GT200600202AA - Proceso para la síntesis de compuestos orgánicos - Google Patents

Proceso para la síntesis de compuestos orgánicos

Info

Publication number
GT200600202AA
GT200600202AA GT200600202AK GT200600202K GT200600202AA GT 200600202A A GT200600202A A GT 200600202AA GT 200600202A K GT200600202A K GT 200600202AK GT 200600202 K GT200600202 K GT 200600202K GT 200600202A A GT200600202A A GT 200600202AA
Authority
GT
Guatemala
Prior art keywords
synthesis
organic compounds
methyl
bencenamine
pyrimidil
Prior art date
Application number
GT200600202AK
Other languages
English (en)
Spanish (es)
Inventor
Stephan Abel
Murat Acemoglu
Bernhard Erb
Christoph Krell
Joseph Sclafani
Mark Meisenbach
Mahavir Prashad
Wen-Chung Shieh
Song Xue
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37149980&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT200600202A(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of GT200600202AA publication Critical patent/GT200600202AA/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/07—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms
    • C07C205/11—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms having nitro groups bound to carbon atoms of six-membered aromatic rings
    • C07C205/12—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms having nitro groups bound to carbon atoms of six-membered aromatic rings the six-membered aromatic ring or a condensed ring system containing that ring being substituted by halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C07D233/61—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms not forming part of a nitro radical, attached to ring nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
GT200600202AK 2005-06-09 2012-05-17 Proceso para la síntesis de compuestos orgánicos GT200600202AA (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US68897605P 2005-06-09 2005-06-09

Publications (1)

Publication Number Publication Date
GT200600202AA true GT200600202AA (es) 2014-06-09

Family

ID=37149980

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200600202AK GT200600202AA (es) 2005-06-09 2012-05-17 Proceso para la síntesis de compuestos orgánicos

Country Status (25)

Country Link
US (2) US7781597B2 (fr)
EP (3) EP2292607B1 (fr)
JP (2) JP5225078B2 (fr)
KR (2) KR101283109B1 (fr)
CN (6) CN102180836B (fr)
AR (1) AR057056A1 (fr)
AT (1) ATE540931T1 (fr)
AU (3) AU2006258050B2 (fr)
BR (1) BRPI0611683A2 (fr)
CA (4) CA2886482C (fr)
DK (2) DK2292607T3 (fr)
ES (3) ES2558696T3 (fr)
GT (1) GT200600202AA (fr)
HU (1) HUE028024T2 (fr)
IN (2) IN2014DN08588A (fr)
JO (1) JO2758B1 (fr)
MX (1) MX2007015609A (fr)
MY (1) MY146795A (fr)
PE (3) PE20100715A1 (fr)
PL (3) PL2292607T3 (fr)
PT (3) PT1896426E (fr)
RU (1) RU2446162C2 (fr)
SI (2) SI2266961T1 (fr)
TW (1) TWI380981B (fr)
WO (1) WO2006135640A2 (fr)

