FI108296B - Menetelmä terapeuttisesti aktiivisten 1,6-diatsabisyklo[3.2.1]oktaani- ja 1,4-diatsabisyklo[3.3.1]nonaanijohdannaisten valmistamiseksi - Google Patents

Menetelmä terapeuttisesti aktiivisten 1,6-diatsabisyklo[3.2.1]oktaani- ja 1,4-diatsabisyklo[3.3.1]nonaanijohdannaisten valmistamiseksi Download PDF

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Publication number
FI108296B
FI108296B FI946140A FI946140A FI108296B FI 108296 B FI108296 B FI 108296B FI 946140 A FI946140 A FI 946140A FI 946140 A FI946140 A FI 946140A FI 108296 B FI108296 B FI 108296B
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FI
Finland
Prior art keywords
formula
diazabicyclo
compounds
compound
substance
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FI946140A
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English (en)
Finnish (fi)
Swedish (sv)
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FI946140A (fi
FI946140A0 (fi
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Jr Harry R Howard
Kevin D Shenk
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Pfizer
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Publication of FI108296B publication Critical patent/FI108296B/fi

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
FI946140A 1993-12-29 1994-12-28 Menetelmä terapeuttisesti aktiivisten 1,6-diatsabisyklo[3.2.1]oktaani- ja 1,4-diatsabisyklo[3.3.1]nonaanijohdannaisten valmistamiseksi FI108296B (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17503493A 1993-12-29 1993-12-29
US17503493 1993-12-29

Publications (3)

Publication Number Publication Date
FI946140A0 FI946140A0 (fi) 1994-12-28
FI946140A FI946140A (fi) 1995-06-30
FI108296B true FI108296B (fi) 2001-12-31

Family

ID=22638565

Family Applications (1)

Application Number Title Priority Date Filing Date
FI946140A FI108296B (fi) 1993-12-29 1994-12-28 Menetelmä terapeuttisesti aktiivisten 1,6-diatsabisyklo[3.2.1]oktaani- ja 1,4-diatsabisyklo[3.3.1]nonaanijohdannaisten valmistamiseksi

Country Status (26)

Country Link
US (2) US5854239A (ru)
EP (1) EP0737194B1 (ru)
JP (1) JP2895630B2 (ru)
KR (1) KR100197454B1 (ru)
CN (1) CN1046515C (ru)
AT (1) ATE177099T1 (ru)
AU (1) AU699465B2 (ru)
BR (1) BR9408450A (ru)
CA (1) CA2180263C (ru)
CO (1) CO4230019A1 (ru)
CZ (1) CZ282567B6 (ru)
DE (1) DE69416869T2 (ru)
DK (1) DK0737194T3 (ru)
ES (1) ES2127946T3 (ru)
FI (1) FI108296B (ru)
GR (1) GR3029853T3 (ru)
HU (1) HUT74682A (ru)
IL (1) IL112118A (ru)
NO (1) NO305600B1 (ru)
NZ (1) NZ274915A (ru)
PE (1) PE49395A1 (ru)
PL (1) PL179435B1 (ru)
RU (1) RU2124014C1 (ru)
TW (1) TW369526B (ru)
WO (1) WO1995018129A1 (ru)
ZA (1) ZA9410339B (ru)

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FR2844273B1 (fr) 2002-09-05 2008-04-04 Aventis Pharma Sa Nouveaux composes heterocycliques, procede et intermediaires de preparation et utilisation comme medicament, notamment comme inhibiteurs de beta-lactamases et anti-bacteriens.
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Also Published As

Publication number Publication date
IL112118A0 (en) 1995-03-15
NO305600B1 (no) 1999-06-28
FI946140A (fi) 1995-06-30
DE69416869D1 (de) 1999-04-08
BR9408450A (pt) 1997-08-05
FI946140A0 (fi) 1994-12-28
US5854239A (en) 1998-12-29
HU9601790D0 (en) 1996-09-30
KR100197454B1 (ko) 1999-06-15
PE49395A1 (es) 1996-01-06
CN1046515C (zh) 1999-11-17
JP2895630B2 (ja) 1999-05-24
CA2180263C (en) 2000-05-16
NO962742D0 (no) 1996-06-28
TW369526B (en) 1999-09-11
CZ282567B6 (cs) 1997-08-13
EP0737194B1 (en) 1999-03-03
CN1139434A (zh) 1997-01-01
PL179435B1 (pl) 2000-09-29
DE69416869T2 (de) 1999-07-01
WO1995018129A1 (en) 1995-07-06
CO4230019A1 (es) 1995-10-19
NZ274915A (en) 1997-11-24
JPH09500904A (ja) 1997-01-28
AU8002194A (en) 1995-07-17
NO962742L (no) 1996-06-28
PL315193A1 (en) 1996-10-14
GR3029853T3 (en) 1999-07-30
HUT74682A (en) 1997-01-28
DK0737194T3 (da) 1999-09-27
US6110919A (en) 2000-08-29
AU699465B2 (en) 1998-12-03
ES2127946T3 (es) 1999-05-01
ZA9410339B (en) 1996-06-28
CZ188696A3 (en) 1996-10-16
EP0737194A1 (en) 1996-10-16
IL112118A (en) 1998-10-30
ATE177099T1 (de) 1999-03-15
RU2124014C1 (ru) 1998-12-27

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