EE04677B1 - Tetrahdropridoeetrid, nende kasutamine ja ravim - Google Patents

Tetrahdropridoeetrid, nende kasutamine ja ravim

Info

Publication number
EE04677B1
EE04677B1 EEP200100172A EEP200100172A EE04677B1 EE 04677 B1 EE04677 B1 EE 04677B1 EE P200100172 A EEP200100172 A EE P200100172A EE P200100172 A EEP200100172 A EE P200100172A EE 04677 B1 EE04677 B1 EE 04677B1
Authority
EE
Estonia
Prior art keywords
ridoethers
tetrah
medicine
drop
naphthyridine
Prior art date
Application number
EEP200100172A
Other languages
English (en)
Estonian (et)
Inventor
Senn-Bilfinger J�rg
Postius Stefan
Simon Wolfgang-Alexander
Grundler Gerhard
Hanauer Guido
Huber Reinhard
Kromer Wolfgang
Sturm Ernst
Original Assignee
Byk Gulden Lomberg Chemische Fabrik Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Byk Gulden Lomberg Chemische Fabrik Gmbh filed Critical Byk Gulden Lomberg Chemische Fabrik Gmbh
Publication of EE200100172A publication Critical patent/EE200100172A/xx
Publication of EE04677B1 publication Critical patent/EE04677B1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
EEP200100172A 1998-09-23 1999-09-17 Tetrahdropridoeetrid, nende kasutamine ja ravim EE04677B1 (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19843504 1998-09-23
EP98117988 1998-09-23
PCT/EP1999/006899 WO2000017200A1 (en) 1998-09-23 1999-09-17 Tetrahydropyridoethers

Publications (2)

Publication Number Publication Date
EE200100172A EE200100172A (et) 2002-06-17
EE04677B1 true EE04677B1 (et) 2006-08-15

Family

ID=26049024

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100172A EE04677B1 (et) 1998-09-23 1999-09-17 Tetrahdropridoeetrid, nende kasutamine ja ravim

Country Status (31)

