FI973750A0 - Framställnig och kristallina former av 2-metyltienobensodiazepin - Google Patents

Framställnig och kristallina former av 2-metyltienobensodiazepin

Info

Publication number
FI973750A0
FI973750A0 FI973750A FI973750A FI973750A0 FI 973750 A0 FI973750 A0 FI 973750A0 FI 973750 A FI973750 A FI 973750A FI 973750 A FI973750 A FI 973750A FI 973750 A0 FI973750 A0 FI 973750A0
Authority
FI
Finland
Prior art keywords
methylthienobenzodiazepine
preparation
crystalline forms
crystalline
forms
Prior art date
Application number
FI973750A
Other languages
English (en)
Finnish (fi)
Other versions
FI973750A (sv
Inventor
Charles Arthur Bunnell
Barry Arnold Hendriksen
Original Assignee
Lilly Co Eli
Lilly Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23621056&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI973750(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli, Lilly Industries Ltd filed Critical Lilly Co Eli
Publication of FI973750A publication Critical patent/FI973750A/sv
Publication of FI973750A0 publication Critical patent/FI973750A0/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicinal Preparation (AREA)
FI973750A 1995-03-24 1997-09-22 Framställnig och kristallina former av 2-metyltienobensodiazepin FI973750A0 (sv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40956695A 1995-03-24 1995-03-24
PCT/US1996/003917 WO1996030375A1 (en) 1995-03-24 1996-03-22 Process and crystal forms of 2-methyl-thieno-benzodiazepine

Publications (2)

Publication Number Publication Date
FI973750A FI973750A (sv) 1997-09-22
FI973750A0 true FI973750A0 (sv) 1997-09-22

Family

ID=23621056

Family Applications (1)

Application Number Title Priority Date Filing Date
FI973750A FI973750A0 (sv) 1995-03-24 1997-09-22 Framställnig och kristallina former av 2-metyltienobensodiazepin

Country Status (49)

Country Link
US (1) US5736541A (sv)
EP (3) EP0733635B1 (sv)
JP (1) JPH11502535A (sv)
KR (1) KR100399688B1 (sv)
CN (1) CN1065536C (sv)
AP (1) AP828A (sv)
AR (2) AR010448A1 (sv)
AT (4) AT406771B (sv)
AU (1) AU706471B2 (sv)
BG (1) BG62619B1 (sv)
BR (1) BR9607790A (sv)
CA (1) CA2214005C (sv)
CH (1) CH690579A5 (sv)
CO (1) CO4650278A1 (sv)
CZ (1) CZ292688B6 (sv)
DE (4) DE19681286T1 (sv)
DK (4) DK0733635T3 (sv)
EA (1) EA000149B1 (sv)
EE (1) EE03489B1 (sv)
EG (1) EG23659A (sv)
ES (3) ES2208220T3 (sv)
FI (1) FI973750A0 (sv)
GB (1) GB2313835B (sv)
HK (1) HK1013988A1 (sv)
HU (1) HU224989B1 (sv)
IL (1) IL117610A (sv)
IS (1) IS1896B (sv)
LT (1) LT4349B (sv)
LU (1) LU90096B1 (sv)
LV (1) LV12018B (sv)
MY (1) MY114701A (sv)
NO (1) NO314663B1 (sv)
NZ (1) NZ306110A (sv)
OA (1) OA10510A (sv)
PA (1) PA8353701A1 (sv)
PE (1) PE44897A1 (sv)
PL (1) PL183723B1 (sv)
PT (3) PT1445259E (sv)
RO (1) RO118872B1 (sv)
SE (1) SE9703205D0 (sv)
SI (4) SI0733635T1 (sv)
SK (1) SK284143B6 (sv)
SV (1) SV1996000031A (sv)
TR (1) TR199701017T1 (sv)
TW (2) TW442488B (sv)
UA (1) UA44765C2 (sv)
WO (1) WO1996030375A1 (sv)
YU (1) YU49478B (sv)
ZA (2) ZA962342B (sv)

