country Status (28)

Country Link
US (6) US7105530B2 (fr)
EP (2) EP1343782B1 (fr)
JP (1) JP4253188B2 (fr)
KR (1) KR100847169B1 (fr)
CN (1) CN1307173C (fr)
AT (1) ATE430742T1 (fr)
AU (1) AU2002246723B2 (fr)
BE (1) BE2010C030I2 (fr)
BR (1) BR0116452A (fr)
CA (1) CA2432000C (fr)
CY (2) CY1109160T1 (fr)
CZ (1) CZ304059B6 (fr)
DE (2) DE60138645D1 (fr)
DK (2) DK2311825T3 (fr)
ES (2) ES2324981T3 (fr)
FR (1) FR10C0037I2 (fr)
HK (2) HK1059926A1 (fr)
HU (2) HU230574B1 (fr)
IL (2) IL156306A0 (fr)
LU (1) LU91710I2 (fr)
MX (1) MXPA03005696A (fr)
NO (3) NO325987B1 (fr)
NZ (1) NZ526542A (fr)
PL (1) PL214667B1 (fr)
PT (2) PT2311825E (fr)
SI (2) SI2311825T1 (fr)
WO (1) WO2002059110A1 (fr)
ZA (1) ZA200304482B (fr)

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CA2432000C (fr) 2011-03-15
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CZ20031748A3 (en) 2004-04-14
LU91710I2 (fr) 2010-09-21
DK1343782T3 (da) 2009-08-24
NO2010020I1 (no) 2010-11-22
CN1307173C (zh) 2007-03-28
ATE430742T1 (de) 2009-05-15
EP2311825A1 (fr) 2011-04-20
BE2010C030I2 (fr) 2021-06-17
CY2010014I2 (el) 2012-01-25
CN1549813A (zh) 2004-11-24
US20040242578A1 (en) 2004-12-02
CA2432000A1 (fr) 2002-08-01
FR10C0037I2 (fr) 2011-04-29
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NZ526542A (en) 2005-01-28
EP1343782B1 (fr) 2009-05-06
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JP2004517925A (ja) 2004-06-17
SI2311825T1 (sl) 2016-02-29
PT2311825E (pt) 2016-01-22
EP1343782A1 (fr) 2003-09-17
US7858626B2 (en) 2010-12-28
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US20100105712A1 (en) 2010-04-29
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US8114885B2 (en) 2012-02-14
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PL214667B1 (pl) 2013-08-30
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US20070270427A1 (en) 2007-11-22
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