HRP20120490T1 - Spojevi za inhibiciju napredovanja mitoze - Google Patents

Spojevi za inhibiciju napredovanja mitoze Download PDF

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Publication number
HRP20120490T1
HRP20120490T1 HRP20120490TT HRP20120490T HRP20120490T1 HR P20120490 T1 HRP20120490 T1 HR P20120490T1 HR P20120490T T HRP20120490T T HR P20120490TT HR P20120490 T HRP20120490 T HR P20120490T HR P20120490 T1 HRP20120490 T1 HR P20120490T1
Authority
HR
Croatia
Prior art keywords
aliphatic
group
fluoroaliphatic
compound according
fluoro
Prior art date
Application number
HRP20120490TT
Other languages
English (en)
Croatian (hr)
Inventor
Christopher@F@@Claiborne
Todd@B@@Sells
Stephen@G@@Stroud
Original Assignee
Millennium@Pharmaceuticals
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39315133&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20120490(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Millennium@Pharmaceuticals filed Critical Millennium@Pharmaceuticals
Publication of HRP20120490T1 publication Critical patent/HRP20120490T1/hr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HRP20120490TT 2006-11-16 2007-11-14 Spojevi za inhibiciju napredovanja mitoze HRP20120490T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US85934006P 2006-11-16 2006-11-16
PCT/US2007/023948 WO2008063525A1 (en) 2006-11-16 2007-11-14 Compounds for inhibiting mitotic progression

Publications (1)

Publication Number Publication Date
HRP20120490T1 true HRP20120490T1 (hr) 2012-07-31

Family

ID=39315133

Family Applications (2)

Application Number Title Priority Date Filing Date
HRP20120490TT HRP20120490T1 (hr) 2006-11-16 2007-11-14 Spojevi za inhibiciju napredovanja mitoze
HRP20150047TT HRP20150047T1 (en) 2006-11-16 2015-01-13 Compound for inhibiting mitotic progression

Family Applications After (1)

Application Number Title Priority Date Filing Date
HRP20150047TT HRP20150047T1 (en) 2006-11-16 2015-01-13 Compound for inhibiting mitotic progression

Country Status (34)

Country Link
US (7) US8026246B2 (enExample)
EP (4) EP2086981B1 (enExample)
JP (3) JP5102839B2 (enExample)
KR (2) KR101342014B1 (enExample)
CN (2) CN103483343B (enExample)
AR (1) AR064246A1 (enExample)
AT (1) ATE556076T1 (enExample)
AU (1) AU2007322046B2 (enExample)
BR (1) BRPI0718803B8 (enExample)
CA (1) CA2669680C (enExample)
CL (1) CL2007003244A1 (enExample)
CR (3) CR10782A (enExample)
CY (1) CY1112828T1 (enExample)
DK (2) DK2086981T3 (enExample)
EA (1) EA015779B1 (enExample)
ES (3) ES2528793T3 (enExample)
GE (1) GEP20125459B (enExample)
HR (2) HRP20120490T1 (enExample)
IL (1) IL198690A0 (enExample)
MA (1) MA30988B1 (enExample)
MX (3) MX2009004670A (enExample)
MY (1) MY153243A (enExample)
NO (1) NO343338B1 (enExample)
NZ (3) NZ597252A (enExample)
PH (1) PH12012502057B1 (enExample)
PL (2) PL2497772T3 (enExample)
PT (2) PT2086981E (enExample)
RS (2) RS53788B1 (enExample)
SG (2) SG10201503350TA (enExample)
SI (2) SI2497772T1 (enExample)
TW (1) TWI401255B (enExample)
UA (1) UA94129C2 (enExample)
WO (1) WO2008063525A1 (enExample)
ZA (1) ZA200903279B (enExample)

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JP6955485B2 (ja) 2015-09-09 2021-10-27 アイカーン スクール オブ メディスン アット マウント サイナイＩｃａｈｎ Ｓｃｈｏｏｌ ｏｆ Ｍｅｄｉｃｉｎｅ ａｔ Ｍｔ． Ｓｉｎａｉ 抗がん剤としての複素環式の限定された三環系スルホンアミド
JP6591036B2 (ja) 2016-02-26 2019-10-16 公益財団法人がん研究会 Ｈｐ１の機能に着目した抗癌剤のスクリーニング方法及び評価系
WO2017157825A1 (en) 2016-03-15 2017-09-21 F. Hoffmann-La Roche Ag Combinations of lsd1 inhibitors for use in the treatment of solid tumors
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Also Published As

