IL145430A0 - N-cyanomethyl amides, processes for the preparation thereof and pharmaceutical compositions containing the same - Google Patents

N-cyanomethyl amides, processes for the preparation thereof and pharmaceutical compositions containing the same

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Publication number
IL145430A0
IL145430A0 IL14543000A IL14543000A IL145430A0 IL 145430 A0 IL145430 A0 IL 145430A0 IL 14543000 A IL14543000 A IL 14543000A IL 14543000 A IL14543000 A IL 14543000A IL 145430 A0 IL145430 A0 IL 145430A0
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IL
Israel
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processes
preparation
same
pharmaceutical compositions
compositions containing
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IL14543000A
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English (en)
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Axys Pharm Inc
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Publication of IL145430A0 publication Critical patent/IL145430A0/xx

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
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    • C07C255/29—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton containing cyano groups and acylated amino groups bound to the carbon skeleton
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