ES2393962T3 - Sales de compuestos inhibidores del VIH. - Google Patents
Sales de compuestos inhibidores del VIH. Download PDFInfo
- Publication number
- ES2393962T3 ES2393962T3 ES09790117T ES09790117T ES2393962T3 ES 2393962 T3 ES2393962 T3 ES 2393962T3 ES 09790117 T ES09790117 T ES 09790117T ES 09790117 T ES09790117 T ES 09790117T ES 2393962 T3 ES2393962 T3 ES 2393962T3
- Authority
- ES
- Spain
- Prior art keywords
- salt
- fluoro
- purin
- phenoxyphosphinoyl
- oxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
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- A61P31/18—Antivirals for RNA viruses for HIV
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| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US7898908P | 2008-07-08 | 2008-07-08 | |
| US78989 | 2008-07-08 | ||
| PCT/US2009/049838 WO2010005986A1 (en) | 2008-07-08 | 2009-07-07 | Salts of hiv inhibitor compounds |
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| ES2393962T3 true ES2393962T3 (es) | 2013-01-03 |
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| ES09790117T Active ES2393962T3 (es) | 2008-07-08 | 2009-07-07 | Sales de compuestos inhibidores del VIH. |
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Families Citing this family (9)
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| EP1628685B1 (en) | 2003-04-25 | 2010-12-08 | Gilead Sciences, Inc. | Antiviral phosphonate analogs |
| WO2006110157A2 (en) * | 2004-07-27 | 2006-10-19 | Gilead Sciences, Inc. | Nucleoside phosphonate conjugates as anti hiv agents |
| HRP20120700T1 (hr) * | 2008-07-08 | 2012-09-30 | Gilead Sciences | SOLI SPOJEVA INHIBITORA HIV-a |
| WO2012138907A2 (en) * | 2011-04-05 | 2012-10-11 | Translational Genomics Research Institute | Solid forms of curcumin |
| EP3450438A1 (en) * | 2011-05-19 | 2019-03-06 | Gilead Sciences, Inc. | Processes and intermediates for preparing anti-hiv agents |
| CN118286245A (zh) | 2014-12-26 | 2024-07-05 | 埃莫里大学 | N4-羟基胞苷和衍生物及与其相关的抗病毒用途 |
| US20180085387A1 (en) * | 2016-09-27 | 2018-03-29 | Gilead Sciences, Inc. | Therapeutic compositions for treatment of human immunodeficiency virus |
| ES2892402T3 (es) | 2017-08-01 | 2022-02-04 | Gilead Sciences Inc | Formas cristalinas de ((S)-((((2R,5R)-5-(6-amino-9H-purin-9-il)-4-fluoro-2,5-dihidrofuran-2-il)oxi)metil)(fenoxi)fosforil)-L-alaninato de etilo para tratar infecciones virales |
| US11331331B2 (en) | 2017-12-07 | 2022-05-17 | Emory University | N4-hydroxycytidine and derivatives and anti-viral uses related thereto |
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