FR16C0031I1 - - Google Patents

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Publication number
FR16C0031I1
FR16C0031I1 FR16C0031C FR16C0031I1 FR 16C0031 I1 FR16C0031 I1 FR 16C0031I1 FR 16C0031 C FR16C0031 C FR 16C0031C FR 16C0031 I1 FR16C0031 I1 FR 16C0031I1
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FR
France
Prior art keywords
hiv
mercaptoacetanilides
conr
triazolyl
useful
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English (en)
French (fr)
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36000576&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR16C0031(I1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of FR16C0031I1 publication Critical patent/FR16C0031I1/fr
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Publication of FR16C0031I2 publication Critical patent/FR16C0031I2/fr
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/101,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/12Oxygen or sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41961,2,4-Triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/101,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/14Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Road Signs Or Road Markings (AREA)
  • Pens And Brushes (AREA)
FR16C0031C 2004-08-25 2016-07-29 S-triazolyl alpha -mercaptoacetanilides en tant qu'inhibiteurs de la transcriptase inverse du vih Active FR16C0031I2 (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US60421904P 2004-08-25 2004-08-25
US60422004P 2004-08-25 2004-08-25
US68635105P 2005-05-31 2005-05-31
EP05790722A EP1789039B1 (en) 2004-08-25 2005-08-25 S-triazolyl alpha -mercaptoacetanildes as inhibitors of hiv reverse transcriptase

Publications (2)

Publication Number Publication Date
FR16C0031I1 true FR16C0031I1 (enrdf_load_stackoverflow) 2016-09-23
FR16C0031I2 FR16C0031I2 (fr) 2017-03-31

Family

ID=36000576

Family Applications (1)

Application Number Title Priority Date Filing Date
FR16C0031C Active FR16C0031I2 (fr) 2004-08-25 2016-07-29 S-triazolyl alpha -mercaptoacetanilides en tant qu'inhibiteurs de la transcriptase inverse du vih

Country Status (31)

Country Link
US (8) US7947721B2 (enrdf_load_stackoverflow)
EP (5) EP2433633A1 (enrdf_load_stackoverflow)
JP (2) JP4952943B2 (enrdf_load_stackoverflow)
KR (1) KR101241716B1 (enrdf_load_stackoverflow)
CN (2) CN101083987B (enrdf_load_stackoverflow)
AT (2) ATE528001T1 (enrdf_load_stackoverflow)
AU (2) AU2005280130C9 (enrdf_load_stackoverflow)
BR (2) BRPI0520870B8 (enrdf_load_stackoverflow)
CA (1) CA2578068C (enrdf_load_stackoverflow)
CY (2) CY1112221T1 (enrdf_load_stackoverflow)
DK (1) DK2135608T3 (enrdf_load_stackoverflow)
EA (2) EA015846B1 (enrdf_load_stackoverflow)
EC (1) ECSP077322A (enrdf_load_stackoverflow)
ES (2) ES2380604T3 (enrdf_load_stackoverflow)
FR (1) FR16C0031I2 (enrdf_load_stackoverflow)
HR (1) HRP20130075T1 (enrdf_load_stackoverflow)
HU (1) HUS1600034I1 (enrdf_load_stackoverflow)
IL (3) IL181523A (enrdf_load_stackoverflow)
IN (1) IN2014CN03762A (enrdf_load_stackoverflow)
LT (1) LTC2135608I2 (enrdf_load_stackoverflow)
LU (1) LU93169I2 (enrdf_load_stackoverflow)
ME (1) ME01512B (enrdf_load_stackoverflow)
MX (1) MX2007002236A (enrdf_load_stackoverflow)
NL (1) NL300825I2 (enrdf_load_stackoverflow)
NZ (2) NZ581376A (enrdf_load_stackoverflow)
PL (1) PL2135608T3 (enrdf_load_stackoverflow)
PT (1) PT2135608E (enrdf_load_stackoverflow)
RS (1) RS52632B (enrdf_load_stackoverflow)
SG (2) SG155246A1 (enrdf_load_stackoverflow)
SI (1) SI2135608T1 (enrdf_load_stackoverflow)
WO (1) WO2006026356A2 (enrdf_load_stackoverflow)