Country Link
US (4) US6436953B1 (zh)
EP (1) EP1115725B1 (zh)
JP (1) JP4145492B2 (zh)
KR (1) KR100668400B1 (zh)
CN (2) CN1155598C (zh)
AT (1) ATE231862T1 (zh)
AU (1) AU763463B2 (zh)
BG (1) BG65195B1 (zh)
BR (1) BR9914044A (zh)
CA (1) CA2344251A1 (zh)
CZ (1) CZ292335B6 (zh)
DE (1) DE69905178T2 (zh)
DK (1) DK1115725T3 (zh)
EA (1) EA005377B1 (zh)
EE (1) EE04677B1 (zh)
ES (1) ES2191464T3 (zh)
GE (1) GEP20032926B (zh)
HK (1) HK1038360B (zh)
HR (1) HRP20010224A2 (zh)
HU (1) HUP0102990A3 (zh)
ID (1) ID28896A (zh)
IL (2) IL142063A0 (zh)
NO (1) NO317304B1 (zh)
NZ (1) NZ510610A (zh)
PL (1) PL193616B1 (zh)
PT (1) PT1115725E (zh)
RS (1) RS50145B (zh)
SI (1) SI1115725T1 (zh)
SK (1) SK285165B6 (zh)
TR (1) TR200100805T2 (zh)
WO (1) WO2000017200A1 (zh)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EE04677B1 (et) 1998-09-23 2006-08-15 Byk Gulden Lomberg Chemische Fabrik Gmbh Tetrahdropridoeetrid, nende kasutamine ja ravim
CA2370231A1 (en) 1999-04-17 2000-10-26 Byk Gulden Lomberg Chemische Fabrik Gmbh Haloalkoxy imidazonaphthyridines
CA2721484A1 (en) * 1999-05-12 2000-11-12 President And Fellows Of Harvard College Dopamine transporter imaging agents
DE60115466T2 (de) * 2000-03-29 2006-07-20 Altana Pharma Ag Wirkstoffvorläufer von imidazopyridin-derivaten
BR0109512A (pt) * 2000-03-29 2002-12-17 Altana Pharma Ag Imidazopiridinas tricìclicas
NZ525281A (en) * 2000-10-25 2004-11-26 Altana Pharma Ag Polysubstituted imidazopyridines as gastric secretion inhibitors
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
CZ20032398A3 (cs) * 2001-03-08 2004-02-18 Astrazeneca Ab Nové použití derivátů 6-karboxamidoimidazo [1,2-a] pyridinu
ES2271317T3 (es) 2001-08-02 2007-04-16 Altana Pharma Ag Epoxidos triciclicos.
WO2003014120A1 (en) * 2001-08-03 2003-02-20 Altana Pharma Ag Amino-substituted imidazopyridines for the treatment of gastrointestinal diseases
JP2005504048A (ja) * 2001-08-03 2005-02-10 アルタナ ファルマ アクチエンゲゼルシャフト 胃腸障害治療用のアルカリ置換されたイミダゾピリジン
EP1476445A1 (en) 2002-02-15 2004-11-17 ALTANA Pharma AG Tricyclic n-acyl compounds
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
BR0309808A (pt) * 2002-05-07 2005-03-01 Altana Pharma Ag Combinação para o tratamento de distúrbios das vias aéreas
JP2006508142A (ja) 2002-11-19 2006-03-09 アルタナ ファルマ アクチエンゲゼルシャフト 8−置換イミダゾピリジン
PT1572217E (pt) 2002-12-12 2008-11-28 Nycomed Gmbh Medicamento combinado de r,r-formoterol e ciclesonida
WO2004056362A2 (en) * 2002-12-20 2004-07-08 Altana Pharma Ag 8-trialkysyloxy-2-methyl-9-phenyl-7-0 xo-7,8,9,10- tetrahydroimidazo ‘1,2-h! ‘1,7! naphthyridines
RS20050603A (en) * 2003-02-17 2007-09-21 Altana Pharma Ag., New combinations and new application of pharmaceutically active compounds
CN100471840C (zh) 2003-03-10 2009-03-25 尼科梅德有限责任公司 制备罗氟司特的方法
TW200503783A (en) * 2003-04-11 2005-02-01 Altana Pharma Ag Oral pharmaceutical preparation for proton pump antagonists
SA04250092B1 (ar) * 2003-05-14 2008-05-04 التانا فاروا ايه جي مركب وسيط جديد لتحضير مركبات إيميدازوبيريدين imidazopyridines فعالة علاجياً
EP1644043A1 (en) * 2003-05-27 2006-04-12 ALTANA Pharma AG Pharmaceutical combinations of a proton pump inhibitor and a compound which modifies gastrointestinal motility
JP2007507425A (ja) * 2003-08-29 2007-03-29 ダイノゲン ファーマシューティカルズ,インコーポレイテッド 胃腸管運動障害を処置するために有用な組成物
US8371292B2 (en) 2003-09-16 2013-02-12 Nycomed Gmbh Use of ciclesonide for the treatment of respiratory diseases
EP1682133A1 (en) * 2003-11-03 2006-07-26 AstraZeneca AB Imidazo 1,2-a pyridine derivatives for the treatment of silent gastro-esophageal reflux
US7326784B2 (en) 2003-12-19 2008-02-05 Altana Pharma Ag Intermediates for the preparation of tricyclic dihydropyrano-imidazo-pyridines derivatives
NZ549011A (en) * 2004-02-17 2009-04-30 Altana Pharma Ag Tricyclic imidazopyridines and intermediates for the synthesis thereof
ES2426920T3 (es) 2004-09-03 2013-10-25 Yuhan Corporation Derivados de pirrolo[3,2-B]piridina y procesos para su preparación
ES2367312T3 (es) 2004-09-03 2011-11-02 Yuhan Corporation DERIVADOS DE PIRROLO [3,2-c] PIRIDINA Y PROCESOS PARA LA PREPARACIÓN DE LOS MISMOS.
PL1784404T3 (pl) 2004-09-03 2012-04-30 Yuhan Corp Pochodne pirolo[2,3-c]pirydyny i sposoby ich wytwarzania
AU2006224619B2 (en) * 2005-03-16 2012-06-07 Takeda Gmbh Taste masked dosage form containing roflumilast
EP2080513A1 (en) 2008-01-16 2009-07-22 Schraermeyer, Ulrich, Prof. Dr. rer. nat Tetrahydropyridoethers for treatment of AMD
ES2767251T3 (es) * 2009-07-09 2020-06-17 Raqualia Pharma Inc Antagonista de la bomba de ácido para el tratamiento de enfermedades involucradas en la motilidad gastrointestinal anormal
WO2012027240A1 (en) * 2010-08-23 2012-03-01 Schering Corporation Fused tricyclic inhibitors of mammalian target of rapamycin
ES2635067T3 (es) * 2012-06-15 2017-10-02 Bio-Pharm Solutions Co., Ltd. Compuesto de sulfamato de fenilalquilo y composición de relajante muscular que comprende el mismo
WO2015052256A1 (en) 2013-10-08 2015-04-16 Katairo Gmbh Tetrahydropyridoethers for the treatment of stargardt's disease

