MX2009008574A - Moduladores del receptor de grelina macrociclicos y metodos para usar el mismo. - Google Patents

Moduladores del receptor de grelina macrociclicos y metodos para usar el mismo.

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Publication number
MX2009008574A
MX2009008574A MX2009008574A MX2009008574A MX2009008574A MX 2009008574 A MX2009008574 A MX 2009008574A MX 2009008574 A MX2009008574 A MX 2009008574A MX 2009008574 A MX2009008574 A MX 2009008574A MX 2009008574 A MX2009008574 A MX 2009008574A
Authority
MX
Mexico
Prior art keywords
disorders
ghrelin receptor
methods
compounds
same
Prior art date
Application number
MX2009008574A
Other languages
English (en)
Spanish (es)
Inventor
Hamid Hoveyda
Graeme Fraser
Sophie Beauchemin
Martin Brassard
David Drutz
Eric Marsault
Luc Ouellet
Mark L Peterson
Zhigang Wang
Kamel Benakli
Original Assignee
Tranzyme Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tranzyme Pharma Inc filed Critical Tranzyme Pharma Inc
Publication of MX2009008574A publication Critical patent/MX2009008574A/es

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Hospice & Palliative Care (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Psychiatry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Otolaryngology (AREA)
  • Endocrinology (AREA)
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MX2009008574A 2007-02-09 2008-02-08 Moduladores del receptor de grelina macrociclicos y metodos para usar el mismo. MX2009008574A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88916307P 2007-02-09 2007-02-09
PCT/US2008/001754 WO2008130464A1 (en) 2007-02-09 2008-02-08 Macrocyclic ghrelin receptor modulators and methods of using the same

Publications (1)

Publication Number Publication Date
MX2009008574A true MX2009008574A (es) 2009-12-09

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MX2009008574A MX2009008574A (es) 2007-02-09 2008-02-08 Moduladores del receptor de grelina macrociclicos y metodos para usar el mismo.

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US (3) US9371297B2 (OSRAM)
EP (2) EP2118080B1 (OSRAM)
JP (2) JP2010518090A (OSRAM)
KR (1) KR20090107088A (OSRAM)
CN (1) CN101657436A (OSRAM)
AU (1) AU2008241532A1 (OSRAM)
BR (1) BRPI0807046A2 (OSRAM)
CA (1) CA2677399C (OSRAM)
EA (1) EA200901077A1 (OSRAM)
ES (2) ES2602789T3 (OSRAM)
MX (1) MX2009008574A (OSRAM)
WO (1) WO2008130464A1 (OSRAM)

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US20090198050A1 (en) * 2003-06-18 2009-08-06 Tranzyme Pharma Inc. Macrocyclic Modulators of the Ghrelin Receptor
US8921521B2 (en) 2003-06-18 2014-12-30 Ocera Therapeutics, Inc. Macrocyclic modulators of the Ghrelin receptor
US7491695B2 (en) 2003-06-18 2009-02-17 Tranzyme Pharma Inc. Methods of using macrocyclic modulators of the ghrelin receptor
CA2528375C (en) 2003-06-18 2013-11-19 Tranzyme Pharma, Inc. Macrocyclic antagonists of the motilin receptor
US7476653B2 (en) * 2003-06-18 2009-01-13 Tranzyme Pharma, Inc. Macrocyclic modulators of the ghrelin receptor
US8088733B2 (en) * 2006-07-06 2012-01-03 Tranzyme Pharma Inc. Methods of using macrocyclic agonists of the ghrelin receptor for treatment of gastrointestinal motility disorders
EP2118123B1 (en) 2007-01-31 2015-10-14 Dana-Farber Cancer Institute, Inc. Stabilized p53 peptides and uses thereof
CN101686966A (zh) * 2007-02-13 2010-03-31 赫尔辛医疗（美国）有限公司 使用生长激素促分泌素治疗细胞增生疾病的方法
EP3159352B1 (en) 2007-03-28 2023-08-02 President and Fellows of Harvard College Stitched polypeptides
TWI429436B (zh) * 2007-04-10 2014-03-11 Helsinn Therapeutics Us Inc 使用生長激素促泌素治療或預防嘔吐之方法
US20080287371A1 (en) * 2007-05-17 2008-11-20 Tranzyme Pharma Inc. Macrocyclic antagonists of the motilin receptor for modulation of the migrating motor complex
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