FR18C1036I2 - Derives de dioxa-bicyclo[3.2.1.]octane-2,3,4-triol - Google Patents

Derives de dioxa-bicyclo[3.2.1.]octane-2,3,4-triol

Info

Publication number
FR18C1036I2
FR18C1036I2 FR18C1036C FR18C1036C FR18C1036I2 FR 18C1036 I2 FR18C1036 I2 FR 18C1036I2 FR 18C1036 C FR18C1036 C FR 18C1036C FR 18C1036 C FR18C1036 C FR 18C1036C FR 18C1036 I2 FR18C1036 I2 FR 18C1036I2
Authority
FR
France
Prior art keywords
dioxa
bicyclo
octane
triol derivatives
triol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
FR18C1036C
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English (en)
French (fr)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41208284&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR18C1036(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of FR18C1036I1 publication Critical patent/FR18C1036I1/fr
Application granted granted Critical
Publication of FR18C1036I2 publication Critical patent/FR18C1036I2/fr
Active legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H9/00—Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical
    • C07H9/02—Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical the hetero ring containing only oxygen as ring hetero atoms
    • C07H9/04—Cyclic acetals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Biochemistry (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FR18C1036C 2008-08-28 2018-08-24 Derives de dioxa-bicyclo[3.2.1.]octane-2,3,4-triol Active FR18C1036I2 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US9247008P 2008-08-28 2008-08-28
US22721209P 2009-07-21 2009-07-21
PCT/IB2009/053626 WO2010023594A1 (en) 2008-08-28 2009-08-17 Dioxa-bicyclo[3.2.1.]octane-2,3,4-triol derivatives

Publications (2)

Publication Number Publication Date
FR18C1036I1 FR18C1036I1 (pt) 2018-10-05
FR18C1036I2 true FR18C1036I2 (fr) 2020-07-24

Family

ID=41208284

Family Applications (1)

Application Number Title Priority Date Filing Date
FR18C1036C Active FR18C1036I2 (fr) 2008-08-28 2018-08-24 Derives de dioxa-bicyclo[3.2.1.]octane-2,3,4-triol

Country Status (47)

Country Link
US (1) US8080580B2 (pt)
EP (1) EP2334687B9 (pt)
JP (1) JP4825322B1 (pt)
KR (2) KR101446454B1 (pt)
CN (2) CN102149717B (pt)
AP (1) AP2728A (pt)
AR (1) AR073138A1 (pt)
AT (1) ATE540040T1 (pt)
AU (1) AU2009286380B2 (pt)
BR (1) BRPI0918841B8 (pt)
CA (1) CA2733795C (pt)
CL (1) CL2011000394A1 (pt)
CO (1) CO6341636A2 (pt)
CR (1) CR20110077A (pt)
CY (2) CY1112497T1 (pt)
DK (1) DK2334687T5 (pt)
DO (1) DOP2011000058A (pt)
EA (1) EA018492B1 (pt)
EC (1) ECSP11010854A (pt)
ES (1) ES2380408T3 (pt)
FR (1) FR18C1036I2 (pt)
GE (1) GEP20135803B (pt)
HK (2) HK1156616A1 (pt)
HN (1) HN2009001652A (pt)
HR (1) HRP20120104T1 (pt)
HU (1) HUS1800031I1 (pt)
IL (2) IL211226A (pt)
LT (1) LTC2334687I2 (pt)
MA (1) MA32590B1 (pt)
ME (1) ME01285A (pt)
MX (1) MX2011002166A (pt)
MY (1) MY155418A (pt)
NI (1) NI201100043A (pt)
NL (1) NL300943I2 (pt)
NO (1) NO2018019I2 (pt)
NZ (1) NZ591027A (pt)
PA (1) PA8840801A1 (pt)
PE (1) PE20110288A1 (pt)
PL (1) PL2334687T3 (pt)
PT (1) PT2334687E (pt)
RS (1) RS52236B (pt)
SI (1) SI2334687T1 (pt)
SV (1) SV2011003842A (pt)
TW (1) TWI387598B (pt)
UY (1) UY32073A (pt)
WO (1) WO2010023594A1 (pt)
ZA (1) ZA201101341B (pt)

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