AU646582B2 - Imidazo (2,1-b) benzothiazole-3-acetamide derivatives, their preparation and their use in therapeutics - Google Patents

Imidazo (2,1-b) benzothiazole-3-acetamide derivatives, their preparation and their use in therapeutics

Info

Publication number
AU646582B2
AU646582B2 AU20380/92A AU2038092A AU646582B2 AU 646582 B2 AU646582 B2 AU 646582B2 AU 20380/92 A AU20380/92 A AU 20380/92A AU 2038092 A AU2038092 A AU 2038092A AU 646582 B2 AU646582 B2 AU 646582B2
Authority
AU
Australia
Prior art keywords
imidazo
benzothiazole
therapeutics
preparation
acetamide derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU20380/92A
Other versions
AU2038092A (en
Inventor
Danielle De Peretti
Pascal George
Jean-Francois Gibert
Odette Legalloudec
Michel Mangane
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9109138A external-priority patent/FR2679233B1/en
Priority claimed from FR9109139A external-priority patent/FR2679136A1/en
Priority claimed from FR9109137A external-priority patent/FR2679232B1/en
Priority claimed from FR9109136A external-priority patent/FR2679231B1/en
Application filed by Synthelabo SA filed Critical Synthelabo SA
Publication of AU2038092A publication Critical patent/AU2038092A/en
Application granted granted Critical
Publication of AU646582B2 publication Critical patent/AU646582B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AU20380/92A 1991-07-19 1992-07-17 Imidazo (2,1-b) benzothiazole-3-acetamide derivatives, their preparation and their use in therapeutics Ceased AU646582B2 (en)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
FR9109138A FR2679233B1 (en) 1991-07-19 1991-07-19 IMIDAZO [2,1-B] BENZOTHIAZOLE-3-ACETAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION.
FR9109139A FR2679136A1 (en) 1991-07-19 1991-07-19 Medicaments and pharmaceutical compositions based on imidazo[2,1-b]benzothiazol-3-acetamide derivatives
FR9109137A FR2679232B1 (en) 1991-07-19 1991-07-19 ALPHA-HYDROXYIMIDAZO [2,1-B] BENZOTHIAZOLE-3-ACETAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION.
FR9109138 1991-07-19
FR9109136A FR2679231B1 (en) 1991-07-19 1991-07-19 IMIDAZO [2,1-B] BENZOTHIAZOLE-3-ACETAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION, IN THERAPEUTICS.
FR9109137 1991-07-19
FR9109136 1991-07-19
FR9109139 1991-07-19

Publications (2)

Publication Number Publication Date
AU2038092A AU2038092A (en) 1993-01-21
AU646582B2 true AU646582B2 (en) 1994-02-24

Family

ID=27446813

Family Applications (1)

Application Number Title Priority Date Filing Date
AU20380/92A Ceased AU646582B2 (en) 1991-07-19 1992-07-17 Imidazo (2,1-b) benzothiazole-3-acetamide derivatives, their preparation and their use in therapeutics

Country Status (15)

