BR9914044A - ésteres tetrahidropirido - Google Patents
ésteres tetrahidropiridoInfo
- Publication number
- BR9914044A BR9914044A BR9914044-6A BR9914044A BR9914044A BR 9914044 A BR9914044 A BR 9914044A BR 9914044 A BR9914044 A BR 9914044A BR 9914044 A BR9914044 A BR 9914044A
- Authority
- BR
- Brazil
- Prior art keywords
- esters
- tetrahydropyride
- tetrahydropirid
- substituents
- prevention
- Prior art date
Links
- 150000002148 esters Chemical class 0.000 title abstract 2
- 208000018522 Gastrointestinal disease Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Communicable Diseases (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Oncology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Patente de Invenção: "éSTERES TETRAHIDROPIRIDO".Compostos da fórmula (I), nos quais os substituintes que possuemos significados mencionados na descrição, são apropriados paraprevenção e tratamento de doenças gastrintestinais.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19843504 | 1998-09-23 | ||
EP98117988 | 1998-09-23 | ||
PCT/EP1999/006899 WO2000017200A1 (en) | 1998-09-23 | 1999-09-17 | Tetrahydropyridoethers |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9914044A true BR9914044A (pt) | 2001-12-04 |
Family
ID=26049024
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9914044-6A BR9914044A (pt) | 1998-09-23 | 1999-09-17 | ésteres tetrahidropirido |
Country Status (31)
Country | Link |
---|---|
US (4) | US6436953B1 (pt) |
EP (1) | EP1115725B1 (pt) |
JP (1) | JP4145492B2 (pt) |
KR (1) | KR100668400B1 (pt) |
CN (2) | CN1155598C (pt) |
AT (1) | ATE231862T1 (pt) |
AU (1) | AU763463B2 (pt) |
BG (1) | BG65195B1 (pt) |
BR (1) | BR9914044A (pt) |
CA (1) | CA2344251A1 (pt) |
CZ (1) | CZ292335B6 (pt) |
DE (1) | DE69905178T2 (pt) |
DK (1) | DK1115725T3 (pt) |
EA (1) | EA005377B1 (pt) |
EE (1) | EE04677B1 (pt) |
ES (1) | ES2191464T3 (pt) |
GE (1) | GEP20032926B (pt) |
HK (1) | HK1038360B (pt) |
HR (1) | HRP20010224A2 (pt) |
HU (1) | HUP0102990A3 (pt) |
ID (1) | ID28896A (pt) |
IL (2) | IL142063A0 (pt) |
NO (1) | NO317304B1 (pt) |
NZ (1) | NZ510610A (pt) |
PL (1) | PL193616B1 (pt) |
PT (1) | PT1115725E (pt) |
RS (1) | RS50145B (pt) |
SI (1) | SI1115725T1 (pt) |
SK (1) | SK285165B6 (pt) |
TR (1) | TR200100805T2 (pt) |
WO (1) | WO2000017200A1 (pt) |
Families Citing this family (36)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA005377B1 (ru) | 1998-09-23 | 2005-02-24 | Алтана Фарма Аг | ТЕТРАГИДРОИМИДАЗО [1,2-h][1,7] НАФТИРИДИНОВЫЕ СОЕДИНЕНИЯ |
DK1173439T3 (da) | 1999-04-17 | 2003-09-08 | Altana Pharma Ag | Halogenalkoxy-imidazonaphthyridiner |
CA2721484A1 (en) * | 1999-05-12 | 2000-11-12 | President And Fellows Of Harvard College | Dopamine transporter imaging agents |
AU783724B2 (en) * | 2000-03-29 | 2005-12-01 | Altana Pharma Ag | Tricyclic imidazopyridines |
IL151200A0 (en) * | 2000-03-29 | 2003-04-10 | Altana Pharma Ag | Tricyclic imidazopyridine prodrug derivatives and pharmaceutical compositions containing the same |
US6869949B2 (en) * | 2000-10-25 | 2005-03-22 | Altana Pharma Ag | Polysubstituted imidazopyridines as gastric secretion inhibitors |
UA80393C2 (uk) | 2000-12-07 | 2007-09-25 | Алтана Фарма Аг | Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці |
US20040082605A1 (en) * | 2001-03-08 | 2004-04-29 | Arne Eek | Use |
CA2452802A1 (en) | 2001-08-02 | 2003-02-20 | Altana Pharma Ag | Tricyclic epoxides |
EP1417208A1 (en) * | 2001-08-03 | 2004-05-12 | ALTANA Pharma AG | Amino-substituted imidazopyridines for the treatment of gastrointestinal diseases |
PL368586A1 (en) * | 2001-08-03 | 2005-04-04 | Altana Pharma Ag | Alkyl-substituted imidazopyridines for the treatment of gastrointestinal disorders |
