ES480113A1 - Procedimiento para la preparacion de nuevos derivados de 2- iminoimidazolidina. - Google Patents
Procedimiento para la preparacion de nuevos derivados de 2- iminoimidazolidina.Info
- Publication number
- ES480113A1 ES480113A1 ES480113A ES480113A ES480113A1 ES 480113 A1 ES480113 A1 ES 480113A1 ES 480113 A ES480113 A ES 480113A ES 480113 A ES480113 A ES 480113A ES 480113 A1 ES480113 A1 ES 480113A1
- Authority
- ES
- Spain
- Prior art keywords
- imino
- imidazolidine
- derivatives
- intermediates
- processes
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C335/40—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of thiourea or isothiourea groups further bound to other hetero atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
- Indole Compounds (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Abstract
Procedimiento para la preparación de nuevos derivados de 2- iminoimidazolidina los productos del procedimiento y sus sales aceptables en farmacia pueden utilizarse como medicamentos, or ejemplo en forma de preparados farmacéuticos que los contengan o sus sales, en mezcla con un material de vehículo inerte y farmacéutico, orgánico o inorgánico, apto para administración enteral o parental tal como, por ejemplo, agua, gelatina, goma arábiga, lactosa, almidón, estearato de magnesio, talco, aceites vegetales, polialquilenglicoles, vaselina, etc. los preparados farmacéuticos pueden adoptar forma sólida, por ejemplo de pastillas, gráficas supositorios o capsulas, o forma líquida, por ejemplo de soluciones suspensiones o emulsiones. Puedes opcionalmente, esterilizarse y/o contener coadyuvantes o emulgentes sales para modificar la presión osmótica o tampones. Adicionalmente pueden contener también otras sustancias terapéuticamente valiosas.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
LU78467 | 1977-11-07 | ||
CH966878 | 1978-09-15 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES480113A1 true ES480113A1 (es) | 1980-04-01 |
Family
ID=25705131
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES480112A Expired ES480112A1 (es) | 1977-11-07 | 1979-04-30 | Procedimiento para la preparacion de nuevos derivados de 2- iminoimidazolidina. |
ES480111A Expired ES480111A1 (es) | 1977-11-07 | 1979-04-30 | Procedimiento para la preparacion de nuevos derivados de 2- iminoimidazolidina. |
ES480113A Expired ES480113A1 (es) | 1977-11-07 | 1979-04-30 | Procedimiento para la preparacion de nuevos derivados de 2- iminoimidazolidina. |
Family Applications Before (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES480112A Expired ES480112A1 (es) | 1977-11-07 | 1979-04-30 | Procedimiento para la preparacion de nuevos derivados de 2- iminoimidazolidina. |
ES480111A Expired ES480111A1 (es) | 1977-11-07 | 1979-04-30 | Procedimiento para la preparacion de nuevos derivados de 2- iminoimidazolidina. |
Country Status (30)
Country | Link |
---|---|
US (3) | US4244957A (es) |
EP (1) | EP0002010B1 (es) |
JP (1) | JPS5473779A (es) |
AR (1) | AR223656A1 (es) |
AT (1) | AT371112B (es) |
AU (1) | AU4132478A (es) |
BR (1) | BR7807317A (es) |
CA (1) | CA1106847A (es) |
CS (1) | CS212309B2 (es) |
DD (1) | DD139847A5 (es) |
DE (2) | DE2847766A1 (es) |
DK (1) | DK494978A (es) |
EG (1) | EG13665A (es) |
ES (3) | ES480112A1 (es) |
FI (1) | FI783393A (es) |
FR (1) | FR2407919A1 (es) |
GB (2) | GB2008579B (es) |
IL (1) | IL55832A0 (es) |
IT (1) | IT1160046B (es) |
MC (1) | MC1223A1 (es) |
MT (1) | MTP837B (es) |
NL (1) | NL7811070A (es) |
NO (1) | NO783719L (es) |
NZ (1) | NZ188798A (es) |
OA (1) | OA06084A (es) |
PL (1) | PL210759A1 (es) |
PT (1) | PT68752A (es) |
RO (1) | RO76151A (es) |
SE (1) | SE7811455L (es) |
