CR10782A - Compuestos para inhibir la progresion mitotica - Google Patents

Compuestos para inhibir la progresion mitotica

Info

Publication number
CR10782A
CR10782A CR10782A CR10782A CR10782A CR 10782 A CR10782 A CR 10782A CR 10782 A CR10782 A CR 10782A CR 10782 A CR10782 A CR 10782A CR 10782 A CR10782 A CR 10782A
Authority
CR
Costa Rica
Prior art keywords
compounds
mythical
progression
inhibit
cancer
Prior art date
Application number
CR10782A
Other languages
English (en)
Spanish (es)
Inventor
Christopher F Claiborne
Todd B Sells
Stephen G Stroud
Original Assignee
Millenium Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39315133&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR10782(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Millenium Pharmaceuticals Inc filed Critical Millenium Pharmaceuticals Inc
Publication of CR10782A publication Critical patent/CR10782A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CR10782A 2006-11-16 2009-05-08 Compuestos para inhibir la progresion mitotica CR10782A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US85934006P 2006-11-16 2006-11-16

Publications (1)

Publication Number Publication Date
CR10782A true CR10782A (es) 2009-06-24

Family

ID=39315133

Family Applications (3)

Application Number Title Priority Date Filing Date
CR10782A CR10782A (es) 2006-11-16 2009-05-08 Compuestos para inhibir la progresion mitotica
CR20140154A CR20140154A (es) 2006-11-16 2014-04-04 Compuestos para inhibir la progresión mitotica
CR20140544A CR20140544A (es) 2006-11-16 2014-11-27 Compuestos para inhibir la progresión mitotica

Family Applications After (2)

Application Number Title Priority Date Filing Date
CR20140154A CR20140154A (es) 2006-11-16 2014-04-04 Compuestos para inhibir la progresión mitotica
CR20140544A CR20140544A (es) 2006-11-16 2014-11-27 Compuestos para inhibir la progresión mitotica

Country Status (34)

Country Link
US (7) US8026246B2 (enExample)
EP (4) EP2944639B1 (enExample)
JP (3) JP5102839B2 (enExample)
KR (2) KR101342014B1 (enExample)
CN (2) CN103483343B (enExample)
AR (1) AR064246A1 (enExample)
AT (1) ATE556076T1 (enExample)
AU (1) AU2007322046B2 (enExample)
BR (1) BRPI0718803B8 (enExample)
CA (1) CA2669680C (enExample)
CL (1) CL2007003244A1 (enExample)
CR (3) CR10782A (enExample)
CY (1) CY1112828T1 (enExample)
DK (2) DK2086981T3 (enExample)
EA (1) EA015779B1 (enExample)
ES (3) ES2537451T3 (enExample)
GE (1) GEP20125459B (enExample)
HR (2) HRP20120490T1 (enExample)
IL (1) IL198690A0 (enExample)
MA (1) MA30988B1 (enExample)
MX (3) MX348568B (enExample)
MY (1) MY153243A (enExample)
NO (1) NO343338B1 (enExample)
NZ (3) NZ611898A (enExample)
PH (1) PH12012502057B1 (enExample)
PL (2) PL2086981T3 (enExample)
PT (2) PT2086981E (enExample)
RS (2) RS52313B (enExample)
SG (2) SG176443A1 (enExample)
SI (2) SI2086981T1 (enExample)
TW (1) TWI401255B (enExample)
UA (1) UA94129C2 (enExample)
WO (1) WO2008063525A1 (enExample)
ZA (1) ZA200903279B (enExample)

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JO3635B1 (ar) 2009-05-18 2020-08-27 Millennium Pharm Inc مركبات صيدلانية صلبة وطرق لانتاجها
JO3434B1 (ar) * 2009-07-31 2019-10-20 Millennium Pharm Inc مركبات صيدلانية لمعالجة السرطان وامراض واضطرابات اخري
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US20120107304A1 (en) 2010-04-27 2012-05-03 Boehringer Ingelheim International Gmbh Combination therapy in treatment of oncological and fibrotic diseases
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UY34114A (es) 2011-06-03 2013-01-03 Millennium Pharm Inc Combinación de inhibidores de mek e inhibidores selectivos de la quiinasa aurora a
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EP2976086B1 (en) * 2013-03-22 2020-10-14 Millennium Pharmaceuticals, Inc. Combination of catalytic mtorc 1/2 inhibitors and selective inhibitors of aurora a kinase
JP6525474B2 (ja) 2013-12-06 2019-06-05 ミレニアム ファーマシューティカルズ， インコーポレイテッドＭｉｌｌｅｎｎｉｕｍ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ， Ｉｎｃ． オーロラキナーゼ阻害剤と抗ｃｄ３０抗体の併用
CA2972076A1 (en) * 2014-12-23 2016-06-30 Millennium Pharmaceuticals, Inc. Combination of raf inhibitors and aurora kinase inhibitors
EP3324976A4 (en) 2015-07-21 2019-03-27 Millennium Pharmaceuticals, Inc. ADMINISTRATION OF KINASE AURORA INHIBITOR AND CHEMOTHERAPEUTIC AGENTS
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CA2997784A1 (en) 2015-09-09 2017-03-16 Icahn School Of Medicine At Mount Sinai Heterocyclic constrained tricyclic sulfonamides as anti-cancer agents
WO2017146253A1 (ja) 2016-02-26 2017-08-31 公益財団法人がん研究会 Ｈｐ１の機能に着目した抗癌剤のスクリーニング方法及び評価系
AU2017233898B2 (en) 2016-03-15 2022-12-15 Oryzon Genomics, S.A. Combinations of LSD1 inhibitors for use in the treatment of solid tumors
JP6188986B1 (ja) * 2017-03-23 2017-08-30 株式会社ノエビア 時計遺伝子発現量調整剤及びエラスチン産生促進剤
WO2019195658A1 (en) 2018-04-05 2019-10-10 Dana-Farber Cancer Institute, Inc. Sting levels as a biomarker for cancer immunotherapy
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WO2021041532A1 (en) 2019-08-26 2021-03-04 Dana-Farber Cancer Institute, Inc. Use of heparin to promote type 1 interferon signaling
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WO2025075211A1 (en) 2023-10-03 2025-04-10 Takeda Pharmaceutical Company Limited Alisertib and paclitaxel for treating small cell lung cancer
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Also Published As

