EE04578B1 - Farmatseutiline kompositsioon N-piperidino-3-pürasoolkarboksamiidi derivaadi, tema soolade ja nendesolvaatide suu kaudu manustamiseks - Google Patents

Farmatseutiline kompositsioon N-piperidino-3-pürasoolkarboksamiidi derivaadi, tema soolade ja nendesolvaatide suu kaudu manustamiseks

Info

Publication number
EE04578B1
EE04578B1 EEP199900441A EEP9900441A EE04578B1 EE 04578 B1 EE04578 B1 EE 04578B1 EE P199900441 A EEP199900441 A EE P199900441A EE P9900441 A EEP9900441 A EE P9900441A EE 04578 B1 EE04578 B1 EE 04578B1
Authority
EE
Estonia
Prior art keywords
piperidino
solvates
salts
pharmaceutical composition
oral administration
Prior art date
Application number
EEP199900441A
Other languages
English (en)
Inventor
Abramovici Bernard
Condamine Christian
Gromenil Jean-Claude
Original Assignee
Sanofi-Synthlabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi-Synthlabo filed Critical Sanofi-Synthlabo
Publication of EE9900441A publication Critical patent/EE9900441A/et
Publication of EE04578B1 publication Critical patent/EE04578B1/et

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
EEP199900441A 1997-03-28 1998-03-27 Farmatseutiline kompositsioon N-piperidino-3-pürasoolkarboksamiidi derivaadi, tema soolade ja nendesolvaatide suu kaudu manustamiseks EE04578B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9703835A FR2761266B1 (fr) 1997-03-28 1997-03-28 Composition pharmaceutique formee par granulation humide pour l'administration orale d'un derive du n-piperidino-3- pyrazolecarboxamide, de ses sels et de leurs solvates
PCT/FR1998/000631 WO1998043636A1 (fr) 1997-03-28 1998-03-27 Composition pharmaceutique pour administration orale d'un derive du n-piperidino-3-pyrazolecarboxamide, de ses sels et de leurs s olvates

Publications (2)

Publication Number Publication Date
EE9900441A EE9900441A (et) 2000-04-17
EE04578B1 true EE04578B1 (et) 2006-02-15

Family

ID=9505295

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP199900441A EE04578B1 (et) 1997-03-28 1998-03-27 Farmatseutiline kompositsioon N-piperidino-3-pürasoolkarboksamiidi derivaadi, tema soolade ja nendesolvaatide suu kaudu manustamiseks

Country Status (41)

Country Link
US (1) US6893659B2 (et)
EP (1) EP0969832B1 (et)
JP (1) JP3805797B2 (et)
KR (1) KR100479521B1 (et)
CN (1) CN1126543C (et)
AR (1) AR012160A1 (et)
AT (1) ATE202703T1 (et)
AU (1) AU740486B2 (et)
BR (1) BR9808429A (et)
CA (1) CA2284051C (et)
CO (1) CO4950527A1 (et)
CY (2) CY2275B1 (et)
CZ (1) CZ292129B6 (et)
DE (1) DE69801045T2 (et)
DK (1) DK0969832T3 (et)
DZ (1) DZ2453A1 (et)
EE (1) EE04578B1 (et)
ES (1) ES2161049T3 (et)
FR (1) FR2761266B1 (et)
GR (1) GR3036382T3 (et)
HK (1) HK1022831A1 (et)
HR (1) HRP980163B1 (et)
HU (1) HU224838B1 (et)
ID (1) ID22973A (et)
IL (1) IL131818A (et)
IS (1) IS1960B (et)
MY (1) MY121733A (et)
NO (1) NO321615B1 (et)
NZ (1) NZ337736A (et)
PL (1) PL191107B1 (et)
PT (1) PT969832E (et)
RS (1) RS49606B (et)
RU (1) RU2193886C2 (et)
SA (1) SA98190095B1 (et)
SI (1) SI0969832T1 (et)
SK (1) SK283265B6 (et)
TR (1) TR199902236T2 (et)
TW (1) TW565450B (et)
UA (1) UA49056C2 (et)
WO (1) WO1998043636A1 (et)
ZA (1) ZA982609B (et)

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HUP0001894A3 (en) 2002-01-28
PT969832E (pt) 2001-11-30
US6893659B2 (en) 2005-05-17
KR100479521B1 (ko) 2005-03-30
HRP980163A2 (en) 1998-12-31
EP0969832B1 (fr) 2001-07-04
DK0969832T3 (da) 2001-10-22
NO994706D0 (no) 1999-09-27
TR199902236T2 (xx) 1999-12-21
US20030003145A1 (en) 2003-01-02
IL131818A (en) 2003-07-31
BR9808429A (pt) 2000-05-23
CY2006005I1 (el) 2009-11-04
SK283265B6 (sk) 2003-04-01
SA98190095B1 (ar) 2006-06-18
FR2761266A1 (fr) 1998-10-02
IS1960B (is) 2004-11-15
CZ344199A3 (cs) 2000-01-12
ES2161049T3 (es) 2001-11-16
GR3036382T3 (en) 2001-11-30
AR012160A1 (es) 2000-09-27
NO994706L (no) 1999-11-25
AU7052798A (en) 1998-10-22
EE9900441A (et) 2000-04-17
CA2284051C (en) 2005-01-11
PL335942A1 (en) 2000-05-22
JP3805797B2 (ja) 2006-08-09
KR20010005752A (ko) 2001-01-15
CO4950527A1 (es) 2000-09-01
CY2275B1 (en) 2003-07-04
CA2284051A1 (en) 1998-10-08
SK130999A3 (en) 2000-03-13
HU224838B1 (en) 2006-03-28
IL131818A0 (en) 2001-03-19
CZ292129B6 (cs) 2003-08-13
UA49056C2 (uk) 2002-09-16
SI0969832T1 (et) 2001-12-31
ZA982609B (en) 1998-09-30
YU47099A (sh) 2002-06-19
NZ337736A (en) 2001-02-23
ID22973A (id) 1999-12-23
FR2761266B1 (fr) 1999-07-02
WO1998043636A1 (fr) 1998-10-08
CY2006005I2 (el) 2009-11-04
NO321615B1 (no) 2006-06-12
CN1126543C (zh) 2003-11-05
RS49606B (sr) 2007-06-04
CN1251524A (zh) 2000-04-26
DZ2453A1 (fr) 2004-07-14
RU2193886C2 (ru) 2002-12-10
PL191107B1 (pl) 2006-03-31
EP0969832A1 (fr) 2000-01-12
TW565450B (en) 2003-12-11
DE69801045T2 (de) 2002-03-14
HK1022831A1 (en) 2000-08-25
DE69801045D1 (de) 2001-08-09
AU740486B2 (en) 2001-11-08
HRP980163B1 (en) 2002-10-31
IS5190A (is) 1999-09-23
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