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KR101197482B1 (ko) 2004-03-05 2012-11-09 닛산 가가쿠 고교 가부시키 가이샤 이속사졸린 치환 벤즈아미드 화합물 및 유해생물 방제제
MY146795A (en) * 2005-06-09 2012-09-28 Novartis Ag Process for the synthesis of organic compounds
TW200803740A (en) 2005-12-16 2008-01-16 Du Pont 5-aryl isoxazolines for controlling invertebrate pests
TWI412322B (zh) 2005-12-30 2013-10-21 Du Pont 控制無脊椎害蟲之異唑啉
EP2155701B1 (fr) 2007-06-13 2013-12-11 E. I. Du Pont de Nemours and Company Insecticides à l'isoxazoline
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
PL2957284T3 (pl) 2007-06-27 2018-08-31 E. I. Du Pont De Nemours And Company Sposób zwalczania szkodników zwierzęcych
TWI649303B (zh) 2007-08-17 2019-02-01 杜邦股份有限公司 製備４-乙醯基-ｎ-〔２-側氧基-２-〔（２，２，２-三氟乙基）胺基〕乙基〕-１-萘甲醯胺之化合物及方法
EP2193124B1 (fr) 2007-10-03 2012-12-19 E. I. du Pont de Nemours and Company Composés de naphtalène isoxazoline destinés à la lutte contre les organismes nuisibles invertébrés
TWI455919B (zh) * 2008-04-09 2014-10-11 Du Pont 製備３－三氟甲基查耳酮（ｃｈａｌｃｏｎｅ）之方法
EP2305667A3 (fr) 2008-07-17 2011-05-11 Teva Pharmaceutical Industries Ltd. Produits intermédiaires du nilotinib et préparation de ceux-ci
EP2262793B1 (fr) 2008-11-05 2012-10-03 Teva Pharmaceutical Industries Ltd. Formes cristallines de nilotinib hcl
WO2010060074A1 (fr) * 2008-11-24 2010-05-27 Teva Pharmaceutical Industries Ltd. Synthèse du nilotinib et ses intermédiaires
US20110053968A1 (en) 2009-06-09 2011-03-03 Auspex Pharmaceuticals, Inc. Aminopyrimidine inhibitors of tyrosine kinase
HUE028501T2 (en) 2010-05-27 2016-12-28 Du Pont 4- [5- [3-Chloro-5- (trifluoromethyl) phenyl] -4,5-dihydro-5- (trifluoromethyl) -3-isoxazolyl] -N- [2-oxo-2 - [(2.2, 2-Trifluoroethyl) amino] ethyl] -1-naphthalenecarboxamide crystalline form
PE20141404A1 (es) 2011-12-30 2014-10-28 Hanmi Pharm Ind Co Ltd Derivados de tieno[3,2-d]pirimidina que tienen actividad inhibidora por las quinasas de las proteinas
CN102592837B (zh) * 2012-03-12 2014-01-15 河北师范大学 制备超级电容器用四氯合金属季铵盐掺杂聚苯胺电极的方法
CN103694176B (zh) 2014-01-07 2015-02-18 苏州立新制药有限公司 尼洛替尼中间体的制备方法
CN104592122B (zh) * 2014-12-09 2018-01-23 凯莱英医药集团（天津）股份有限公司 3‑(4‑甲基‑1h‑咪唑‑1‑基)‑5‑(三氟甲基)苯胺的制备方法
CN105985293B (zh) * 2015-03-04 2018-04-03 埃斯特维华义制药有限公司 尼洛替尼中间体的制备方法
EP3095782A1 (fr) 2015-05-18 2016-11-23 Esteve Química, S.A. Nouveau procédé de préparation de 3- (4-methyl-1h-imidazol-1-yl) -5- (trifluorométhyl) benzénamine
CN107201532B (zh) * 2017-05-09 2019-08-27 吉林凯莱英医药化学有限公司 芳香化合物的硝化方法
WO2019130254A1 (fr) * 2018-01-01 2019-07-04 Laurus Labs Ltd Procédé amélioré pour 3-(4-méthyl-1h-imidazol-1-yl)-5-(trifluorométhyl) aniline
CN108530364B (zh) 2018-04-10 2020-01-21 江苏创诺制药有限公司 一种3-(4-甲基-1h-咪唑-1-基)-5-三氟甲基苯胺单盐酸盐的晶型及其应用
AU2019285066B2 (en) 2018-06-15 2024-06-13 Handa Pharmaceuticals, Inc. Kinase inhibitor salts and compositions thereof
CN112105603B (zh) * 2019-04-06 2024-01-30 特里纳普克公司 磺酰基二唑和n-(氟磺酰基)唑及其制备方法
EP3904342A1 (fr) 2020-04-28 2021-11-03 Grindeks, A Joint Stock Company Procédé de préparation de 3-(trifluorométhyl)-5-(4-méthyl-1h-imidazole-1-yl)-benzèneamine hydrochlorure
CN114751836B (zh) * 2021-02-23 2024-05-31 四川青木制药有限公司 3-(4-甲基-1h-咪唑-1-基)-5-(三氟甲基)苯胺合成方法及其中间体
CN114853734A (zh) * 2022-06-14 2022-08-05 海南鑫开源医药科技有限公司 一种尼洛替尼游离碱的制备方法
CN115626880B (zh) * 2022-11-15 2023-11-14 常州大学 3-硝基-5-氰基三氟甲苯的合成方法