SU (2) | SU831073A3 (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4287201A (en) * | 1980-03-03 | 1981-09-01 | Merck & Co., Inc. | Anovulatory method and chicken feed compositions |
CA1175434A (en) * | 1980-09-10 | 1984-10-02 | Hoffmann-La Roche Limited | ¬(2-phenylamino-1-imidazolidinyloxy)methyl| pyridine 1-oxide derivatives |
DE3642453A1 (de) * | 1986-12-12 | 1988-06-23 | Bayer Ag | Neue, fluor enthaltende 5-trihalogenmethyl-isoxazole und ein verfahren zu deren herstellung |
DE19514579A1 (de) * | 1995-04-20 | 1996-10-24 | Boehringer Ingelheim Kg | Verwendung von alpha¶1¶¶L¶-Agonisten zur Behandlung der Harninkontinenz |
WO2002004421A2 (en) * | 2000-07-07 | 2002-01-17 | Medicure International Inc. | Pyridoxine and pyridoxal analogues: cardiovascular therapeutics |
GB2374251A (en) * | 2001-04-04 | 2002-10-09 | Secr Defence | Base station transmitter |
WO2003042193A1 (en) * | 2001-11-09 | 2003-05-22 | Geneva Pharmaceuticals, Inc. | Process for preparing 5-methylisoxazole-4-carboxylic-(4'-trifluoromethyl)-anilide |
US6703409B2 (en) | 2002-01-31 | 2004-03-09 | Boehringer Ingelheim Pharma Gmbh & Co Kg | 2′-Halo-3′,5′-dialkoxyphen-1′-yl-imino-2-imidazolidine and the use thereof as a drug |
EP1333028A1 (en) * | 2002-01-31 | 2003-08-06 | Boehringer Ingelheim Pharma GmbH & Co.KG | 2'-Halo-3',5'-dialkoxyphen-1'-yl-imino-2-imidazolidine derivatives and the use thereof for the treatment of urinary incontinence |
AU2009282747B2 (en) | 2008-08-22 | 2015-04-02 | Takeda Pharmaceutical Company Limited | Polymeric benzyl carbonate-derivatives |
Family Cites Families (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1670274U (de) | 1953-07-30 | 1954-01-14 | Leo Schirk | Stahlblechschalttafel. |
DE1815788U (de) | 1959-12-12 | 1960-07-28 | Walther Loeffler | Ventil fuer spuelbecken, waschbecken, bidets, wannen. |
US3236857A (en) | 1961-10-09 | 1966-02-22 | Boehringer Sohn Ingelheim | 2-(phenyl-amino)-1, 3-diazacyclopentene-(2) substitution products |
NL123037C (es) | 1963-10-04 | |||
DE1545628A1 (de) | 1965-10-01 | 1970-06-25 | Boehringer Sohn Ingelheim | Verfahren zur Herstellung von blutdrucksenkend und sedativ wirksamen Derivaten des 2-(2-Halogenanilino)-1,3-diazacyclopentens-(2) |
DE1670274A1 (de) * | 1966-10-31 | 1970-07-16 | Boehringer Sohn Ingelheim | Neues Verfahren zur Herstellung von 2-Arylamino-1,3-diazacycloalkenen-(2) |
DE1670230A1 (de) | 1967-05-26 | 1971-01-21 | Boehringer Sohn Ingelheim | Neues Verfahren zur Herstellung von in 2-Stellung substituierten 1,3-Diazacycloalkenen(2) |
ES352379A1 (es) | 1967-05-26 | 1969-08-01 | Boehringer Sohn Ingelheim | Procedimiento para la preparacion de 1,3-diazaciclopenteno-(2) sustituido en posicion 2. |
US3454301A (en) * | 1967-09-29 | 1969-07-08 | John W Lehmann | Glare-inhibiting device |
GB1246312A (en) * | 1968-01-10 | 1971-09-15 | Syntex Energy Res Inc | 4,5-substituted n-oxy and hydroxy hydroimidazoles |
DE1770872A1 (de) | 1968-08-26 | 1972-01-13 | Dresden Arzneimittel | Verfahren zur Herstellung von Imidazolin-2-Derivaten |
BE721781A (es) | 1968-10-03 | 1969-04-03 | ||
BE759048A (fr) * | 1969-11-17 | 1971-05-17 | Boehringer Sohn Ingelheim | Nouvelles n-aminoalcoyl-arylamino-imidazolines-(2) substituees et procedes pour les fabriquer |
DE2016290A1 (de) * | 1970-04-06 | 1971-11-04 | C H Boehrmger Sohn, 6507 Ingel heim | Substituierte N Hydroxylakyl 2 arylamine) imidazoline (2) und Verfahren zu deren Herstellung |
US3740412A (en) * | 1970-04-08 | 1973-06-19 | Synvar Ass | Imidazoline-3-oxide-1-oxyl derivatives |
DE2038107A1 (de) * | 1970-07-31 | 1972-02-10 | Henkel & Cie Gmbh | Fluessige,gegebenenfalls als Wasch- oder Reinigungsmittel brauchbare stabilisierte Enzympraeparate |
US3799942A (en) * | 1971-04-12 | 1974-03-26 | Syva Corp | 4,5-substituted n-oxy and hydroxy hydroimidazoles |