Publication number Publication date
ATE556076T1 (de) 2012-05-15
US20110312943A1 (en) 2011-12-22
CA2669680A1 (en) 2008-05-29
PL2086981T3 (pl) 2012-09-28
BRPI0718803A2 (pt) 2013-12-03
MA30988B1 (fr) 2009-12-01
CA2669680C (en) 2012-04-10
US20190031662A1 (en) 2019-01-31
US11958855B2 (en) 2024-04-16
DK2086981T3 (da) 2012-08-06
US8026246B2 (en) 2011-09-27
CN101547924A (zh) 2009-09-30
US20080167292A1 (en) 2008-07-10
AR064246A1 (es) 2009-03-25
NZ611898A (en) 2015-01-30
IL198690A0 (en) 2010-02-17
SG176443A1 (en) 2011-12-29
TWI401255B (zh) 2013-07-11
GEP20125459B (en) 2012-03-26
CY1112828T1 (el) 2016-02-10
CR20140544A (es) 2015-01-12
PH12012502057A1 (en) 2015-09-14
RS52313B (sr) 2012-12-31
SG10201503350TA (en) 2015-06-29
EP2944639B1 (en) 2017-01-04
BRPI0718803B8 (pt) 2021-05-25
EP2497773A1 (en) 2012-09-12
US10836766B2 (en) 2020-11-17
CN103483343B (zh) 2016-06-01
UA94129C2 (ru) 2011-04-11
ES2384123T3 (es) 2012-06-29
AU2007322046B2 (en) 2012-04-05
MX348568B (es) 2017-06-20
HK1134672A1 (en) 2010-05-07
CN101547924B (zh) 2013-09-25
PT2497772E (pt) 2015-02-05
CL2007003244A1 (es) 2008-04-04
EP2086981A1 (en) 2009-08-12
RS53788B1 (sr) 2015-06-30
NO343338B1 (no) 2019-02-04
MY153243A (en) 2015-01-29
BRPI0718803B1 (pt) 2020-11-17
KR101110458B1 (ko) 2012-03-13
EP2497772A1 (en) 2012-09-12
MX343391B (es) 2016-11-04
US20210214361A1 (en) 2021-07-15
KR101342014B1 (ko) 2013-12-19
HK1175778A1 (en) 2013-07-12
EP2497772B1 (en) 2014-10-29
EA200970486A1 (ru) 2009-10-30
KR20090091173A (ko) 2009-08-26
US9765076B2 (en) 2017-09-19
CN103483343A (zh) 2014-01-01
PL2497772T3 (pl) 2015-05-29
US9988384B2 (en) 2018-06-05
CR20140154A (es) 2014-07-23
JP5102839B2 (ja) 2012-12-19
ZA200903279B (en) 2010-07-28
SI2086981T1 (sl) 2012-12-31
JP2010510215A (ja) 2010-04-02
EA015779B1 (ru) 2011-12-30
HRP20120490T1 (hr) 2012-07-31
ES2537451T3 (es) 2015-06-08
EP2944639A1 (en) 2015-11-18
PH12012502057B1 (en) 2018-10-24
HRP20150047T1 (en) 2015-03-13
US20110312942A1 (en) 2011-12-22
DK2497772T3 (en) 2015-01-19
KR20110113210A (ko) 2011-10-14
JP5452811B2 (ja) 2014-03-26
US20240400567A1 (en) 2024-12-05
NZ577042A (en) 2012-03-30
ES2528793T3 (es) 2015-02-12
EP2086981B1 (en) 2012-05-02
NZ597252A (en) 2013-06-28
AU2007322046A1 (en) 2008-05-29
JP2014055166A (ja) 2014-03-27
HK1175777A1 (en) 2013-07-12
SI2497772T1 (sl) 2015-03-31
EP2497773B1 (en) 2015-02-25
MX2009004670A (es) 2009-05-15
PT2086981E (pt) 2012-06-20
TW200829589A (en) 2008-07-16
JP2012006965A (ja) 2012-01-12
NO20091864L (no) 2009-06-15
HK1217699A1 (en) 2017-01-20
US20150166545A1 (en) 2015-06-18
WO2008063525A1 (en) 2008-05-29

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