IL129018A0 - 1H-pyrido (3,4-b) indole-4-carboxamide derivatives their preparation and application thereof in therapeutics - Google Patents

1H-pyrido (3,4-b) indole-4-carboxamide derivatives their preparation and application thereof in therapeutics

Info

Publication number
IL129018A0
IL129018A0 IL12901897A IL12901897A IL129018A0 IL 129018 A0 IL129018 A0 IL 129018A0 IL 12901897 A IL12901897 A IL 12901897A IL 12901897 A IL12901897 A IL 12901897A IL 129018 A0 IL129018 A0 IL 129018A0
Authority
IL
Israel
Prior art keywords
pyrido
therapeutics
indole
preparation
application
Prior art date
Application number
IL12901897A
Other languages
English (en)
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of IL129018A0 publication Critical patent/IL129018A0/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
IL12901897A 1996-10-08 1997-10-03 1H-pyrido (3,4-b) indole-4-carboxamide derivatives their preparation and application thereof in therapeutics IL129018A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9612229A FR2754262B1 (fr) 1996-10-08 1996-10-08 Derives de 1h-pyrido[3,4-b]indole-4-carboxamide, leur preparation et leur application en therapeutique
PCT/FR1997/001750 WO1998015552A1 (fr) 1996-10-08 1997-10-03 DERIVES DE 1H-PYRIDO[3,4-b]INDOLE-4-CARBOXAMIDE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE

Publications (1)

Publication Number Publication Date
IL129018A0 true IL129018A0 (en) 2000-02-17

Family

ID=9496449

Family Applications (1)

Application Number Title Priority Date Filing Date
IL12901897A IL129018A0 (en) 1996-10-08 1997-10-03 1H-pyrido (3,4-b) indole-4-carboxamide derivatives their preparation and application thereof in therapeutics

Country Status (33)

