GT200100023A - Carboxamidas de pirimidina utiles como inhibidores de isozimas pde4. - Google Patents

Carboxamidas de pirimidina utiles como inhibidores de isozimas pde4.

Info

Publication number
GT200100023A
GT200100023A GT200100023A GT200100023A GT200100023A GT 200100023 A GT200100023 A GT 200100023A GT 200100023 A GT200100023 A GT 200100023A GT 200100023 A GT200100023 A GT 200100023A GT 200100023 A GT200100023 A GT 200100023A
Authority
GT
Guatemala
Prior art keywords
inhibitors
isozimas
carboxamids
pde4
useful
Prior art date
Application number
GT200100023A
Other languages
English (en)
Spanish (es)
Inventor
Robert James Chambers
Thomas Victor Magee
Anthony Marfat
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of GT200100023A publication Critical patent/GT200100023A/es

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    • C07—ORGANIC CHEMISTRY
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    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
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    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
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    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Molecular Biology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Biotechnology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Vascular Medicine (AREA)
GT200100023A 2000-01-31 2001-01-31 Carboxamidas de pirimidina utiles como inhibidores de isozimas pde4. GT200100023A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17928200P 2000-01-31 2000-01-31

Publications (1)

Publication Number Publication Date
GT200100023A true GT200100023A (es) 2001-12-19

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Application Number Title Priority Date Filing Date
GT200100023A GT200100023A (es) 2000-01-31 2001-01-31 Carboxamidas de pirimidina utiles como inhibidores de isozimas pde4.

Country Status (44)

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US (1) US6740655B2 (en, 2012)
EP (1) EP1252157B1 (en, 2012)
JP (1) JP2003522165A (en, 2012)
KR (1) KR20020071029A (en, 2012)
CN (1) CN1404480A (en, 2012)
AP (1) AP2002002590A0 (en, 2012)
AR (1) AR027336A1 (en, 2012)
AT (1) ATE269860T1 (en, 2012)
AU (1) AU2700301A (en, 2012)
BG (1) BG106868A (en, 2012)
BR (1) BR0107934A (en, 2012)
CA (1) CA2396458C (en, 2012)
CO (1) CO5271669A1 (en, 2012)
CR (1) CR6714A (en, 2012)
CZ (1) CZ20022413A3 (en, 2012)
DE (1) DE60103976T2 (en, 2012)
DK (1) DK1252157T3 (en, 2012)
DZ (1) DZ3406A1 (en, 2012)
EA (1) EA005028B1 (en, 2012)
EE (1) EE200200426A (en, 2012)
ES (1) ES2223772T3 (en, 2012)
GE (1) GEP20043385B (en, 2012)
GT (1) GT200100023A (en, 2012)
HK (1) HK1054232A1 (en, 2012)
HN (1) HN2001000018A (en, 2012)
HU (1) HUP0204271A3 (en, 2012)
IL (1) IL150486A0 (en, 2012)
IS (1) IS6444A (en, 2012)
MA (1) MA26871A1 (en, 2012)
MX (1) MXPA02007465A (en, 2012)
NO (1) NO20023614L (en, 2012)
NZ (1) NZ519726A (en, 2012)
OA (1) OA12170A (en, 2012)
PA (1) PA8511301A1 (en, 2012)
PE (1) PE20011059A1 (en, 2012)
PL (1) PL357555A1 (en, 2012)
PT (1) PT1252157E (en, 2012)
SK (1) SK10342002A3 (en, 2012)
SV (1) SV2001000298A (en, 2012)
TN (1) TNSN01019A1 (en, 2012)
TR (1) TR200402292T4 (en, 2012)
UY (1) UY26570A1 (en, 2012)
WO (1) WO2001057025A1 (en, 2012)
ZA (1) ZA200206034B (en, 2012)

Families Citing this family (86)

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Publication number Priority date Publication date Assignee Title
ES2165768B1 (es) 1999-07-14 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen.
DE60019167T2 (de) * 1999-12-24 2006-05-11 Glaxo Group Ltd., Greenford Pharmazeutische aerosol formulierung enthaltend salmeterol und fluticason
DE10110772A1 (de) * 2001-03-07 2002-09-12 Boehringer Ingelheim Pharma Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und PDE-IV-Inhibitoren
US7776315B2 (en) 2000-10-31 2010-08-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmaceutical compositions based on anticholinergics and additional active ingredients
YU39503A (sh) * 2000-11-22 2006-05-25 F. Hoffmann-La Roche Ag. Derivati pirimidina
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