EA200001212A1 - Усовершенствованный способ получения производных норбензоморфана с ценными фармацевтическими свойствами - Google Patents
Усовершенствованный способ получения производных норбензоморфана с ценными фармацевтическими свойствамиInfo
- Publication number
- EA200001212A1 EA200001212A1 EA200001212A EA200001212A EA200001212A1 EA 200001212 A1 EA200001212 A1 EA 200001212A1 EA 200001212 A EA200001212 A EA 200001212A EA 200001212 A EA200001212 A EA 200001212A EA 200001212 A1 EA200001212 A1 EA 200001212A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- norbenzomorphan
- derivatives
- producing
- improved method
- pharmaceutical properties
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/22—Bridged ring systems
- C07D221/26—Benzomorphans
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
Abstract
В заявке описывается новый способ получения производных норбензоморфана общей формулы (1).Международная заявка была опубликована вместе с отчетом о международном поиске.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19822822A DE19822822A1 (de) | 1998-05-20 | 1998-05-20 | Verbessertes Verfahren zur Herstellung von pharmazeutisch wertvollen Norbenzomorphanderivaten |
PCT/EP1999/003142 WO1999059976A1 (de) | 1998-05-20 | 1999-05-07 | Verbessertes verfahren zur herstellung von pharmazeutisch wertvollen norbenzomorphanderivaten |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200001212A1 true EA200001212A1 (ru) | 2001-04-23 |
EA003059B1 EA003059B1 (ru) | 2002-12-26 |
Family
ID=7868527
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200001212A EA003059B1 (ru) | 1998-05-20 | 1999-05-07 | Усовершенствованный способ получения производных норбензоморфана с ценными фармацевтическими свойствами |
Country Status (38)
Country | Link |
---|---|
US (1) | US6124459A (ru) |
EP (1) | EP1080076B1 (ru) |
JP (1) | JP4526185B2 (ru) |
KR (1) | KR20010043703A (ru) |
CN (1) | CN1113058C (ru) |
AR (1) | AR016040A1 (ru) |
AT (1) | ATE254605T1 (ru) |
AU (1) | AU753563B2 (ru) |
BG (1) | BG104964A (ru) |
BR (1) | BR9910603A (ru) |
CA (1) | CA2330669C (ru) |
CO (1) | CO5060460A1 (ru) |
DE (2) | DE19822822A1 (ru) |
DK (1) | DK1080076T3 (ru) |
EA (1) | EA003059B1 (ru) |
EE (1) | EE04305B1 (ru) |
EG (1) | EG21526A (ru) |
ES (1) | ES2211093T3 (ru) |
HK (1) | HK1035728A1 (ru) |
HR (1) | HRP20000793A2 (ru) |
HU (1) | HUP0102034A3 (ru) |
ID (1) | ID27014A (ru) |
IL (1) | IL138998A0 (ru) |
MY (1) | MY120806A (ru) |
NO (1) | NO317302B1 (ru) |
NZ (1) | NZ508845A (ru) |
PE (1) | PE20000558A1 (ru) |
PL (1) | PL343935A1 (ru) |
PT (1) | PT1080076E (ru) |
SI (1) | SI1080076T1 (ru) |
SK (1) | SK283996B6 (ru) |
TR (1) | TR200003360T2 (ru) |
TW (1) | TW455582B (ru) |
UA (1) | UA59448C2 (ru) |
UY (1) | UY25515A1 (ru) |
WO (1) | WO1999059976A1 (ru) |
YU (1) | YU71400A (ru) |
ZA (1) | ZA200005740B (ru) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7405149B1 (en) * | 1998-12-21 | 2008-07-29 | Megica Corporation | Post passivation method for semiconductor chip or wafer |
WO2016044546A1 (en) * | 2014-09-17 | 2016-03-24 | Purdue Pharma L.P. | Benzomorphan analogs and the use thereof |
CN107089948B (zh) * | 2017-04-28 | 2020-07-17 | 云南大学 | 吗吩衍生物及其制备方法和应用 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IE34235B1 (en) * | 1969-06-04 | 1975-03-19 | Acf Chemiefarma Nv | 6,7-benzomorphans and their preparation |
US4255579A (en) * | 1974-05-20 | 1981-03-10 | Sterling Drug Inc. | 11-Substituted hexahydro-2,6-methano-3-benzazocines |