Publication number Publication date
MX343391B (es) 2016-11-04
US20190031662A1 (en) 2019-01-31
JP5452811B2 (ja) 2014-03-26
BRPI0718803B1 (pt) 2020-11-17
NO343338B1 (no) 2019-02-04
ES2537451T3 (es) 2015-06-08
BRPI0718803B8 (pt) 2021-05-25
NZ597252A (en) 2013-06-28
SG176443A1 (en) 2011-12-29
TW200829589A (en) 2008-07-16
PL2086981T3 (pl) 2012-09-28
HK1175777A1 (en) 2013-07-12
US20150166545A1 (en) 2015-06-18
ES2384123T3 (es) 2012-06-29
EP2497772A1 (en) 2012-09-12
US10836766B2 (en) 2020-11-17
NZ611898A (en) 2015-01-30
HK1175778A1 (en) 2013-07-12
MX2009004670A (es) 2009-05-15
PT2086981E (pt) 2012-06-20
CA2669680A1 (en) 2008-05-29
DK2497772T3 (en) 2015-01-19
JP2012006965A (ja) 2012-01-12
US9765076B2 (en) 2017-09-19
PH12012502057A1 (en) 2015-09-14
CL2007003244A1 (es) 2008-04-04
US20240400567A1 (en) 2024-12-05
ZA200903279B (en) 2010-07-28
HRP20150047T1 (en) 2015-03-13
MX348568B (es) 2017-06-20
PT2497772E (pt) 2015-02-05
MY153243A (en) 2015-01-29
TWI401255B (zh) 2013-07-11
CR20140544A (es) 2015-01-12
CA2669680C (en) 2012-04-10
CN101547924A (zh) 2009-09-30
EP2086981B1 (en) 2012-05-02
IL198690A0 (en) 2010-02-17
MA30988B1 (fr) 2009-12-01
US20080167292A1 (en) 2008-07-10
SI2086981T1 (sl) 2012-12-31
EA015779B1 (ru) 2011-12-30
SI2497772T1 (sl) 2015-03-31
CN103483343B (zh) 2016-06-01
SG10201503350TA (en) 2015-06-29
AR064246A1 (es) 2009-03-25
KR101110458B1 (ko) 2012-03-13
WO2008063525A1 (en) 2008-05-29
DK2086981T3 (da) 2012-08-06
CR10782A (es) 2009-06-24
ES2528793T3 (es) 2015-02-12
EP2944639B1 (en) 2017-01-04
US20110312942A1 (en) 2011-12-22
UA94129C2 (ru) 2011-04-11
EP2497773B1 (en) 2015-02-25
PH12012502057B1 (en) 2018-10-24
KR20090091173A (ko) 2009-08-26
JP2010510215A (ja) 2010-04-02
RS52313B (sr) 2012-12-31
EA200970486A1 (ru) 2009-10-30
EP2497773A1 (en) 2012-09-12
BRPI0718803A2 (pt) 2013-12-03
CY1112828T1 (el) 2016-02-10
CR20140154A (es) 2014-07-23
KR20110113210A (ko) 2011-10-14
ATE556076T1 (de) 2012-05-15
AU2007322046A1 (en) 2008-05-29
US20110312943A1 (en) 2011-12-22
JP5102839B2 (ja) 2012-12-19
HK1217699A1 (en) 2017-01-20
NO20091864L (no) 2009-06-15
KR101342014B1 (ko) 2013-12-19
NZ577042A (en) 2012-03-30
PL2497772T3 (pl) 2015-05-29
CN103483343A (zh) 2014-01-01
US8026246B2 (en) 2011-09-27
EP2086981A1 (en) 2009-08-12
US20210214361A1 (en) 2021-07-15
EP2497772B1 (en) 2014-10-29
GEP20125459B (en) 2012-03-26
JP2014055166A (ja) 2014-03-27
AU2007322046B2 (en) 2012-04-05
US9988384B2 (en) 2018-06-05
US11958855B2 (en) 2024-04-16
EP2944639A1 (en) 2015-11-18
HK1134672A1 (en) 2010-05-07
RS53788B1 (sr) 2015-06-30
CN101547924B (zh) 2013-09-25

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