Country Link
US (1) US6075021A (es)
EP (1) EP0934319B1 (es)
JP (1) JP4227197B2 (es)
KR (1) KR100488095B1 (es)
CN (1) CN1089765C (es)
AR (1) AR009112A1 (es)
AT (1) ATE218567T1 (es)
AU (1) AU721102B2 (es)
BG (1) BG63751B1 (es)
BR (1) BR9711879A (es)
CA (1) CA2266376A1 (es)
CO (1) CO4910141A1 (es)
CY (1) CY2291B1 (es)
CZ (1) CZ298906B6 (es)
DE (1) DE69713124T2 (es)
DK (1) DK0934319T3 (es)
EE (1) EE03830B1 (es)
ES (1) ES2178008T3 (es)
FR (1) FR2754262B1 (es)
HK (1) HK1023338A1 (es)
HU (1) HUP9904623A3 (es)
IL (1) IL129018A0 (es)
NO (1) NO311938B1 (es)
NZ (1) NZ334708A (es)
PL (1) PL188244B1 (es)
PT (1) PT934319E (es)
RU (1) RU2180904C2 (es)
SK (1) SK282970B6 (es)
TR (1) TR199900712T2 (es)
TW (1) TW461889B (es)
UA (1) UA57037C2 (es)
WO (1) WO1998015552A1 (es)
ZA (1) ZA978970B (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2766823B1 (fr) * 1997-07-30 1999-10-08 Synthelabo Derives de 4-oxo-3,5-dihydro-4h-pyridazino[4,5-b] indole-1-acetamide, leur preparation et leur application en therapeutique
FR2788696B1 (fr) * 1999-01-26 2004-03-05 Synthelabo Utilisation de derives de pyridazino [4,5-b] indole-1-acetamide pour la preparation de medicaments destines aux maladies du systeme nerveux central
FR2788776B1 (fr) * 1999-01-26 2001-02-23 Synthelabo Derives de 4-oxo-3, 5-dihydro-4h-pyridazino [4,5-b] indole-1 -carboxamide, leur preparation et leur application en therapeutique
FR2811897A1 (fr) * 2000-07-24 2002-01-25 Sanofi Synthelabo UTILISATION DE DERIVES DE PYRIDAZINO[4,5-b]INDOLE-1- ACETAMIDE POUR LA PREPARATION DE MEDICAMENTS DESTINES AU TRAITEMENT DES DYSFONCTIONNEMENTS DES RECEPTEURS DE TYPE PERIPHERIQUE AUX BENZODIAZEPINES
FR2811990A1 (fr) * 2000-07-24 2002-01-25 Sanofi Synthelabo DERIVES DE 1-(4-OXO-3,5-DIHYDRO-4H-PYRIDAZINO[4,5-b]INDOLE-1 -CARBONYL)PIPERAZINE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
FR2833953B1 (fr) * 2001-12-21 2004-12-03 Sanofi Synthelabo DERIVES DE 3-HETEROARYL-3,5-DIHYDRO-4-OXO-4H-PYRIDAZINO [4,5-b]INDOLE-1-CARBOXAMIDE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
FR2838124B1 (fr) 2002-04-03 2004-05-28 Sanofi Synthelabo Derives de 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino [4,5-b]indole-1-acetamide, leur preparation et leur application en therapeutique
PA8586801A1 (es) * 2002-10-31 2005-02-04 Pfizer Inhibidores de hiv-integrasa, composiciones farmaceuticas y metodos para su uso
BRPI0407052A (pt) * 2003-01-27 2006-01-17 Pfizer Inibidores da hiv-integrase, composições farmacêuticas, e métodos para sua utilização
BRPI0510319A (pt) * 2004-04-26 2007-10-16 Pfizer inibidores da enzima integrase de hiv
DE602005002746T2 (de) * 2004-04-26 2008-02-07 Pfizer Inc. Inhibitoren des hiv-integrase-enzyms
JP5483874B2 (ja) * 2005-05-05 2014-05-07 サノフィ−アベンティス・ユー・エス・エルエルシー 安定なナノ粒子処方物
BRPI0616657A2 (pt) * 2005-10-07 2011-06-28 Pfizer Prod Inc inibidores da enzima hiv integrase
UA95788C2 (en) 2005-12-15 2011-09-12 Ф. Хоффманн-Ля Рош Аг Fused pyrrole derivatives
WO2007143597A2 (en) * 2006-06-05 2007-12-13 Novartis Ag Organic compounds
CN1946120B (zh) * 2006-10-20 2010-05-12 华为技术有限公司 实现话单关联的方法及系统
KR100688448B1 (ko) * 2006-12-06 2007-03-02 (주)경진건축사사무소 건축물 내부 조적구조

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2724384B1 (fr) * 1994-09-14 1999-04-16 Cemaf Nouveaux derives de la 3,4-dihydro beta-carboline agonistes de la melatonine, leur procede de preparation et leur utilisation a titre de medicament

Also Published As

Publication number Publication date
CA2266376A1 (en) 1998-04-16
SK45199A3 (en) 2000-02-14
HK1023338A1 (en) 2000-09-08
NZ334708A (en) 2000-10-27
US6075021A (en) 2000-06-13
AU4559497A (en) 1998-05-05
CN1233248A (zh) 1999-10-27
EP0934319B1 (fr) 2002-06-05
BG103301A (en) 2000-05-31
AR009112A1 (es) 2000-03-08
EE03830B1 (et) 2002-08-15
JP4227197B2 (ja) 2009-02-18
FR2754262A1 (fr) 1998-04-10
CO4910141A1 (es) 2000-04-24
KR100488095B1 (ko) 2005-05-09
NO991624L (no) 1999-06-07
CY2291B1 (en) 2003-07-04
CN1089765C (zh) 2002-08-28
DK0934319T3 (da) 2002-09-30
PT934319E (pt) 2002-10-31
UA57037C2 (uk) 2003-06-16
FR2754262B1 (fr) 1998-10-30
BG63751B1 (bg) 2002-11-29
KR20000048992A (ko) 2000-07-25
RU2180904C2 (ru) 2002-03-27
WO1998015552A1 (fr) 1998-04-16
CZ298906B6 (cs) 2008-03-12
ATE218567T1 (de) 2002-06-15
NO991624D0 (no) 1999-04-06
DE69713124D1 (de) 2002-07-11
BR9711879A (pt) 1999-08-24
ZA978970B (en) 1998-04-20
TW461889B (en) 2001-11-01
NO311938B1 (no) 2002-02-18
ES2178008T3 (es) 2002-12-16
TR199900712T2 (xx) 1999-06-21
JP2001508403A (ja) 2001-06-26
EE9900155A (et) 1999-12-15
PL332643A1 (en) 1999-09-27
AU721102B2 (en) 2000-06-22
PL188244B1 (pl) 2005-01-31
CZ119399A3 (cs) 1999-07-14
HUP9904623A3 (en) 2001-03-28
HUP9904623A2 (hu) 2000-06-28
EP0934319A1 (fr) 1999-08-11
SK282970B6 (sk) 2003-01-09
DE69713124T2 (de) 2003-01-30