BE787477A (fr) * | 1971-08-12 | 1973-02-12 | Bayer Ag | 1-phenyl-2-imino-imidazolidines, leur procede de preparation etleur application comme repulsifs a l'egard des oiseaux |
DE2457979A1 (de) | 1974-12-07 | 1976-06-16 | Beiersdorf Ag | 2-n-aryl-hydroxyamino-imidazoline-(2) und verfahren zu deren herstellung |
DE2523103C3 (de) * | 1975-05-24 | 1979-11-29 | C.H. Boehringer Sohn, 6507 Ingelheim | Substituierte 2-[N-Progargyl-N-(2-chlorphenyl)amino] -imidazoline-^), deren Säureadditionssalze, Verfahren zu ihrer Herstellung und deren Verwendung |
AT339897B (de) * | 1975-09-25 | 1977-11-10 | Chemie Linz Ag | Verfahren zur herstellung des neuen 1-benzoyl-2- (2',6'-dichlorphenylamino) -2-imidazolins und von dessen salzen |
DE2626128A1 (de) * | 1976-06-11 | 1977-12-22 | Beiersdorf Ag | N-substituierte benzimidazolin-2-one und verfahren zu deren herstellung |
DE2709720A1 (de) * | 1977-03-05 | 1978-09-07 | Beiersdorf Ag | N-substituierte 2-arylamino-imidazoline-(2), verfahren zu deren herstellung und neue hydroxylamine als zwischenprodukte |
US4131679A (en) * | 1977-07-26 | 1978-12-26 | Sandoz, Inc. | Substituted 4-hydroxy pyridones |
DE2811847A1 (de) * | 1978-03-17 | 1979-09-20 | Lentia Gmbh | Neue arylaminoimidazolinderivate, deren herstellung und verwendung als arzneimittel |
-
1978
- 1978-10-26 MT MT837A patent/MTP837B/xx unknown
- 1978-10-31 IL IL7855832A patent/IL55832A0/xx unknown
- 1978-11-01 NZ NZ188798A patent/NZ188798A/xx unknown
- 1978-11-02 FR FR7831026A patent/FR2407919A1/fr not_active Withdrawn
- 1978-11-02 OA OA56651A patent/OA06084A/xx unknown
- 1978-11-03 EP EP78101299A patent/EP0002010B1/de not_active Expired
- 1978-11-03 AU AU41324/78A patent/AU4132478A/en active Pending
- 1978-11-03 CS CS787188A patent/CS212309B2/cs unknown
- 1978-11-03 DD DD78208873A patent/DD139847A5/de unknown
- 1978-11-03 MC MC781338A patent/MC1223A1/xx unknown
- 1978-11-03 DE DE19782847766 patent/DE2847766A1/de not_active Withdrawn
- 1978-11-03 DE DE7878101299T patent/DE2861952D1/de not_active Expired
- 1978-11-03 RO RO7895588A patent/RO76151A/ro unknown
- 1978-11-04 SU SU782680652A patent/SU831073A3/ru active
- 1978-11-05 EG EG646/78A patent/EG13665A/xx active
- 1978-11-06 US US05/958,300 patent/US4244957A/en not_active Expired - Lifetime
- 1978-11-06 CA CA315,866A patent/CA1106847A/en not_active Expired
- 1978-11-06 IT IT29486/78A patent/IT1160046B/it active
- 1978-11-06 SE SE7811455A patent/SE7811455L/xx not_active Application Discontinuation
- 1978-11-06 GB GB7843271A patent/GB2008579B/en not_active Expired
- 1978-11-06 AT AT0791378A patent/AT371112B/de not_active IP Right Cessation
- 1978-11-06 DK DK494978A patent/DK494978A/da not_active Application Discontinuation
- 1978-11-06 PT PT68752A patent/PT68752A/pt unknown
- 1978-11-06 GB GB8125779A patent/GB2086379B/en not_active Expired
- 1978-11-06 JP JP13593678A patent/JPS5473779A/ja active Pending
- 1978-11-06 NO NO783719A patent/NO783719L/no unknown
- 1978-11-07 FI FI783393A patent/FI783393A/fi unknown
- 1978-11-07 PL PL21075978A patent/PL210759A1/xx unknown
- 1978-11-07 NL NL7811070A patent/NL7811070A/xx not_active Application Discontinuation
- 1978-11-07 BR BR7807317A patent/BR7807317A/pt unknown
- 1978-11-07 AR AR274367A patent/AR223656A1/es active
-
1979
- 1979-04-30 ES ES480112A patent/ES480112A1/es not_active Expired
- 1979-04-30 ES ES480111A patent/ES480111A1/es not_active Expired
- 1979-04-30 ES ES480113A patent/ES480113A1/es not_active Expired
- 1979-08-31 SU SU792806102A patent/SU910119A3/ru active
-
1980
- 1980-08-14 US US06/178,223 patent/US4355033A/en not_active Expired - Lifetime
-
1982
- 1982-08-05 US US06/405,476 patent/US4511720A/en not_active Expired - Fee Related
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