DK1252157T3 - Pyrimidin-carboxamider anvendelige som inhibitorer af PDE4 isozymer - Google Patents

Pyrimidin-carboxamider anvendelige som inhibitorer af PDE4 isozymer

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Publication number
DK1252157T3
DK1252157T3 DK01901334T DK01901334T DK1252157T3 DK 1252157 T3 DK1252157 T3 DK 1252157T3 DK 01901334 T DK01901334 T DK 01901334T DK 01901334 T DK01901334 T DK 01901334T DK 1252157 T3 DK1252157 T3 DK 1252157T3
Authority
DK
Denmark
Prior art keywords
inhibitors
pde4 isozymes
carboxamides useful
pyrimidine carboxamides
pyrimidine
Prior art date
Application number
DK01901334T
Other languages
Danish (da)
English (en)
Inventor
Robert James Chambers
Thomas Victor Magee
Anthony Marfat
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of DK1252157T3 publication Critical patent/DK1252157T3/da

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
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  • Health & Medical Sciences (AREA)
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  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
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  • Virology (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurology (AREA)
  • Communicable Diseases (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
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  • Urology & Nephrology (AREA)
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  • Biotechnology (AREA)
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  • Ophthalmology & Optometry (AREA)
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DK01901334T 2000-01-31 2001-01-30 Pyrimidin-carboxamider anvendelige som inhibitorer af PDE4 isozymer DK1252157T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17928200P 2000-01-31 2000-01-31
EP01901334A EP1252157B1 (de) 2000-01-31 2001-01-30 Pyrimidinylcarboxamiden als inhibitoren der pde4 isoenzyme

Publications (1)

Publication Number Publication Date
DK1252157T3 true DK1252157T3 (da) 2004-10-25

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DK01901334T DK1252157T3 (da) 2000-01-31 2001-01-30 Pyrimidin-carboxamider anvendelige som inhibitorer af PDE4 isozymer

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US (1) US6740655B2 (de)
EP (1) EP1252157B1 (de)
JP (1) JP2003522165A (de)
KR (1) KR20020071029A (de)
CN (1) CN1404480A (de)
AP (1) AP2002002590A0 (de)
AR (1) AR027336A1 (de)
AT (1) ATE269860T1 (de)
AU (1) AU2700301A (de)
BG (1) BG106868A (de)
BR (1) BR0107934A (de)
CA (1) CA2396458C (de)
CO (1) CO5271669A1 (de)
CR (1) CR6714A (de)
CZ (1) CZ20022413A3 (de)
DE (1) DE60103976T2 (de)
DK (1) DK1252157T3 (de)
DZ (1) DZ3406A1 (de)
EA (1) EA005028B1 (de)
EE (1) EE200200426A (de)
ES (1) ES2223772T3 (de)
GE (1) GEP20043385B (de)
GT (1) GT200100023A (de)
HK (1) HK1054232A1 (de)
HN (1) HN2001000018A (de)
HU (1) HUP0204271A3 (de)
IL (1) IL150486A0 (de)
IS (1) IS6444A (de)
MA (1) MA26871A1 (de)
MX (1) MXPA02007465A (de)
NO (1) NO20023614L (de)
NZ (1) NZ519726A (de)
OA (1) OA12170A (de)
PA (1) PA8511301A1 (de)
PE (1) PE20011059A1 (de)
PL (1) PL357555A1 (de)
PT (1) PT1252157E (de)
SK (1) SK10342002A3 (de)
SV (1) SV2001000298A (de)
TN (1) TNSN01019A1 (de)
TR (1) TR200402292T4 (de)
UY (1) UY26570A1 (de)
WO (1) WO2001057025A1 (de)
ZA (1) ZA200206034B (de)

Families Citing this family (85)

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Publication number Priority date Publication date Assignee Title
ES2165768B1 (es) 1999-07-14 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen.
EP1248597B1 (de) * 1999-12-24 2005-03-30 Glaxo Group Limited Pharmazeutische aerosol formulierung enthaltend salmeterol und fluticason
DE10110772A1 (de) * 2001-03-07 2002-09-12 Boehringer Ingelheim Pharma Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und PDE-IV-Inhibitoren
US7776315B2 (en) 2000-10-31 2010-08-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmaceutical compositions based on anticholinergics and additional active ingredients
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