ES8305342A1 - "procedimiento para la preparacion de derivados de tiazolina". - Google Patents
"procedimiento para la preparacion de derivados de tiazolina".Info
- Publication number
- ES8305342A1 ES8305342A1 ES508293A ES508293A ES8305342A1 ES 8305342 A1 ES8305342 A1 ES 8305342A1 ES 508293 A ES508293 A ES 508293A ES 508293 A ES508293 A ES 508293A ES 8305342 A1 ES8305342 A1 ES 8305342A1
- Authority
- ES
- Spain
- Prior art keywords
- preparation
- pharmaceutical preparations
- preparations containing
- thiazoline derivatives
- thiazoline
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/18—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Vascular Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DE TIAZOLINA. SE HACE REACCIONAR COMPUESTOS (II) CON TIUREAS (III) EN PROPORCION DE 1:1,5 MOLES. SE OBTIENE EL COMPUESTO (I). LA REACCION TIENE LUGAR EN DISOLVENTES POLARES INERTES TALES COMO DIMETILFORMAMIDA, DIMETILACETAIDA, ETERES DE ETILEUGLICOL, ACETONA O TETRAHIDROFURANO. ASI MISMO LA REACCION PUEDE EFECTUARSE SIN DISOLVENTES POR CALENTAMIENTO DE LA MEZCLA DE REACCION A UNA TEMPERATURA DE 100 A 180 C. LA DURACION DE LA REACCION DEPENDE DEL DISOLVENTE Y DE LA TEMPERATURA EMPLEADA PUDIENDO ESTAR COMPRENDIDA ENTRE 15 MINUTOS Y 24 HORAS.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19803049460 DE3049460A1 (de) | 1980-12-30 | 1980-12-30 | "thiazolinderivate, verfahren zu ihrer herstellung, ihre verwendung sowie pharmazeutische praeparate auf basis dieser verbindungen |
Publications (2)
Publication Number | Publication Date |
---|---|
ES508293A0 ES508293A0 (es) | 1983-04-01 |
ES8305342A1 true ES8305342A1 (es) | 1983-04-01 |
Family
ID=6120529
Family Applications (5)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES508293A Expired ES8305342A1 (es) | 1980-12-30 | 1981-12-23 | "procedimiento para la preparacion de derivados de tiazolina". |
ES518273A Granted ES518273A0 (es) | 1980-12-30 | 1982-12-16 | Procedimiento para la preparacion de derivados de tiazolina. |
ES518274A Expired ES8308551A1 (es) | 1980-12-30 | 1982-12-16 | Procedimiento para la preparacion de derivados de tiazolina. |
ES518272A Expired ES8308549A1 (es) | 1980-12-30 | 1982-12-16 | Procedimiento para la preparacion de derivados de tiazolina. |
ES518271A Expired ES8402829A1 (es) | 1980-12-30 | 1982-12-16 | Procedimiento para la preparacion de derivados de tiazolina. |
Family Applications After (4)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES518273A Granted ES518273A0 (es) | 1980-12-30 | 1982-12-16 | Procedimiento para la preparacion de derivados de tiazolina. |
ES518274A Expired ES8308551A1 (es) | 1980-12-30 | 1982-12-16 | Procedimiento para la preparacion de derivados de tiazolina. |
ES518272A Expired ES8308549A1 (es) | 1980-12-30 | 1982-12-16 | Procedimiento para la preparacion de derivados de tiazolina. |
ES518271A Expired ES8402829A1 (es) | 1980-12-30 | 1982-12-16 | Procedimiento para la preparacion de derivados de tiazolina. |
Country Status (17)
Country | Link |
---|---|
US (1) | US4421757A (es) |
EP (1) | EP0055458B1 (es) |
JP (1) | JPS57134472A (es) |
KR (1) | KR830007601A (es) |
AR (2) | AR231134A1 (es) |
AT (1) | ATE11778T1 (es) |
AU (1) | AU542670B2 (es) |
CA (1) | CA1173836A (es) |
DE (2) | DE3049460A1 (es) |
DK (1) | DK581181A (es) |
ES (5) | ES8305342A1 (es) |
FI (1) | FI814175L (es) |
HU (1) | HU184976B (es) |
IE (1) | IE52259B1 (es) |
IL (1) | IL64653A (es) |
NO (1) | NO154551B (es) |
ZA (1) | ZA818968B (es) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4761422A (en) * | 1986-11-20 | 1988-08-02 | Lusofarmaco Istituto Lusofarmaco D'italia Spa | (2-amino-4-aryl-thiazole-5-yl)ethanols and their derivatives having diuretic activity and methods for preparing the same |
IL144031A0 (en) * | 1999-01-14 | 2002-04-21 | Bayer Ag | Substituted 2-arylimino heterocycles and compositions containing them, for use as progesterone receptor binding agents |
US6353006B1 (en) | 1999-01-14 | 2002-03-05 | Bayer Corporation | Substituted 2-arylimino heterocycles and compositions containing them, for use as progesterone receptor binding agents |