US3932422A (en) * | 1974-05-20 | 1976-01-13 | Sterling Drug Inc. | 8-Methylene-3-azabicyclo[3.3.1]non-6-en-4-ones |
DE19528472A1 (de) * | 1995-08-03 | 1997-02-06 | Boehringer Ingelheim Kg | Neues Verfahren zur Herstellung von Norbenzomorphan einer Zwischenstufe bei Herstellung von pharmazeutisch wertvollen Benzomorphanderivaten, insbesondere von (-)-(1R,5S,S"R)-3'-Hydroxy-2-(2-methoxypropyl-)-5,9,9-trimethyl-6,7 benzomorphan |
-
1998
- 1998-05-20 DE DE19822822A patent/DE19822822A1/de not_active Withdrawn
-
1999
- 1999-05-07 TR TR2000/03360T patent/TR200003360T2/xx unknown
- 1999-05-07 AU AU41399/99A patent/AU753563B2/en not_active Ceased
- 1999-05-07 IL IL13899899A patent/IL138998A0/xx unknown
- 1999-05-07 EE EEP200000674A patent/EE04305B1/xx not_active IP Right Cessation
- 1999-05-07 EP EP99924901A patent/EP1080076B1/de not_active Expired - Lifetime
- 1999-05-07 SK SK1731-2000A patent/SK283996B6/sk unknown
- 1999-05-07 PL PL99343935A patent/PL343935A1/xx not_active IP Right Cessation
- 1999-05-07 ES ES99924901T patent/ES2211093T3/es not_active Expired - Lifetime
- 1999-05-07 DE DE59907804T patent/DE59907804D1/de not_active Expired - Lifetime
- 1999-05-07 EA EA200001212A patent/EA003059B1/ru not_active IP Right Cessation
- 1999-05-07 DK DK99924901T patent/DK1080076T3/da active
- 1999-05-07 SI SI9930488T patent/SI1080076T1/xx unknown
- 1999-05-07 CA CA002330669A patent/CA2330669C/en not_active Expired - Fee Related
- 1999-05-07 NZ NZ508845A patent/NZ508845A/xx unknown
- 1999-05-07 CN CN99806339A patent/CN1113058C/zh not_active Expired - Fee Related
- 1999-05-07 AT AT99924901T patent/ATE254605T1/de not_active IP Right Cessation
- 1999-05-07 PT PT99924901T patent/PT1080076E/pt unknown
- 1999-05-07 ID IDW20002394A patent/ID27014A/id unknown
- 1999-05-07 JP JP2000549595A patent/JP4526185B2/ja not_active Expired - Fee Related
- 1999-05-07 HU HU0102034A patent/HUP0102034A3/hu unknown
- 1999-05-07 BR BR9910603-5A patent/BR9910603A/pt not_active IP Right Cessation
- 1999-05-07 KR KR1020007012923A patent/KR20010043703A/ko not_active Application Discontinuation
- 1999-05-07 WO PCT/EP1999/003142 patent/WO1999059976A1/de not_active Application Discontinuation
- 1999-05-07 YU YU71400A patent/YU71400A/sh unknown
- 1999-05-17 EG EG56999A patent/EG21526A/xx active
- 1999-05-17 US US09/313,001 patent/US6124459A/en not_active Expired - Lifetime
- 1999-05-17 PE PE1999000413A patent/PE20000558A1/es not_active Application Discontinuation
- 1999-05-18 TW TW088108090A patent/TW455582B/zh not_active IP Right Cessation
- 1999-05-18 CO CO99030491A patent/CO5060460A1/es unknown
- 1999-05-18 UY UY25515A patent/UY25515A1/es not_active IP Right Cessation
- 1999-05-19 AR ARP990102374A patent/AR016040A1/es not_active Suspension/Interruption
- 1999-05-19 MY MYPI99001967A patent/MY120806A/en unknown
- 1999-07-05 UA UA2000127360A patent/UA59448C2/ru unknown
-
2000
- 2000-10-17 ZA ZA200005740A patent/ZA200005740B/xx unknown
- 2000-11-17 NO NO20005818A patent/NO317302B1/no unknown
- 2000-11-17 BG BG104964A patent/BG104964A/xx active Pending
- 2000-11-17 HR HR20000793A patent/HRP20000793A2/hr not_active Application Discontinuation
-
2001
- 2001-09-12 HK HK01106427A patent/HK1035728A1/xx not_active IP Right Cessation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PD4A | Registration of transfer of a eurasian patent in accordance with the succession in title | ||
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |