DK1723135T3 - Kendte hydroxy-6-heteroarylphenanthridiner og deres anvendelse som pde4-inhibitorer - Google Patents
Kendte hydroxy-6-heteroarylphenanthridiner og deres anvendelse som pde4-inhibitorerInfo
- Publication number
- DK1723135T3 DK1723135T3 DK05716889.0T DK05716889T DK1723135T3 DK 1723135 T3 DK1723135 T3 DK 1723135T3 DK 05716889 T DK05716889 T DK 05716889T DK 1723135 T3 DK1723135 T3 DK 1723135T3
- Authority
- DK
- Denmark
- Prior art keywords
- heteroarylphenanthridines
- pde4 inhibitors
- known hydroxy
- hydroxy
- pde4
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/473—Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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- A61K31/50—Pyridazines; Hydrogenated pyridazines
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- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP04004973 | 2004-03-03 | ||
EP04106359 | 2004-12-07 | ||
PCT/EP2005/050931 WO2005085225A1 (en) | 2004-03-03 | 2005-03-02 | Novel hydroxy-6-heteroarylphenanthridines and their use as pde4 inhibitors |
Publications (2)
Publication Number | Publication Date |
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DK1723135T3 true DK1723135T3 (da) | 2013-09-02 |
DK1723135T5 DK1723135T5 (da) | 2013-09-16 |
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DK05716889.0T DK1723135T5 (da) | 2004-03-03 | 2005-03-02 | Ukendte hydroxy-6-heteroarylphenanthridiner og deres anvendelse som pde4-inhibitorer |
DK12196702T DK2589599T3 (da) | 2004-03-03 | 2005-03-02 | Hidtil ukendte hydroxy-6-heteroarylphenanthridiner og deres anvendelse som PDE4-inhibitorer |
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DK12196702T DK2589599T3 (da) | 2004-03-03 | 2005-03-02 | Hidtil ukendte hydroxy-6-heteroarylphenanthridiner og deres anvendelse som PDE4-inhibitorer |
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US (8) | US8003798B2 (da) |
EP (2) | EP1723135B1 (da) |
JP (2) | JP4801039B2 (da) |
KR (2) | KR101152439B1 (da) |
CN (6) | CN104817534A (da) |
AR (1) | AR049319A1 (da) |
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BR (1) | BRPI0508321B1 (da) |
CA (1) | CA2557752C (da) |
CO (1) | CO5700749A2 (da) |
CY (2) | CY1114319T1 (da) |
DK (2) | DK1723135T5 (da) |
EA (2) | EA017282B1 (da) |
ES (2) | ES2505473T3 (da) |
HK (4) | HK1207635A1 (da) |
HR (2) | HRP20130828T1 (da) |
IL (2) | IL177073A (da) |
ME (1) | ME01955B (da) |
MX (2) | MXPA06009695A (da) |
NO (2) | NO336538B1 (da) |
NZ (1) | NZ549108A (da) |
PL (2) | PL2589599T4 (da) |
PT (2) | PT1723135E (da) |
RS (2) | RS52916B (da) |
SG (1) | SG182194A1 (da) |
SI (2) | SI2589599T1 (da) |
TW (2) | TWI404704B (da) |
WO (1) | WO2005085225A1 (da) |
ZA (1) | ZA200606176B (da) |
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SG182194A1 (en) | 2004-03-03 | 2012-07-30 | Nycomed Gmbh | Novel hydroxy-6-heteroarylphenanthridines and their use as pde4 inhibitors |
ATE461189T1 (de) | 2005-02-01 | 2010-04-15 | Nycomed Gmbh | Neue 6-pyridylphenanthridine |
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