RS49606B - Farmaceutski preparat derivata n- piperidino-3- pirazolkarboksamida, njegovih soli i njihovih solvata za oralnu administraciju - Google Patents

Farmaceutski preparat derivata n- piperidino-3- pirazolkarboksamida, njegovih soli i njihovih solvata za oralnu administraciju

Info

Publication number
RS49606B
RS49606B YUP-470/99A YU47099A RS49606B RS 49606 B RS49606 B RS 49606B YU 47099 A YU47099 A YU 47099A RS 49606 B RS49606 B RS 49606B
Authority
RS
Serbia
Prior art keywords
piperidino
solvates
oral administration
salts
pharmaceutical compositions
Prior art date
Application number
YUP-470/99A
Other languages
English (en)
Inventor
Bernard Abramovici
Christian Condamine
Jean-Claude Gromenil
Original Assignee
Sanofi-Aventis,
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi-Aventis, filed Critical Sanofi-Aventis,
Publication of YU47099A publication Critical patent/YU47099A/sh
Publication of RS49606B publication Critical patent/RS49606B/sr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Psychiatry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Farmaceutski preparat za oralnu andministraciju N-piperidino-5-(4-hlorofenil)-1-(2,4-dihlorofenil)-4-metilpirazol-3-karboksamid formule: jedna od njegovih farmaceutski prihvatljivih soli ili jednog od njihovih solvata (u daljem tekstu: aktivna komponenta), naznačen time, što sadrži: 0.5% do 20% mas. aktivne komponente u mikronizovanom obliku, 0.05% do 0.5% mas. natrijum alkilsulfata, 2.5% do 10% mas. agensa dezintegracije, i farmaceutske eksipijense, gde je preparat formulisan vlažnom granulacijom. Prijava sadrži još 9 patentnih zahteva.
YUP-470/99A 1997-03-28 1998-03-27 Farmaceutski preparat derivata n- piperidino-3- pirazolkarboksamida, njegovih soli i njihovih solvata za oralnu administraciju RS49606B (sr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9703835A FR2761266B1 (fr) 1997-03-28 1997-03-28 Composition pharmaceutique formee par granulation humide pour l'administration orale d'un derive du n-piperidino-3- pyrazolecarboxamide, de ses sels et de leurs solvates

Publications (2)

Publication Number Publication Date
YU47099A YU47099A (sh) 2002-06-19
RS49606B true RS49606B (sr) 2007-06-04

Family

ID=9505295

Family Applications (1)

Application Number Title Priority Date Filing Date
YUP-470/99A RS49606B (sr) 1997-03-28 1998-03-27 Farmaceutski preparat derivata n- piperidino-3- pirazolkarboksamida, njegovih soli i njihovih solvata za oralnu administraciju

Country Status (41)

Country Link
US (1) US6893659B2 (sr)
EP (1) EP0969832B1 (sr)
JP (1) JP3805797B2 (sr)
KR (1) KR100479521B1 (sr)
CN (1) CN1126543C (sr)
AR (1) AR012160A1 (sr)
AT (1) ATE202703T1 (sr)
AU (1) AU740486B2 (sr)
BR (1) BR9808429A (sr)
CA (1) CA2284051C (sr)
CO (1) CO4950527A1 (sr)
CY (2) CY2275B1 (sr)
CZ (1) CZ292129B6 (sr)
DE (1) DE69801045T2 (sr)
DK (1) DK0969832T3 (sr)
DZ (1) DZ2453A1 (sr)
EE (1) EE04578B1 (sr)
ES (1) ES2161049T3 (sr)
FR (1) FR2761266B1 (sr)
GR (1) GR3036382T3 (sr)
HK (1) HK1022831A1 (sr)
HR (1) HRP980163B1 (sr)
HU (1) HU224838B1 (sr)
ID (1) ID22973A (sr)
IL (1) IL131818A (sr)
IS (1) IS1960B (sr)
MY (1) MY121733A (sr)
NO (1) NO321615B1 (sr)
NZ (1) NZ337736A (sr)
PL (1) PL191107B1 (sr)
PT (1) PT969832E (sr)
RS (1) RS49606B (sr)
RU (1) RU2193886C2 (sr)
SA (1) SA98190095B1 (sr)
SI (1) SI0969832T1 (sr)
SK (1) SK283265B6 (sr)
TR (1) TR199902236T2 (sr)
TW (1) TW565450B (sr)
UA (1) UA49056C2 (sr)
WO (1) WO1998043636A1 (sr)
ZA (1) ZA982609B (sr)

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CN1126543C (zh) 2003-11-05
HRP980163A2 (en) 1998-12-31
RU2193886C2 (ru) 2002-12-10
MY121733A (en) 2006-02-28
ID22973A (id) 1999-12-23
PL335942A1 (en) 2000-05-22
ATE202703T1 (de) 2001-07-15
IS5190A (is) 1999-09-23
SK283265B6 (sk) 2003-04-01
AU740486B2 (en) 2001-11-08
CZ292129B6 (cs) 2003-08-13
CZ344199A3 (cs) 2000-01-12
ES2161049T3 (es) 2001-11-16
CA2284051A1 (en) 1998-10-08
AU7052798A (en) 1998-10-22
UA49056C2 (uk) 2002-09-16
HK1022831A1 (en) 2000-08-25
FR2761266B1 (fr) 1999-07-02
CN1251524A (zh) 2000-04-26
SK130999A3 (en) 2000-03-13
TW565450B (en) 2003-12-11
HRP980163B1 (en) 2002-10-31
ZA982609B (en) 1998-09-30
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EP0969832B1 (fr) 2001-07-04
AR012160A1 (es) 2000-09-27
CY2006005I1 (el) 2009-11-04
DZ2453A1 (fr) 2004-07-14
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FR2761266A1 (fr) 1998-10-02
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