HRP20211848T1 - Anti-her2 antitijelo-lijek konjugat - Google Patents

Anti-her2 antitijelo-lijek konjugat Download PDF

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Publication number
HRP20211848T1
HRP20211848T1 HRP20211848TT HRP20211848T HRP20211848T1 HR P20211848 T1 HRP20211848 T1 HR P20211848T1 HR P20211848T T HRP20211848T T HR P20211848TT HR P20211848 T HRP20211848 T HR P20211848T HR P20211848 T1 HRP20211848 T1 HR P20211848T1
Authority
HR
Croatia
Prior art keywords
ch2ch2
ggfg
maleimid
antibody
her2 antibody
Prior art date
Application number
HRP20211848TT
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English (en)
Croatian (hr)
Inventor
Hiroyuki Naito
Yusuke OGITANI
Takeshi Masuda
Takashi Nakada
Masao Yoshida
Shinji Ashida
Koji Morita
Hideki Miyazaki
Yuji Kasuya
Ichiro Hayakawa
Yuki Abe
Original Assignee
Daiichi Sankyo Company, Limited
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=53756672&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20211848(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Daiichi Sankyo Company, Limited filed Critical Daiichi Sankyo Company, Limited
Publication of HRP20211848T1 publication Critical patent/HRP20211848T1/hr

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    • A61K47/6889—Conjugates wherein the antibody being the modifying agent and wherein the linker, binder or spacer confers particular properties to the conjugates, e.g. peptidic enzyme-labile linkers or acid-labile linkers, providing for an acid-labile immuno conjugate wherein the drug may be released from its antibody conjugated part in an acidic, e.g. tumoural or environment
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
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TWI848560B (zh) 2024-07-11
TW202237114A (zh) 2022-10-01
CA2928794A1 (en) 2015-08-06
PL3101032T3 (pl) 2019-07-31
CN105829346A (zh) 2016-08-03
KR102557062B1 (ko) 2023-07-18
SI4212552T1 (sl) 2025-03-31
TWI627967B (zh) 2018-07-01
HRP20241783T1 (hr) 2025-02-28
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TW201613649A (en) 2016-04-16
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