Similar Documents

Publication Publication Date Title
ZA948592B (en) 7H-imidazo[1,2-a]pyrazin-8-one derivatives,and their preparation and use
SI1001955T1 (en) 1,2,4-triazolo 4,3-b)pyrido 3,2-d)pyridazine derivatives and pharmaceutical compositions containing them
IL111148A0 (en) Imidazol-4- ylpiperidine derivatives, their preparation and their application in therapeutics
IL129018A0 (en) 1H-pyrido (3,4-b) indole-4-carboxamide derivatives their preparation and application thereof in therapeutics
NZ322197A (en) Pyrido[2,3-d] pyrimidine derivatives and pharmaceutical compositions thereof
ZA978081B (en) 3-Substituted pyrido ¬4',3':4,5¾thieno¬2,3-d¾pyrimidine derivatives the preparation and use thereof
HUP0102117A2 (hu) Imidazo[1,2-a]piridin-származékok és ezeket tartalmazó gyógyászati készítmények
HUP9904032A3 (en) 1,2,4-benzothiadiazine derivatives,their preparation and use
ZA978089B (en) 3,4-diaryloxazolone derivatives, their methods of preparation, and their use in therapeutics.
ZA988921B (en) 3,4-diarylthiazolin-2-one or -2-thione derivatives their methods of preparation and their uses in therapeutics
HU9502726D0 (en) [1,2,4]triazolo[4,3-a]qunoxaline derivatives, their preparation and use
ZA986786B (en) 4-oxo-3,5-dihydro-4H-pyridazino[4,5-B]indole-1-acetamide-derivatives their preparation and their application in therapeutics
AU646582B2 (en) Imidazo (2,1-b) benzothiazole-3-acetamide derivatives, their preparation and their use in therapeutics
IL131645A (en) Pyrimido ¬1,2-a¾indole derivatives and their preparation
HUP9904091A3 (en) N-(benzothiazol-2-yl) piperidine-1-ethanamine derivatives, their preparation and application in therapeutics
ZA972894B (en) Diarylmethylidenefuran derivatives, processes for their preparation and their uses in therapeutics.
ZA977767B (en) Benzylamine derivatives, their preparation and their application in therapeutics.
ZA982369B (en) Dihydropyrazino[1,2-a]indol-1-one derivatives their preparation and their use in therapy
AU1858692A (en) 2-piperidinylpyrimidine-4-carboxamide derivatives, their preparation and their use in therapeutics
ZA9811642B (en) Pyrido 1,2,4-thiadiazine derivatives their preparation and use
SI0934319T1 (en) 1H-PYRIDO(3,4-b)INDOLE-4-CARBOXAMIDE DERIVATIVES, PREPARATION AND APPLICATION THEREOF IN THERAPEUTICS
GB2324090B (en) 5,6-O-alkylidene glucono-1(4)-lactones and derivatives thereof,their preparation and use
ZA976828B (en) 6,7,8,9-tetrahydro-5H-imidazo[1,2-a]azepine-3-acetic acid derivatives, their preparation and their application in therapy.
ZA9710515B (en) N-(imidazolybutyl) benezenesulphonamide derivatives, their preparation and their application in therapeutics.
ZA925388B (en) Imidazo(2,1-b)benzothiazole-3-acetamide derivatives,their preparation and their use in therapeutics

Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
KB Patent renewed
KB Patent renewed
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees