ES2602789T3 - Productos intermedios conectores para la síntesis de moduladores macrocíclicos del receptor de la grelina - Google Patents

Productos intermedios conectores para la síntesis de moduladores macrocíclicos del receptor de la grelina Download PDF

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Publication number
ES2602789T3
ES2602789T3 ES12195556.1T ES12195556T ES2602789T3 ES 2602789 T3 ES2602789 T3 ES 2602789T3 ES 12195556 T ES12195556 T ES 12195556T ES 2602789 T3 ES2602789 T3 ES 2602789T3
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boc
bts
compound
nmeala
ghrelin
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Spanish (es)
Inventor
Hamid Hoveyda
Graeme Fraser
Sophie Beauchemin
Martin Brassard
David Drutz
Eric Marsault
Luc Quellet
Mark L Peterson
Zhigang Wang
Kamel Benkali
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Ocera Therapeutics Inc
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Ocera Therapeutics Inc
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ES12195556.1T 2007-02-09 2008-02-08 Productos intermedios conectores para la síntesis de moduladores macrocíclicos del receptor de la grelina Active ES2602789T3 (es)

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US88916307P 2007-02-09 2007-02-09
US889163P 2007-02-09

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ES12195556.1T Active ES2602789T3 (es) 2007-02-09 2008-02-08 Productos intermedios conectores para la síntesis de moduladores macrocíclicos del receptor de la grelina
ES08799889.4T Active ES2604943T3 (es) 2007-02-09 2008-02-08 Moduladores macrocíclicos del receptor de la grelina y procedimientos de uso de los mismos

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US (3) US9371297B2 (OSRAM)
EP (2) EP2118080B1 (OSRAM)
JP (2) JP2010518090A (OSRAM)
KR (1) KR20090107088A (OSRAM)
CN (1) CN101657436A (OSRAM)
AU (1) AU2008241532A1 (OSRAM)
BR (1) BRPI0807046A2 (OSRAM)
CA (1) CA2677399C (OSRAM)
EA (1) EA200901077A1 (OSRAM)
ES (2) ES2602789T3 (OSRAM)
MX (1) MX2009008574A (OSRAM)
WO (1) WO2008130464A1 (OSRAM)

Families Citing this family (41)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20090198050A1 (en) * 2003-06-18 2009-08-06 Tranzyme Pharma Inc. Macrocyclic Modulators of the Ghrelin Receptor
US8921521B2 (en) 2003-06-18 2014-12-30 Ocera Therapeutics, Inc. Macrocyclic modulators of the Ghrelin receptor
US7491695B2 (en) 2003-06-18 2009-02-17 Tranzyme Pharma Inc. Methods of using macrocyclic modulators of the ghrelin receptor
CA2528375C (en) 2003-06-18 2013-11-19 Tranzyme Pharma, Inc. Macrocyclic antagonists of the motilin receptor
US7476653B2 (en) * 2003-06-18 2009-01-13 Tranzyme Pharma, Inc. Macrocyclic modulators of the ghrelin receptor
US8088733B2 (en) * 2006-07-06 2012-01-03 Tranzyme Pharma Inc. Methods of using macrocyclic agonists of the ghrelin receptor for treatment of gastrointestinal motility disorders
EP2118123B1 (en) 2007-01-31 2015-10-14 Dana-Farber Cancer Institute, Inc. Stabilized p53 peptides and uses thereof
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