MXPA04007895A (es) | 2002-02-15 | 2004-10-15 | Altana Pharma Ag | Compuestos n-acilo triciclicos. |
MY140561A (en) * | 2002-02-20 | 2009-12-31 | Nycomed Gmbh | Dosage form containing pde 4 inhibitor as active ingredient |
JP2005528418A (ja) * | 2002-05-07 | 2005-09-22 | アルタナ ファルマ アクチエンゲゼルシャフト | 気道疾患を治療するための新規組み合わせ |
JP2006508142A (ja) | 2002-11-19 | 2006-03-09 | アルタナ ファルマ アクチエンゲゼルシャフト | 8−置換イミダゾピリジン |
EP1572217B1 (en) | 2002-12-12 | 2008-08-20 | Nycomed GmbH | Combination medicament of r,r-formoterol and ciclesonide |
BR0316752A (pt) * | 2002-12-20 | 2005-10-25 | Altana Pharma Ag | Silil éteres |
MXPA05008490A (es) * | 2003-02-17 | 2005-10-18 | Altana Pharma Ag | Combinaciones que contienen imidazopiridinas y su uso en el tratamiento de enfermedades gastrointestinales inflamatorias. |
US7470791B2 (en) | 2003-03-10 | 2008-12-30 | Nycomed Gmbh | Process for the preparation of roflumilast |
TW200503783A (en) * | 2003-04-11 | 2005-02-01 | Altana Pharma Ag | Oral pharmaceutical preparation for proton pump antagonists |
SA04250092B1 (ar) * | 2003-05-14 | 2008-05-04 | التانا فاروا ايه جي | مركب وسيط جديد لتحضير مركبات إيميدازوبيريدين imidazopyridines فعالة علاجياً |
US20060241134A1 (en) * | 2003-05-27 | 2006-10-26 | Altana Pharma Ga | Pharmaceutical combinations of a proton pump inhibitor and a compound which modifies gastrointestinal motility |
BRPI0414046A (pt) * | 2003-08-29 | 2006-10-24 | Dynogen Pharmaceuticals Inc | método de tratamento de um distúrbio de motilidade gastrintestinal, de tratamento de "gerd", de "gerd" noturno, composição farmacêutica, kit que compreende um composto e método para aumentar a motilidade esofágica em um paciente |
PT1670482E (pt) | 2003-09-16 | 2014-03-12 | Takeda Gmbh | Utilização de ciclesonida para o tratamento de doenças respiratórias |
EP1974730A1 (en) | 2003-11-03 | 2008-10-01 | AstraZeneca AB | Imidazo[1,2-a]pyridine derivatives for use in the treatment of sleep disturbance due to silent gastro-esophageal reflux |
AU2004298453A1 (en) | 2003-12-19 | 2005-06-30 | Altana Pharma Ag | Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives |
NZ549011A (en) * | 2004-02-17 | 2009-04-30 | Altana Pharma Ag | Tricyclic imidazopyridines and intermediates for the synthesis thereof |
WO2006025714A1 (en) | 2004-09-03 | 2006-03-09 | Yuhan Corporation | PYRROLO[3,2-c]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF |
CN101010321B (zh) | 2004-09-03 | 2011-10-26 | 株式会社柳韩洋行 | 吡咯并[3,2-b]吡啶衍生物及其制备方法 |
JP4898683B2 (ja) | 2004-09-03 | 2012-03-21 | ユーハン・コーポレイション | ピロロ[2,3−c]ピリジン誘導体及びその製造方法 |
ES2421916T3 (es) * | 2005-03-16 | 2013-09-06 | Nycomed Gmbh | Forma farmacéutica de sabor enmascarado que contiene roflumilast |
EP2080513A1 (en) | 2008-01-16 | 2009-07-22 | Schraermeyer, Ulrich, Prof. Dr. rer. nat | Tetrahydropyridoethers for treatment of AMD |
CN105919998B (zh) | 2009-07-09 | 2021-08-24 | 拉夸里亚创药株式会社 | 用于治疗与异常肠胃运动有关的疾病的酸泵拮抗剂 |
WO2012027240A1 (en) * | 2010-08-23 | 2012-03-01 | Schering Corporation | Fused tricyclic inhibitors of mammalian target of rapamycin |
US9221783B2 (en) * | 2012-06-15 | 2015-12-29 | Bio-Pharm Solutions Co., Ltd. | Phenylalkyl sulfamate compound and muscle relaxant composition comprising the same |
US20160235724A1 (en) | 2013-10-08 | 2016-08-18 | Katairo Gmbh | Tetrahydropyridoethers for the treatment of stargardt's disease |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4468400A (en) * | 1982-12-20 | 1984-08-28 | Schering Corporation | Antiulcer tricyclic imidazo [1,2-a]pyridines |
DE3855692D1 (de) | 1987-07-16 | 1997-01-16 | Byk Gulden Lomberg Chem Fab | Imidazo[1,2-a]pyridine |
SE9401197D0 (sv) * | 1994-04-11 | 1994-04-11 | Astra Ab | Active compounds |