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Also Published As

Publication number Publication date
SI1445259T1 (sl) 2006-10-31
FI973750A (sv) 1997-09-22
ES2159346T3 (es) 2001-10-01
LT4349B (lt) 1998-05-25
AU5427996A (en) 1996-10-16
HK1013988A1 (en) 1999-09-17
IS4564A (is) 1997-09-22
BR9607790A (pt) 1998-07-07
DK1445259T3 (da) 2006-10-16
AT406771B (de) 2000-08-25
SE9703205L (sv) 1997-09-05
ZA962342B (en) 1997-09-22
IL117610A0 (en) 1996-07-23
LV12018B (en) 1998-09-20
EP1445259A1 (en) 2004-08-11
US5736541A (en) 1998-04-07
GB2313835A (en) 1997-12-10
MX9707183A (es) 1997-11-29
KR19980703188A (ko) 1998-10-15
ES2208220T3 (es) 2004-06-16
CN1179160A (zh) 1998-04-15
YU17796A (sh) 1999-03-04
GB9719819D0 (en) 1997-11-19
JPH11502535A (ja) 1999-03-02
EP1445259B1 (en) 2006-06-28
AU706471B2 (en) 1999-06-17
BG101900A (en) 1999-03-31
ATA902196A (de) 2000-01-15
CH690579A5 (de) 2000-10-31
CZ292688B6 (cs) 2003-11-12
CZ300097A3 (en) 1997-12-17
UA44765C2 (uk) 2002-03-15
LV12018A (lv) 1998-04-20
OA10510A (en) 2002-04-24
DE69630324D1 (de) 2003-11-13
DE69614426D1 (de) 2001-09-20
PL322501A1 (en) 1998-02-02
ATE331719T1 (de) 2006-07-15
TR199701017T1 (xx) 1998-01-21
PT1095941E (pt) 2004-02-27
HUP9802824A3 (en) 2000-01-28
ES2266719T3 (es) 2007-03-01
CN1065536C (zh) 2001-05-09
CA2214005A1 (en) 1996-10-03
DE69636313D1 (de) 2006-08-10
HU224989B1 (en) 2006-05-29
NO974365L (no) 1997-09-22
DE69614426T2 (de) 2002-05-23
EA199700262A1 (ru) 1998-02-26
SK121897A3 (en) 1998-03-04
LT97148A (en) 1998-01-26
LU90096B1 (fr) 1997-07-22
ATE204280T1 (de) 2001-09-15
SI1095941T1 (en) 2003-12-31
CO4650278A1 (es) 1998-09-03
EE9700232A (et) 1998-04-15
PT733635E (pt) 2001-12-28
CA2214005C (en) 2001-07-03
EP0733635B1 (en) 2001-08-16
DK1095941T3 (da) 2004-02-16
BG62619B1 (bg) 2000-03-31
YU49478B (sh) 2006-05-25
EP0733635A1 (en) 1996-09-25
GB2313835B (en) 1998-09-16
TW513432B (en) 2002-12-11
SI9620040A (sl) 1998-06-30
IL117610A (en) 2001-08-26
EG23659A (en) 2007-03-26
SI0733635T1 (en) 2002-06-30
KR100399688B1 (ko) 2004-02-18
AP828A (en) 2000-04-28
ZA962344B (en) 1997-09-22
DE69630324T2 (de) 2004-07-29
SE9703205D0 (sv) 1997-09-05
EA000149B1 (ru) 1998-10-29
DK108997A (da) 1997-11-12
SI9620040B (sl) 2002-02-28
MY114701A (en) 2002-12-31
DE69636313T2 (de) 2007-05-31
HUP9802824A2 (hu) 1999-06-28
ATE251627T1 (de) 2003-10-15
PE44897A1 (es) 1997-10-22
PL183723B1 (pl) 2002-07-31
IS1896B (is) 2003-10-20
AR002719A1 (es) 1998-04-29
EP1095941B1 (en) 2003-10-08
SK284143B6 (sk) 2004-10-05
TW442488B (en) 2001-06-23
DK0733635T3 (da) 2001-10-08
AP9701065A0 (en) 1997-10-31
AR010448A1 (es) 2000-06-28
RO118872B1 (ro) 2003-12-30
PA8353701A1 (es) 1998-09-18
PT1445259E (pt) 2006-10-31
DE19681286T1 (de) 1998-04-02
NO314663B1 (no) 2003-04-28
NZ306110A (en) 1998-09-24
SV1996000031A (es) 1998-03-27
NO974365D0 (no) 1997-09-22
WO1996030375A1 (en) 1996-10-03
EE03489B1 (et) 2001-08-15
EP1095941A1 (en) 2001-05-02

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