Country Link
EP (1) EP0524055A1 (en)
JP (1) JPH05202063A (en)
KR (1) KR930002358A (en)
CN (1) CN1068826A (en)
AU (1) AU646582B2 (en)
CA (1) CA2074112A1 (en)
CZ (1) CZ224492A3 (en)
FI (1) FI923290A (en)
HU (1) HU9202358D0 (en)
IE (1) IE922342A1 (en)
IL (1) IL102536A0 (en)
MX (1) MX9204179A (en)
NO (1) NO922842L (en)
NZ (1) NZ243595A (en)
PL (1) PL295306A1 (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2699921B1 (en) * 1992-12-30 1995-02-10 Synthelabo 2- (Thien-2-yl) imidazo [2,1-b] benzothiazole-3-acetic acid derivatives, their preparation and their therapeutic use.
CA2215197A1 (en) * 1995-03-13 1996-09-19 Shigeyuki Tasaka Imidazothiazole compound
AU3783497A (en) * 1996-08-09 1998-03-06 Yamanouchi Pharmaceutical Co., Ltd. Metabotropic glutamate receptor agonists
FR2759698B1 (en) * 1997-02-20 1999-03-19 Synthelabo 1,4-DIPHENYLIMIDAZOLE-5-ACETAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
EP0891978B1 (en) * 1997-07-18 2002-03-20 F. Hoffmann-La Roche Ag 5H-Thiazolo (3,2-a) pyrimidine derivatives
CA2436589C (en) * 2001-01-30 2010-10-19 Zenyaku Kogyo Kabushiki Kaisha Heterocyclic compounds and cognitive enhancers comprising the same as effective components
JP2005502623A (en) * 2001-07-02 2005-01-27 ノボ　ノルディスク　アクティーゼルスカブ Substituted piperazines and diazepanes
AU2003297153B2 (en) * 2002-12-18 2010-06-10 Mallinckrodt Inc. Synthesis of heteroaryl acetamides
US20040198783A1 (en) * 2003-04-03 2004-10-07 Semafore Pharmaceuticals Inc. Targeted bone marrow protection agents
KR101549364B1 (en) 2006-03-17 2015-09-01 암비트 바이오사이언시즈 코포레이션 Imidazolothiazole compounds for the treatment of disease
ES2573292T3 (en) 2007-09-19 2016-06-07 Ambit Biosciences Corporation Solid forms comprising N- (5-tert-butyl-isoxazol-3-yl) -N '- {4- [7- (2-morpholin-4-yl-ethoxy) imidazo [2,1-b] [1 , 3] benzothiazol-2-yl] phenyl} urea, compositions thereof and uses thereof
US20190292204A1 (en) * 2018-03-26 2019-09-26 University of Sharjah C/o Dr. Mohamed Al Hemairy MAlhemairy@sharjah.ac.ae Novel heterocyclic systems and pharmaceutical compositions thereof

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU630766B2 (en) * 1989-11-24 1992-11-05 Janssen Pharmaceutica N.V. Immunostimulating 6-aryl-5,6-dihydroimidazo(2,1-b) thiazole derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4464384A (en) * 1981-12-23 1984-08-07 Yamanouchi Pharmaceutical Co., Ltd. 2-Phenylimidazo[2,1-b]benzothiazole compounds, salts thereof, process of producing them, and pharmaceutical compositions containing them
GB8724566D0 (en) * 1987-10-20 1987-11-25 Roussel Lab Ltd Chemical compounds
JP2726999B2 (en) * 1988-06-22 1998-03-11 日研化学株式会社 Imidazo [2,1-b] benzothiazole derivatives and anti-ulcer agents containing the compounds as active ingredients
GB8908845D0 (en) * 1989-04-19 1989-06-07 Roussel Lab Ltd Chemical compounds

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU630766B2 (en) * 1989-11-24 1992-11-05 Janssen Pharmaceutica N.V. Immunostimulating 6-aryl-5,6-dihydroimidazo(2,1-b) thiazole derivatives

Also Published As

Publication number Publication date
HU9202358D0 (en) 1992-10-28
NZ243595A (en) 1994-08-26
JPH05202063A (en) 1993-08-10
MX9204179A (en) 1993-08-01
NO922842L (en) 1993-01-20
EP0524055A1 (en) 1993-01-20
FI923290A (en) 1993-01-20
CZ224492A3 (en) 1993-02-17
NO922842D0 (en) 1992-07-17
IL102536A0 (en) 1993-01-14
IE922342A1 (en) 1993-01-27
CN1068826A (en) 1993-02-10
KR930002358A (en) 1993-02-23
PL295306A1 (en) 1993-03-08
CA2074112A1 (en) 1993-01-20
FI923290A0 (en) 1992-07-17
AU2038092A (en) 1993-01-21

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