RS50145B - Tetrahidropiridoetri - Google Patents

Tetrahidropiridoetri

Info

Publication number
RS50145B
RS50145B YUP-214/01A YU21401A RS50145B RS 50145 B RS50145 B RS 50145B YU 21401 A YU21401 A YU 21401A RS 50145 B RS50145 B RS 50145B
Authority
RS
Serbia
Prior art keywords
hydroxy
methoxypropoxy
methoxyethoxy
isopropoxy
ethoxy
Prior art date
Application number
YUP-214/01A
Other languages
English (en)
Inventor
Wolfgang-Alexander Simon
Wolfgang Kromer
Jorg Senn-Bilfinger
Stefan Postius
Gerhard Grundler
Guido Hanauer
Reinhard Huber
Ernst Sturm
Original Assignee
Altana Pharma Ag.,
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Altana Pharma Ag., filed Critical Altana Pharma Ag.,
Publication of YU21401A publication Critical patent/YU21401A/sh
Publication of RS50145B publication Critical patent/RS50145B/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)

Abstract

Jedinjenje formule I u kojoj R1 je metil ili hidroksimetil, jedan od supstituenata R2a i R2b je vodonik a drugi je hidroksi, metoksi, etoksi, izopropoksi, metoksietoksi ili metoksipropoksi, jedan od supstituenata R3a i R3b je vodonik a drugi je hidroksi, metoksi, etoksi, izopropoksi, metoksietoksi ili metoksipropoksi, gde R2a ili R2b s jedne strane i R3a ili R3b s druge strane nisu istovremeno hidroksi, i njegove soli. Prijava sadrži još 10 patentnih zahteva.
YUP-214/01A 1998-09-23 1999-09-17 Tetrahidropiridoetri RS50145B (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19843504 1998-09-23
EP98117988 1998-09-23

Publications (2)

Publication Number Publication Date
YU21401A YU21401A (sh) 2004-03-12
RS50145B true RS50145B (sr) 2009-03-25

Family

ID=26049024

Family Applications (1)

Application Number Title Priority Date Filing Date
YUP-214/01A RS50145B (sr) 1998-09-23 1999-09-17 Tetrahidropiridoetri

Country Status (31)

Country Link
US (4) US6436953B1 (sr)
EP (1) EP1115725B1 (sr)
JP (1) JP4145492B2 (sr)
KR (1) KR100668400B1 (sr)
CN (2) CN1155598C (sr)
AT (1) ATE231862T1 (sr)
AU (1) AU763463B2 (sr)
BG (1) BG65195B1 (sr)
BR (1) BR9914044A (sr)
CA (1) CA2344251A1 (sr)
CZ (1) CZ292335B6 (sr)
DE (1) DE69905178T2 (sr)
DK (1) DK1115725T3 (sr)
EA (1) EA005377B1 (sr)
EE (1) EE04677B1 (sr)
ES (1) ES2191464T3 (sr)
GE (1) GEP20032926B (sr)
HK (1) HK1038360B (sr)
HR (1) HRP20010224A2 (sr)
HU (1) HUP0102990A3 (sr)
ID (1) ID28896A (sr)
IL (2) IL142063A0 (sr)
NO (1) NO317304B1 (sr)
NZ (1) NZ510610A (sr)
PL (1) PL193616B1 (sr)
PT (1) PT1115725E (sr)
RS (1) RS50145B (sr)
SI (1) SI1115725T1 (sr)
SK (1) SK285165B6 (sr)
TR (1) TR200100805T2 (sr)
WO (1) WO2000017200A1 (sr)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU763463B2 (en) * 1998-09-23 2003-07-24 Takeda Gmbh Tetrahydropyridoethers
PT1173439E (pt) 1999-04-17 2003-10-31 Altana Pharma Ag Haloalcoxi imidazonaftiridinas
CA2285516C (en) * 1999-05-12 2010-12-07 President And Fellows Of Harvard College Dopamine transporter imaging agents
AU783633B2 (en) * 2000-03-29 2005-11-17 Altana Pharma Ag Prodrugs of imidazopyridine derivatives
PL365165A1 (en) * 2000-03-29 2004-12-27 Altana Pharma Ag Tricyclic imidazopyridines
MXPA03003706A (es) * 2000-10-25 2005-01-25 Altana Pharma Ag Imidazopiridinas polisustituidas, como inhibidores de secrecion gastrica.
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
CN1496259A (zh) * 2001-03-08 2004-05-12 新用途
US6927292B2 (en) 2001-08-02 2005-08-09 Altana Pharma Ag Tricyclic epoxides
JP2005504048A (ja) * 2001-08-03 2005-02-10 アルタナ　ファルマ　アクチエンゲゼルシャフト 胃腸障害治療用のアルカリ置換されたイミダゾピリジン
US20040235882A1 (en) * 2001-08-03 2004-11-25 Jorg Senn-Bilfinger Amino-substituted imidazopyridines for the treatment of gastrointestial diseases
KR20040081204A (ko) 2002-02-15 2004-09-20 알타나 파마 아게 트리시클릭 ｎ-아실 화합물
MY140561A (en) * 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
AU2003227710A1 (en) * 2002-05-07 2003-11-11 Altana Pharma Ag New combination of reversible proton pump inhibitors and airway therapeutics for treating airway disorders
EP1565465A1 (en) 2002-11-19 2005-08-24 ALTANA Pharma AG 8-substituted imidazopyridines
JP4755495B2 (ja) 2002-12-12 2011-08-24 ニコメッド ゲゼルシャフト ミット ベシュレンクテル ハフツング 組合せ医薬品
MXPA05006349A (es) * 2002-12-20 2005-08-26 Altana Pharma Ag 8-trialquisiloxi -2-metil -9-fenil -7- oxo-7, 8, 9, 10- tetrahidroimidazo [1, 2h] [1, 7].
MXPA05008490A (es) * 2003-02-17 2005-10-18 Altana Pharma Ag Combinaciones que contienen imidazopiridinas y su uso en el tratamiento de enfermedades gastrointestinales inflamatorias.
RS52908B (sr) 2003-03-10 2014-02-28 Takeda Gmbh Novi postupak za dobijanje roflumilasta
TW200503783A (en) * 2003-04-11 2005-02-01 Altana Pharma Ag Oral pharmaceutical preparation for proton pump antagonists
SA04250092B1 (ar) * 2003-05-14 2008-05-04 التانا فاروا ايه جي مركب وسيط جديد لتحضير مركبات إيميدازوبيريدين imidazopyridines فعالة علاجياً
WO2004105795A1 (en) * 2003-05-27 2004-12-09 Altana Pharma Ag Pharmaceutical combinations of a proton pump inhibitor and a compound which modifies gastrointestinal motility
EP1663313A2 (en) * 2003-08-29 2006-06-07 Dynogen Pharmaceuticals Inc. Compositions useful for treating gastrointestinal motility disorders
DK1670482T4 (da) 2003-09-16 2022-08-22 Covis Pharma B V Anvendelse af ciclesonid til behandlingen af respiratoriske sygdomme
CA2544325A1 (en) * 2003-11-03 2005-05-12 Astrazeneca Ab Imidazo [1,2-a] pyridine derivatives for the treatment of silent gastro-esophageal reflux
CA2549860A1 (en) 2003-12-19 2005-06-30 Altana Pharma Ag Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives
NZ549011A (en) * 2004-02-17 2009-04-30 Altana Pharma Ag Tricyclic imidazopyridines and intermediates for the synthesis thereof
PT1784402E (pt) 2004-09-03 2011-08-23 Yuhan Corp Derivados de pirrolo[3,2-c]piridina e processos para a sua preparação
WO2006025717A1 (en) 2004-09-03 2006-03-09 Yuhan Corporation PYRROLO[2,3-c]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF
RU2397170C2 (ru) 2004-09-03 2010-08-20 Юхан Корпорейшн ПРОИЗВОДНЫЕ ПИРРОЛО[3,2-b]ПИРИДИНА И СПОСОБЫ ИХ ПОЛУЧЕНИЯ
ES2421916T3 (es) * 2005-03-16 2013-09-06 Nycomed Gmbh Forma farmacéutica de sabor enmascarado que contiene roflumilast
EP2080513A1 (en) 2008-01-16 2009-07-22 Schraermeyer, Ulrich, Prof. Dr. rer. nat Tetrahydropyridoethers for treatment of AMD
KR101605063B1 (ko) 2009-07-09 2016-03-21 라퀄리아 파마 인코포레이티드 소화관 운동이상이 관여하는 질환의 치료용 산 펌프 길항제
WO2012027240A1 (en) * 2010-08-23 2012-03-01 Schering Corporation Fused tricyclic inhibitors of mammalian target of rapamycin
WO2013187727A1 (en) * 2012-06-15 2013-12-19 Bio-Pharm Solutions Co., Ltd. Phenylalkyl sulfamate compound and muscle relaxant composition comprising the same
WO2015052256A1 (en) 2013-10-08 2015-04-16 Katairo Gmbh Tetrahydropyridoethers for the treatment of stargardt's disease

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4468400A (en) * 1982-12-20 1984-08-28 Schering Corporation Antiulcer tricyclic imidazo [1,2-a]pyridines
US5112834A (en) 1987-07-16 1992-05-12 Byk Gulden Lomberg Chemische Fabrik Gmbh Imidazole protectorant for the stomach and intestine
SE9401197D0 (sv) * 1994-04-11 1994-04-11 Astra Ab Active compounds
WO1996003404A1 (de) * 1994-07-28 1996-02-08 Byk Gulden Lomberg Chemische Fabrik Gmbh Acylimidazopyridine
CN1251102A (zh) * 1997-03-24 2000-04-19 比克·古尔顿·劳姆贝尔格化学公司 四氢吡啶并化合物
WO1998042707A1 (en) * 1997-03-24 1998-10-01 Byk Gulden Lomberg Chemische Fabrik Gmbh Tetrahydropyrido compounds
AU763463B2 (en) 1998-09-23 2003-07-24 Takeda Gmbh Tetrahydropyridoethers

Also Published As

Publication number Publication date
ATE231862T1 (de) 2003-02-15
EP1115725B1 (en) 2003-01-29
PL193616B1 (pl) 2007-02-28
US20040162310A1 (en) 2004-08-19
EA200100315A1 (ru) 2001-10-22
IL142063A0 (en) 2002-03-10
SK285165B6 (sk) 2006-07-07
US6696460B2 (en) 2004-02-24
SI1115725T1 (en) 2003-06-30
PT1115725E (pt) 2003-06-30
CN1560055A (zh) 2005-01-05
TR200100805T2 (tr) 2001-08-21
JP4145492B2 (ja) 2008-09-03
NZ510610A (en) 2003-07-25
ID28896A (id) 2001-07-12
EP1115725A1 (en) 2001-07-18
EE04677B1 (et) 2006-08-15
BG65195B1 (bg) 2007-06-29
GEP20032926B (en) 2003-03-25
US6436953B1 (en) 2002-08-20
CZ292335B6 (cs) 2003-09-17
DK1115725T3 (da) 2003-06-23
HRP20010224A2 (en) 2002-04-30
IL142063A (en) 2007-10-31
JP2002526499A (ja) 2002-08-20
HK1038360A1 (en) 2002-03-15
BG105270A (en) 2001-11-30
CN1319101A (zh) 2001-10-24
WO2000017200A1 (en) 2000-03-30
PL346617A1 (en) 2002-02-25
CN100506821C (zh) 2009-07-01
AU6192099A (en) 2000-04-10
US20020169320A1 (en) 2002-11-14
EE200100172A (et) 2002-06-17
CA2344251A1 (en) 2000-03-30
KR100668400B1 (ko) 2007-01-17
NO20011243L (no) 2001-03-12
DE69905178D1 (de) 2003-03-06
NO317304B1 (no) 2004-10-04
KR20010075223A (ko) 2001-08-09
EA005377B1 (ru) 2005-02-24
ES2191464T3 (es) 2003-09-01
HUP0102990A3 (en) 2002-09-30
CZ20011082A3 (cs) 2001-09-12
US7105676B2 (en) 2006-09-12
SK3992001A3 (en) 2001-12-03
AU763463B2 (en) 2003-07-24
US7393860B1 (en) 2008-07-01
NO20011243D0 (no) 2001-03-12
DE69905178T2 (de) 2003-07-17
HK1038360B (zh) 2003-05-16
BR9914044A (pt) 2001-12-04
CN1155598C (zh) 2004-06-30
HUP0102990A2 (hu) 2002-01-28
YU21401A (sh) 2004-03-12

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