FR2819508B1 (fr) * | 2001-01-12 | 2005-01-21 | Sod Conseils Rech Applic | Derives de 2-arylimino-2, 3-dihydorthiazoles, leurs procedes de preparation et leur utilisation therapeutiques |
FR2796643B1 (fr) * | 1999-07-22 | 2005-04-29 | Sod Conseils Rech Applic | Derives de 2-arylimino-2, 3-dihydrothiazoles, leurs procedes de preparation et leur utilisation therapeutique |
ATE393150T1 (de) * | 1999-09-14 | 2008-05-15 | Shionogi & Co | 2-imino-1,3-thiazin-derivate |
US7271195B2 (en) | 2003-06-10 | 2007-09-18 | Kalypsys, Inc. | Carbonyl compounds as inhibitors of histone deacetylase for the treatment of disease |
CA2528003A1 (en) * | 2003-06-10 | 2004-12-23 | Kalypsys, Inc. | Carbonyl compounds as inhibitors of histone deacetylase for the treatment of disease |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2436263C2 (de) * | 1974-07-27 | 1983-02-17 | Hoechst Ag, 6000 Frankfurt | Thiazolidinderivate und Verfahren zu ihrer Herstellung |
DE2533821A1 (de) * | 1975-07-29 | 1977-02-17 | Hoechst Ag | Thiazolidinderivate und verfahren zu ihrer herstellung |
DE2546165A1 (de) * | 1975-10-15 | 1977-04-28 | Hoechst Ag | Thiazolidinderivate und verfahren zu ihrer herstellung |
SE7700436L (sv) * | 1976-01-17 | 1977-07-18 | Hoechst Ag | Tiazolidinderivat och forfarande for deras framstellning |
DE2926771A1 (de) * | 1979-07-03 | 1981-01-15 | Hoechst Ag | Thiazolidinderivate und verfahren zu ihrer herstellung |
-
1980
- 1980-12-30 DE DE19803049460 patent/DE3049460A1/de not_active Withdrawn
-
1981
- 1981-12-22 DE DE8181110677T patent/DE3168978D1/de not_active Expired
- 1981-12-22 AT AT81110677T patent/ATE11778T1/de not_active IP Right Cessation
- 1981-12-22 EP EP81110677A patent/EP0055458B1/de not_active Expired
- 1981-12-23 IE IE3057/81A patent/IE52259B1/en unknown
- 1981-12-23 ES ES508293A patent/ES8305342A1/es not_active Expired
- 1981-12-28 FI FI814175A patent/FI814175L/fi not_active Application Discontinuation
- 1981-12-28 JP JP56210093A patent/JPS57134472A/ja active Pending
- 1981-12-28 IL IL64653A patent/IL64653A/xx unknown
- 1981-12-28 US US06/335,149 patent/US4421757A/en not_active Expired - Fee Related
- 1981-12-28 AR AR287966A patent/AR231134A1/es active
- 1981-12-29 HU HU813984A patent/HU184976B/hu unknown
- 1981-12-29 DK DK581181A patent/DK581181A/da not_active Application Discontinuation
- 1981-12-29 NO NO814468A patent/NO154551B/no unknown
- 1981-12-29 ZA ZA818968A patent/ZA818968B/xx unknown
- 1981-12-29 CA CA000393285A patent/CA1173836A/en not_active Expired
- 1981-12-30 AU AU79068/81A patent/AU542670B2/en not_active Ceased
- 1981-12-30 KR KR1019810005232A patent/KR830007601A/ko unknown
-
1982
- 1982-11-30 AR AR291445A patent/AR231978A1/es active
- 1982-12-16 ES ES518273A patent/ES518273A0/es active Granted
- 1982-12-16 ES ES518274A patent/ES8308551A1/es not_active Expired
- 1982-12-16 ES ES518272A patent/ES8308549A1/es not_active Expired
- 1982-12-16 ES ES518271A patent/ES8402829A1/es not_active Expired
Also Published As
Publication number | Publication date |
---|---|
IE52259B1 (en) | 1987-08-19 |
ES8308550A1 (es) | 1983-09-01 |
ES508293A0 (es) | 1983-04-01 |
AU542670B2 (en) | 1985-02-28 |
NO814468L (no) | 1982-07-01 |
AU7906881A (en) | 1982-07-08 |
ES518271A0 (es) | 1984-02-16 |
DK581181A (da) | 1982-07-01 |
NO154551B (no) | 1986-07-07 |
AR231134A1 (es) | 1984-09-28 |
ES518274A0 (es) | 1983-09-01 |
IL64653A (en) | 1985-09-29 |
EP0055458A2 (de) | 1982-07-07 |
IL64653A0 (en) | 1982-03-31 |
US4421757A (en) | 1983-12-20 |
HU184976B (en) | 1984-11-28 |
ATE11778T1 (de) | 1985-02-15 |
ES8402829A1 (es) | 1984-02-16 |
ES518272A0 (es) | 1983-09-01 |
EP0055458B1 (de) | 1985-02-13 |
JPS57134472A (en) | 1982-08-19 |
ES8308549A1 (es) | 1983-09-01 |
CA1173836A (en) | 1984-09-04 |
AR231978A1 (es) | 1985-04-30 |
DE3168978D1 (en) | 1985-03-28 |
DE3049460A1 (de) | 1982-07-29 |
EP0055458A3 (en) | 1982-10-20 |
ZA818968B (en) | 1982-11-24 |
IE813057L (en) | 1982-06-30 |
FI814175L (fi) | 1982-07-01 |
ES8308551A1 (es) | 1983-09-01 |
KR830007601A (ko) | 1983-11-04 |
ES518273A0 (es) | 1983-09-01 |
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