HN2001000018A - Carboxamidas de pirimidina utiles como inhibidores de isozimas pde4. - Google Patents

Carboxamidas de pirimidina utiles como inhibidores de isozimas pde4.

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Publication number
HN2001000018A
HN2001000018A HN2001000018A HN2001000018A HN2001000018A HN 2001000018 A HN2001000018 A HN 2001000018A HN 2001000018 A HN2001000018 A HN 2001000018A HN 2001000018 A HN2001000018 A HN 2001000018A HN 2001000018 A HN2001000018 A HN 2001000018A
Authority
HN
Honduras
Prior art keywords
pde4
isozimas
carboxamids
inhibitors
pyrimidine
Prior art date
Application number
HN2001000018A
Other languages
English (en)
Inventor
Chambers Robert James
Magee Thomas Victor
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of HN2001000018A publication Critical patent/HN2001000018A/es

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
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  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
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  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
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  • Virology (AREA)
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  • Hematology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
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  • Biomedical Technology (AREA)
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  • Urology & Nephrology (AREA)
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  • Vascular Medicine (AREA)
  • Biotechnology (AREA)
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Abstract

LA PRESENTE INVENCION ESTA RELACIONADA ESENCIALMENTE CON LOS CUATRO PRODUCTOS GENICOS DE LA CUARTA FAMILIA DE PDE4.
HN2001000018A 2000-01-31 2001-06-30 Carboxamidas de pirimidina utiles como inhibidores de isozimas pde4. HN2001000018A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17928200P 2000-01-31 2000-01-31

Publications (1)

Publication Number Publication Date
HN2001000018A true HN2001000018A (es) 2001-09-11

Family

ID=22655926

Family Applications (1)

Application Number Title Priority Date Filing Date
HN2001000018A HN2001000018A (es) 2000-01-31 2001-06-30 Carboxamidas de pirimidina utiles como inhibidores de isozimas pde4.

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US (1) US6740655B2 (es)
EP (1) EP1252157B1 (es)
JP (1) JP2003522165A (es)
KR (1) KR20020071029A (es)
CN (1) CN1404480A (es)
AP (1) AP2002002590A0 (es)
AR (1) AR027336A1 (es)
AT (1) ATE269860T1 (es)
AU (1) AU2700301A (es)
BG (1) BG106868A (es)
BR (1) BR0107934A (es)
CA (1) CA2396458C (es)
CO (1) CO5271669A1 (es)
CR (1) CR6714A (es)
CZ (1) CZ20022413A3 (es)
DE (1) DE60103976T2 (es)
DK (1) DK1252157T3 (es)
DZ (1) DZ3406A1 (es)
EA (1) EA005028B1 (es)
EE (1) EE200200426A (es)
ES (1) ES2223772T3 (es)
GE (1) GEP20043385B (es)
GT (1) GT200100023A (es)
HK (1) HK1054232A1 (es)
HN (1) HN2001000018A (es)
HU (1) HUP0204271A3 (es)
IL (1) IL150486A0 (es)
IS (1) IS6444A (es)
MA (1) MA26871A1 (es)
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NO (1) NO20023614L (es)
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SK (1) SK10342002A3 (es)
SV (1) SV2001000298A (es)
TN (1) TNSN01019A1 (es)
TR (1) TR200402292T4 (es)
UY (1) UY26570A1 (es)
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ZA (1) ZA200206034B (es)

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ES2165768B1 (es) 1999-07-14 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen.
EP1248597B1 (en) * 1999-12-24 2005-03-30 Glaxo Group Limited Pharmaceutical aerosol formulation of salmeterol and fluticasone propionate
US7776315B2 (en) 2000-10-31 2010-08-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmaceutical compositions based on anticholinergics and additional active ingredients
DE10110772A1 (de) * 2001-03-07 2002-09-12 Boehringer Ingelheim Pharma Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und PDE-IV-Inhibitoren
YU39503A (sh) 2000-11-22 2006-05-25 F. Hoffmann-La Roche Ag. Derivati pirimidina
US7250518B2 (en) 2001-01-31 2007-07-31 Pfizer Inc. Nicotinamide acids, amides, and their mimetics active as inhibitors of PDE4 isozymes
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