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Also Published As

Publication number Publication date
CY2016028I1 (el) 2016-12-14
US20150094284A1 (en) 2015-04-02
US20080176850A1 (en) 2008-07-24
MX2007002236A (es) 2007-07-09
US8946273B2 (en) 2015-02-03
EA200700488A1 (ru) 2007-08-31
BRPI0514630A (pt) 2008-06-17
US20180002296A1 (en) 2018-01-04
IN2014CN03762A (enrdf_load_stackoverflow) 2015-09-25
AU2005280130B2 (en) 2009-09-10
EP2135608A1 (en) 2009-12-23
US8003681B2 (en) 2011-08-23
RS52632B (en) 2013-06-28
CY2016028I2 (el) 2016-12-14
LTPA2016024I1 (lt) 2016-09-12
BRPI0520870B1 (pt) 2020-11-10
US8481581B2 (en) 2013-07-09
NZ553534A (en) 2010-10-29
IL181523A (en) 2013-12-31
DK2135608T3 (da) 2012-01-23
NL300825I2 (enrdf_load_stackoverflow) 2017-01-24
BRPI0514630B1 (pt) 2020-09-15
US20110313157A1 (en) 2011-12-22
CN101083987A (zh) 2007-12-05
BRPI0520870B8 (pt) 2021-05-25
EP2402011A1 (en) 2012-01-04
PL2135608T3 (pl) 2012-07-31
US20100069645A1 (en) 2010-03-18
US20100081827A1 (en) 2010-04-01
BRPI0514630B8 (pt) 2021-05-25
EA014737B1 (ru) 2011-02-28
AU2005280130C9 (en) 2010-03-04
JP2012077088A (ja) 2012-04-19
CY1112221T1 (el) 2015-12-09
ES2374773T3 (es) 2012-02-21
ATE540677T1 (de) 2012-01-15
US20110190491A1 (en) 2011-08-04
EP2135608B8 (en) 2012-03-21
ECSP077322A (es) 2007-04-26
ATE528001T1 (de) 2011-10-15
AU2009217458B2 (en) 2009-11-19
EA015846B1 (ru) 2011-12-30
JP5457472B2 (ja) 2014-04-02
US8252828B2 (en) 2012-08-28
SI2135608T1 (sl) 2012-03-30
CN101817793B (zh) 2014-01-08
WO2006026356A3 (en) 2006-08-10
HUS1600034I1 (hu) 2016-09-28
EP2609917A1 (en) 2013-07-03
IL219131A0 (en) 2012-06-28
KR20070054694A (ko) 2007-05-29
CA2578068A1 (en) 2006-03-09
EP1789039A2 (en) 2007-05-30
LU93169I2 (fr) 2016-10-10
EA200901186A1 (ru) 2010-04-30
AU2009217458A1 (en) 2009-10-15
EP1789039B1 (en) 2012-01-11
US20120283301A1 (en) 2012-11-08
EP2135608B1 (en) 2011-10-12
JP2008510828A (ja) 2008-04-10
AU2005280130A1 (en) 2006-03-09
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LTC2135608I2 (lt) 2017-07-25
IL181523A0 (en) 2007-07-04
ME01512B (me) 2014-04-20
EP1789039A4 (en) 2009-08-05
JP4952943B2 (ja) 2012-06-13
KR101241716B1 (ko) 2013-03-08
NZ581376A (en) 2011-05-27
SG185992A1 (en) 2012-12-28
HK1133582A1 (en) 2010-04-01
IL201546A (en) 2013-10-31
WO2006026356A2 (en) 2006-03-09
HRP20130075T1 (hr) 2013-02-28
CN101817793A (zh) 2010-09-01
CN101083987B (zh) 2011-01-26
PT2135608E (pt) 2012-01-13
US20100267724A2 (en) 2010-10-21
SG155246A1 (en) 2009-09-30
EP2433633A1 (en) 2012-03-28
FR16C0031I2 (fr) 2017-03-31
US7947721B2 (en) 2011-05-24
AU2005280130C1 (en) 2010-02-18
AU2009217458A8 (en) 2009-10-29
CA2578068C (en) 2011-08-09
EP2402011B1 (en) 2012-11-14

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