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4468400A (en) * 1982-12-20 1984-08-28 Schering Corporation Antiulcer tricyclic imidazo [1,2-a]pyridines
EP0370056A1 (de) 1987-07-16 1990-05-30 Byk Gulden Lomberg Chemische Fabrik Gmbh Neue diazole
SE9401197D0 (sv) * 1994-04-11 1994-04-11 Astra Ab Active compounds
NZ290819A (en) * 1994-07-28 1998-06-26 Byk Gulden Lomberg Chem Fab Acyl 8-benzyloxy- or 8-benzylaminoimidazopyridines
EP0971922B1 (en) * 1997-03-24 2004-04-28 ALTANA Pharma AG Tetrahydropyrido compounds
CN1250546C (zh) * 1997-03-24 2006-04-12 奥坦纳医药公司 四氢吡啶并化合物
EE04677B1 (et) * 1998-09-23 2006-08-15 Byk Gulden Lomberg Chemische Fabrik Gmbh Tetrahdropridoeetrid, nende kasutamine ja ravim

Also Published As

Publication number Publication date
CN1560055A (zh) 2005-01-05
JP2002526499A (ja) 2002-08-20
BG65195B1 (bg) 2007-06-29
CZ20011082A3 (cs) 2001-09-12
BR9914044A (pt) 2001-12-04
EP1115725A1 (en) 2001-07-18
NO317304B1 (no) 2004-10-04
IL142063A (en) 2007-10-31
YU21401A (sh) 2004-03-12
NO20011243L (no) 2001-03-12
SI1115725T1 (en) 2003-06-30
IL142063A0 (en) 2002-03-10
DK1115725T3 (da) 2003-06-23
US20020169320A1 (en) 2002-11-14
HUP0102990A2 (hu) 2002-01-28
CN100506821C (zh) 2009-07-01
DE69905178T2 (de) 2003-07-17
KR20010075223A (ko) 2001-08-09
NZ510610A (en) 2003-07-25
US7105676B2 (en) 2006-09-12
WO2000017200A1 (en) 2000-03-30
PL346617A1 (en) 2002-02-25
ES2191464T3 (es) 2003-09-01
CN1155598C (zh) 2004-06-30
EE200100172A (et) 2002-06-17
BG105270A (en) 2001-11-30
ATE231862T1 (de) 2003-02-15
HK1038360A1 (en) 2002-03-15
DE69905178D1 (de) 2003-03-06
HUP0102990A3 (en) 2002-09-30
CN1319101A (zh) 2001-10-24
KR100668400B1 (ko) 2007-01-17
EP1115725B1 (en) 2003-01-29
CA2344251A1 (en) 2000-03-30
SK285165B6 (sk) 2006-07-07
US20040162310A1 (en) 2004-08-19
NO20011243D0 (no) 2001-03-12
PL193616B1 (pl) 2007-02-28
SK3992001A3 (en) 2001-12-03
AU6192099A (en) 2000-04-10
US6436953B1 (en) 2002-08-20
GEP20032926B (en) 2003-03-25
EA200100315A1 (ru) 2001-10-22
CZ292335B6 (cs) 2003-09-17
US6696460B2 (en) 2004-02-24
RS50145B (sr) 2009-03-25
AU763463B2 (en) 2003-07-24
EA005377B1 (ru) 2005-02-24
TR200100805T2 (tr) 2001-08-21
JP4145492B2 (ja) 2008-09-03
US7393860B1 (en) 2008-07-01
PT1115725E (pt) 2003-06-30
HK1038360B (zh) 2003-05-16
ID28896A (id) 2001-07-12
HRP20010224A2 (en) 2002-04-30

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