MA26871A1 - Pyrimidinecarboxamides utiles comme inhibiteurs d'isozymes pde4. - Google Patents

Pyrimidinecarboxamides utiles comme inhibiteurs d'isozymes pde4.

Info

Publication number
MA26871A1
MA26871A1 MA26749A MA26749A MA26871A1 MA 26871 A1 MA26871 A1 MA 26871A1 MA 26749 A MA26749 A MA 26749A MA 26749 A MA26749 A MA 26749A MA 26871 A1 MA26871 A1 MA 26871A1
Authority
MA
Morocco
Prior art keywords
chronic
pyrimidinecarboxamides
useful
inhibitors
pde4
Prior art date
Application number
MA26749A
Other languages
English (en)
Inventor
Robert James Chambers
Thomas Victor Magee
Anthony Marfat
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of MA26871A1 publication Critical patent/MA26871A1/fr

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
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  • General Chemical & Material Sciences (AREA)
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  • Diabetes (AREA)
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  • Pain & Pain Management (AREA)
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  • Dermatology (AREA)
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Abstract

DEPOSANT Société dite : PFIZER PRODUCTS INC. REVENDICATION DE PRIORITES US 31 Janvier 2000 60/179,282 Voir en annexe le titre de l'invention et le texte de l'abrégé "Pyrimidinecarboxamides utiles comme inhibiteurs d'isozymes PDE4" Il est décrit des composés de formule (1.0.0.), ainsi que l'utilité d'une composition pharmaceutique pour le traitement de maladies et affections inflammatoires, respiratoires et allergiques, notamment de l'asthme ; d'une maladie pulmonaire obstructrice chronique (COPD), comprenant la bronchite chronique, l'emphysème et la bronchiectasie; de la rhinite chronique , et de la sinusite chronique.
MA26749A 2000-01-31 2002-07-29 Pyrimidinecarboxamides utiles comme inhibiteurs d'isozymes pde4. MA26871A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17928200P 2000-01-31 2000-01-31

Publications (1)

Publication Number Publication Date
MA26871A1 true MA26871A1 (fr) 2004-12-20

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Family Applications (1)

Application Number Title Priority Date Filing Date
MA26749A MA26871A1 (fr) 2000-01-31 2002-07-29 Pyrimidinecarboxamides utiles comme inhibiteurs d'isozymes pde4.

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US (1) US6740655B2 (fr)
EP (1) EP1252157B1 (fr)
JP (1) JP2003522165A (fr)
KR (1) KR20020071029A (fr)
CN (1) CN1404480A (fr)
AP (1) AP2002002590A0 (fr)
AR (1) AR027336A1 (fr)
AT (1) ATE269860T1 (fr)
AU (1) AU2700301A (fr)
BG (1) BG106868A (fr)
BR (1) BR0107934A (fr)
CA (1) CA2396458C (fr)
CO (1) CO5271669A1 (fr)
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DK (1) DK1252157T3 (fr)
DZ (1) DZ3406A1 (fr)
EA (1) EA005028B1 (fr)
EE (1) EE200200426A (fr)
ES (1) ES2223772T3 (fr)
GE (1) GEP20043385B (fr)
GT (1) GT200100023A (fr)
HK (1) HK1054232A1 (fr)
HN (1) HN2001000018A (fr)
HU (1) HUP0204271A3 (fr)
IL (1) IL150486A0 (fr)
IS (1) IS6444A (fr)
MA (1) MA26871A1 (fr)
MX (1) MXPA02007465A (fr)
NO (1) NO20023614L (fr)
NZ (1) NZ519726A (fr)
OA (1) OA12170A (fr)
PA (1) PA8511301A1 (fr)
PE (1) PE20011059A1 (fr)
PL (1) PL357555A1 (fr)
PT (1) PT1252157E (fr)
SK (1) SK10342002A3 (fr)
SV (1) SV2001000298A (fr)
TN (1) TNSN01019A1 (fr)
TR (1) TR200402292T4 (fr)
UY (1) UY26570A1 (fr)
WO (1) WO2001057025A1 (fr)
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ES2165768B1 (es) 1999-07-14 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen.
WO2001047493A1 (fr) * 1999-12-24 2001-07-05 Glaxo Group Limited Formulation pharmaceutique en aerosol de salmeterol et de propionate de fluticasone
US7776315B2 (en) 2000-10-31 2010-08-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmaceutical compositions based on anticholinergics and additional active ingredients
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