ATE181551T1 - Taxol-derivate - Google Patents

Taxol-derivate

Info

Publication number
ATE181551T1
ATE181551T1 AT93912249T AT93912249T ATE181551T1 AT E181551 T1 ATE181551 T1 AT E181551T1 AT 93912249 T AT93912249 T AT 93912249T AT 93912249 T AT93912249 T AT 93912249T AT E181551 T1 ATE181551 T1 AT E181551T1
Authority
AT
Austria
Prior art keywords
taxol derivatives
taxol
derivatives
compounds
chain
Prior art date
Application number
AT93912249T
Other languages
English (en)
Inventor
Geewananda P Gunawardana
Larry L Klein
James B Mcalpine
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Application granted granted Critical
Publication of ATE181551T1 publication Critical patent/ATE181551T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
AT93912249T 1992-04-17 1993-04-14 Taxol-derivate ATE181551T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US87050992A 1992-04-17 1992-04-17
US91472092A 1992-07-16 1992-07-16

Publications (1)

Publication Number Publication Date
ATE181551T1 true ATE181551T1 (de) 1999-07-15

Family

ID=27128160

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93912249T ATE181551T1 (de) 1992-04-17 1993-04-14 Taxol-derivate

Country Status (15)

Country Link
US (3) US5352806A (de)
EP (1) EP0639186B1 (de)
JP (1) JPH07505887A (de)
KR (1) KR100263496B1 (de)
AT (1) ATE181551T1 (de)
AU (1) AU672006B2 (de)
CA (1) CA2130578A1 (de)
DE (1) DE69325454T2 (de)
DK (1) DK0639186T3 (de)
ES (1) ES2134847T3 (de)
GR (1) GR3031126T3 (de)
IL (3) IL105421A (de)
MX (1) MX9302214A (de)
PH (1) PH31610A (de)
WO (1) WO1993021173A1 (de)

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FR2601675B1 (fr) * 1986-07-17 1988-09-23 Rhone Poulenc Sante Derives du taxol, leur preparation et les compositions pharmaceutiques qui les contiennent
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FR2629818B1 (fr) * 1988-04-06 1990-11-16 Centre Nat Rech Scient Procede de preparation du taxol
FR2629819B1 (fr) * 1988-04-06 1990-11-16 Rhone Poulenc Sante Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii
US5175315A (en) * 1989-05-31 1992-12-29 Florida State University Method for preparation of taxol using β-lactam
CA2023645C (fr) * 1989-08-23 2002-03-26 Jean-Noel Denis Procede pour la preparation enantioselective de derives de la phenylisoserine
US5015744A (en) * 1989-11-14 1991-05-14 Florida State University Method for preparation of taxol using an oxazinone
FR2658513B1 (fr) * 1990-02-21 1994-02-04 Rhone Poulenc Sante Procede de preparation de l'acide cis-beta-phenylglycidique-(2r,3r).
FR2658510B1 (fr) * 1990-02-21 1992-04-30 Rhone Poulenc Sante Nouveau derive de la beta-phenylisoserine, sa preparation et son emploi.
US5200534A (en) * 1992-03-13 1993-04-06 University Of Florida Process for the preparation of taxol and 10-deacetyltaxol
FR2711370B1 (fr) * 1993-10-18 1996-01-05 Rhone Poulenc Rorer Sa Nouveaux taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.

Also Published As

Publication number Publication date
AU4286393A (en) 1993-11-18
WO1993021173A1 (en) 1993-10-28
AU672006B2 (en) 1996-09-19
DK0639186T3 (da) 1999-12-13
MX9302214A (es) 1993-10-01
CA2130578A1 (en) 1993-10-28
PH31610A (en) 1998-11-03
DE69325454D1 (de) 1999-07-29
EP0639186B1 (de) 1999-06-23
DE69325454T2 (de) 2000-01-20
KR100263496B1 (ko) 2002-01-09
KR950700894A (ko) 1995-02-20
US5594157A (en) 1997-01-14
IL126339A0 (en) 1999-05-09
US5530020A (en) 1996-06-25
JPH07505887A (ja) 1995-06-29
US5352806A (en) 1994-10-04
ES2134847T3 (es) 1999-10-16
IL105421A0 (en) 1993-08-18
EP0639186A4 (de) 1995-01-10
IL105421A (en) 1999-09-22
GR3031126T3 (en) 1999-12-31
IL126339A (en) 2001-03-19
EP0639186A1 (de) 1995-02-22

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