WO1996003404A1 (de) * | 1994-07-28 | 1996-02-08 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Acylimidazopyridine |
WO1998042707A1 (en) * | 1997-03-24 | 1998-10-01 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Tetrahydropyrido compounds |
PT971922E (pt) * | 1997-03-24 | 2004-09-30 | Altana Pharma Ag | Compostos de tetra-hidropirido |
EA005377B1 (ru) * | 1998-09-23 | 2005-02-24 | Алтана Фарма Аг | ТЕТРАГИДРОИМИДАЗО [1,2-h][1,7] НАФТИРИДИНОВЫЕ СОЕДИНЕНИЯ |
-
1999
- 1999-09-17 EA EA200100315A patent/EA005377B1/ru not_active IP Right Cessation
- 1999-09-17 RS YUP-214/01A patent/RS50145B/sr unknown
- 1999-09-17 SI SI9930207T patent/SI1115725T1/xx unknown
- 1999-09-17 KR KR1020017003553A patent/KR100668400B1/ko not_active IP Right Cessation
- 1999-09-17 CN CNB998112992A patent/CN1155598C/zh not_active Expired - Fee Related
- 1999-09-17 SK SK399-2001A patent/SK285165B6/sk not_active IP Right Cessation
- 1999-09-17 ES ES99948776T patent/ES2191464T3/es not_active Expired - Lifetime
- 1999-09-17 CA CA002344251A patent/CA2344251A1/en not_active Abandoned
- 1999-09-17 JP JP2000574109A patent/JP4145492B2/ja not_active Expired - Lifetime
- 1999-09-17 AT AT99948776T patent/ATE231862T1/de not_active IP Right Cessation
- 1999-09-17 NZ NZ510610A patent/NZ510610A/en unknown
- 1999-09-17 EE EEP200100172A patent/EE04677B1/xx not_active IP Right Cessation
- 1999-09-17 DK DK99948776T patent/DK1115725T3/da active
- 1999-09-17 US US09/582,212 patent/US6436953B1/en not_active Expired - Lifetime
- 1999-09-17 PL PL99346617A patent/PL193616B1/pl not_active IP Right Cessation
- 1999-09-17 EP EP99948776A patent/EP1115725B1/en not_active Expired - Lifetime
- 1999-09-17 TR TR2001/00805T patent/TR200100805T2/xx unknown
- 1999-09-17 GE GEAP19995786A patent/GEP20032926B/en unknown
- 1999-09-17 CZ CZ20011082A patent/CZ292335B6/cs not_active IP Right Cessation
- 1999-09-17 HU HU0102990A patent/HUP0102990A3/hu unknown
- 1999-09-17 PT PT99948776T patent/PT1115725E/pt unknown
- 1999-09-17 CN CNB2004100384351A patent/CN100506821C/zh not_active Expired - Fee Related
- 1999-09-17 DE DE69905178T patent/DE69905178T2/de not_active Expired - Lifetime
- 1999-09-17 IL IL14206399A patent/IL142063A0/xx active IP Right Grant
- 1999-09-17 ID IDW20010682A patent/ID28896A/id unknown
- 1999-09-17 AU AU61920/99A patent/AU763463B2/en not_active Expired
- 1999-09-17 BR BR9914044-6A patent/BR9914044A/pt not_active Application Discontinuation
- 1999-09-17 WO PCT/EP1999/006899 patent/WO2000017200A1/en active IP Right Grant
-
2001
- 2001-02-19 BG BG105270A patent/BG65195B1/bg unknown
- 2001-03-12 NO NO20011243A patent/NO317304B1/no not_active IP Right Cessation
- 2001-03-18 IL IL142063A patent/IL142063A/en not_active IP Right Cessation
- 2001-03-23 HR HR20010224A patent/HRP20010224A2/hr not_active Application Discontinuation
-
2002
- 2002-01-03 HK HK02100042.6A patent/HK1038360B/zh not_active IP Right Cessation
- 2002-03-25 US US10/103,733 patent/US6696460B2/en not_active Expired - Lifetime
-
2004
- 2004-02-23 US US10/783,512 patent/US7105676B2/en not_active Expired - Lifetime
-
2006
- 2006-07-27 US US11/493,707 patent/US7393860B1/en not_active Expired - Fee Related
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B25D | Requested change of name of applicant approved | ||
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B15K | Others concerning applications: alteration of classification |
Free format text: ALTERADA DE INT.CL: C07D 471/14, A61K 31/435 Ipc: C07D 471/14 (2009.01), A61K 31/4375 (2009.01), A61 |
|
B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8, 11 E 13 DA LPI |
|
B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL. |