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SU1051076A1 (ru) * 1982-04-09 1983-10-30 Алтайский политехнический институт Способ получени производных имидазола
GB8413685D0 (en) * 1984-05-29 1984-07-04 Pfizer Ltd Quinolone inotropic agents
GR851296B (fr) * 1984-05-29 1985-11-25 Pfizer
GB8502267D0 (en) * 1985-01-30 1985-02-27 Pfizer Ltd Quinolone inotropic agents
HN2001000008A (es) * 2000-01-21 2003-12-11 Inc Agouron Pharmaceuticals Compuesto de amida y composiciones farmaceuticas para inhibir proteinquinasas, y su modo de empleo
GB0023383D0 (en) * 2000-09-23 2000-11-08 Synprotec Ltd 3,5-Bis (Trifluormethyl)Benzene derivatives
TW200406374A (en) * 2002-05-29 2004-05-01 Novartis Ag Diaryl urea derivatives useful for the treatment of protein kinase dependent diseases
GB0215676D0 (en) * 2002-07-05 2002-08-14 Novartis Ag Organic compounds
GB0222514D0 (en) * 2002-09-27 2002-11-06 Novartis Ag Organic compounds
CN1939910A (zh) * 2004-12-31 2007-04-04 孙飘扬 氨基嘧啶类化合物及其盐和其制备方法与药物用途
GT200600207A (es) * 2005-06-09 2007-01-15 Novartis Ag Proceso para la síntesis de compuestos orgánicos
MY146795A (en) * 2005-06-09 2012-09-28 Novartis Ag Process for the synthesis of organic compounds

Also Published As

Publication number Publication date
CA2611280A1 (fr) 2006-12-21
JP2013035855A (ja) 2013-02-21
EP1896426B1 (fr) 2012-01-11
SI2292607T1 (sl) 2014-09-30
DK2292607T3 (da) 2014-06-30
ATE540931T1 (de) 2012-01-15
EP2266961B1 (fr) 2015-10-21
JP5225078B2 (ja) 2013-07-03
KR101283109B1 (ko) 2013-07-05
JO2758B1 (en) 2014-03-15
EP2266961A2 (fr) 2010-12-29
IN2014DN08588A (fr) 2015-07-10
IN2014DN08578A (fr) 2015-07-10
RU2007148238A (ru) 2009-07-20
EP1896426A2 (fr) 2008-03-12
AU2010241374B2 (en) 2011-11-03
CN102174020B (zh) 2012-11-07
PL2266961T3 (pl) 2016-04-29
AU2006258050A1 (en) 2006-12-21
TW200716563A (en) 2007-05-01
CN102180796A (zh) 2011-09-14
DK2266961T3 (en) 2016-01-25
PE20100715A1 (es) 2010-10-25
KR20080014010A (ko) 2008-02-13
EP2292607B1 (fr) 2014-04-09
CN101189212A (zh) 2008-05-28
AU2010241374A1 (en) 2010-12-02
EP2266961A3 (fr) 2011-07-27
CA2886482A1 (fr) 2006-12-21
BRPI0611683A2 (pt) 2010-09-28
KR101249199B1 (ko) 2013-04-03
PT2266961E (pt) 2016-02-05
ES2465522T3 (es) 2014-06-06
MY146795A (en) 2012-09-28
PT1896426E (pt) 2012-04-12
CA2886482C (fr) 2017-09-05
PT2292607E (pt) 2014-06-24
ES2380489T8 (es) 2012-06-22
CN102174019B (zh) 2013-02-13
ES2558696T3 (es) 2016-02-08
PE20070109A1 (es) 2007-04-02
CA2611280C (fr) 2014-01-28
PE20100716A1 (es) 2010-10-25
TWI380981B (zh) 2013-01-01
CN102174021A (zh) 2011-09-07
US20100280257A1 (en) 2010-11-04
US20080200692A1 (en) 2008-08-21
AR057056A1 (es) 2007-11-14
CA2833394C (fr) 2016-03-29
PL1896426T3 (pl) 2012-06-29
WO2006135640A2 (fr) 2006-12-21
HUE028024T2 (en) 2016-11-28
EP2292607A2 (fr) 2011-03-09
CN102174021B (zh) 2013-02-27
SI2266961T1 (sl) 2016-02-29
AU2006258050B2 (en) 2010-12-09
CN102180836A (zh) 2011-09-14
KR20120099028A (ko) 2012-09-06
CN101189212B (zh) 2011-05-18
PL2292607T3 (pl) 2014-09-30
CA2833394A1 (fr) 2006-12-21
RU2446162C2 (ru) 2012-03-27
US7781597B2 (en) 2010-08-24
CN102174019A (zh) 2011-09-07
CA2942046A1 (fr) 2006-12-21
EP2292607A3 (fr) 2011-04-27
ES2380489T3 (es) 2012-05-14
CN102180836B (zh) 2012-11-21
CN102174020A (zh) 2011-09-07
US8008504B2 (en) 2011-08-30
WO2006135640A3 (fr) 2007-08-02
JP2008546645A (ja) 2008-12-25
MX2007015609A (es) 2008-02-25
AU2011201044A1 (en) 2011-03-31

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