DK1228067T3 - 5-leddede heterocykliske forbindelser med hypoglykæmisk og hypolipidæmisk virkning - Google Patents
5-leddede heterocykliske forbindelser med hypoglykæmisk og hypolipidæmisk virkningInfo
- Publication number
- DK1228067T3 DK1228067T3 DK00974857T DK00974857T DK1228067T3 DK 1228067 T3 DK1228067 T3 DK 1228067T3 DK 00974857 T DK00974857 T DK 00974857T DK 00974857 T DK00974857 T DK 00974857T DK 1228067 T3 DK1228067 T3 DK 1228067T3
- Authority
- DK
- Denmark
- Prior art keywords
- hypoglycemic
- membered heterocyclic
- heterocyclic compounds
- hypolipidemic activity
- hypolipidemic
- Prior art date
Links
Classifications
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- C07—ORGANIC CHEMISTRY
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- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
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- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP32031799 | 1999-11-10 | ||
JP35223799 | 1999-12-10 | ||
PCT/JP2000/007877 WO2001038325A1 (fr) | 1999-11-10 | 2000-11-09 | Composes heterocycliques n a 5 elements a activite hypoglycemique et hypolipidemique |
Publications (1)
Publication Number | Publication Date |
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DK1228067T3 true DK1228067T3 (da) | 2004-12-06 |
Family
ID=26570043
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK00974857T DK1228067T3 (da) | 1999-11-10 | 2000-11-09 | 5-leddede heterocykliske forbindelser med hypoglykæmisk og hypolipidæmisk virkning |
Country Status (30)
Country | Link |
---|---|
US (1) | US7179823B1 (fr) |
EP (2) | EP1228067B1 (fr) |
JP (2) | JP3723071B2 (fr) |
KR (1) | KR100518142B1 (fr) |
CN (1) | CN1260227C (fr) |
AR (1) | AR026414A1 (fr) |
AT (1) | ATE271049T1 (fr) |
AU (1) | AU780948C (fr) |
BR (1) | BR0015466A (fr) |
CA (1) | CA2390923A1 (fr) |
CO (1) | CO5261501A1 (fr) |
CZ (1) | CZ20021604A3 (fr) |
DE (1) | DE60012213T2 (fr) |
DK (1) | DK1228067T3 (fr) |
ES (1) | ES2225252T3 (fr) |
HK (1) | HK1045991B (fr) |
HU (1) | HUP0203165A3 (fr) |
IL (1) | IL149493A0 (fr) |
MX (1) | MXPA02004647A (fr) |
MY (1) | MY141468A (fr) |
NO (1) | NO20022108L (fr) |
NZ (1) | NZ519238A (fr) |
PE (1) | PE20011021A1 (fr) |
PL (1) | PL356487A1 (fr) |
PT (1) | PT1228067E (fr) |
RU (1) | RU2252939C2 (fr) |
SI (1) | SI1228067T1 (fr) |
SK (1) | SK6432002A3 (fr) |
TR (1) | TR200402512T4 (fr) |
WO (1) | WO2001038325A1 (fr) |
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DE60237594D1 (de) * | 2001-04-25 | 2010-10-21 | Takeda Pharmaceutical | Verwendung des abc-expressionspromotors pioglitazon zur behandlung von arteriosklerose obliterans |
US20030092736A1 (en) * | 2001-05-30 | 2003-05-15 | Cheng Peter T. | Substituted azole acid derivatives useful as antidiabetic and antiobesity agents and method |
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JPWO2002098840A1 (ja) | 2001-06-04 | 2004-09-16 | エーザイ株式会社 | カルボン酸誘導体及びその塩もしくはそのエステルからなる医薬 |
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EP2253630A1 (fr) | 2007-05-21 | 2010-11-24 | Takeda Pharmaceutical Company Limited | Composé hétérocyclique et son utilisation |
TWI443090B (zh) * | 2007-05-25 | 2014-07-01 | Abbvie Deutschland | 作為代謝性麩胺酸受體2(mglu2 受體)之正向調節劑之雜環化合物 |
JP5432890B2 (ja) | 2008-04-04 | 2014-03-05 | 武田薬品工業株式会社 | 複素環誘導体及びその用途 |
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BR112013001634A2 (pt) | 2010-07-23 | 2016-05-24 | Takeda Pharmaceutical | composto ou sal, medicamento, métodos para a profilaxia ou tratamento da arteriosclerose, da diabete ou obesidade em um mamífero, e, uso do composto ou sal |
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EA201490152A1 (ru) | 2011-06-24 | 2014-05-30 | Эмджен Инк. | Антагонисты trpm8 и их применение при лечении |
WO2014007228A1 (fr) | 2012-07-03 | 2014-01-09 | 小野薬品工業株式会社 | Composé ayant une activité agoniste sur un récepteur de la somatostatine, et leur utilisation à des fins médicales |
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JP2015535227A (ja) * | 2012-10-26 | 2015-12-10 | エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト | Sykの3,4−二置換1h−ピラゾール及び4,5−二置換チアゾール阻害剤 |
KR20160062023A (ko) | 2013-09-30 | 2016-06-01 | 오노 야꾸힝 고교 가부시키가이샤 | 소마토스타틴 수용체 작동 활성을 갖는 화합물 및 그 의약 용도 |
EA032713B1 (ru) * | 2013-12-30 | 2019-07-31 | Лайфсай Фармасьютикалс, Инк. | Терапевтические ингибирующие соединения |
PT3210973T (pt) | 2014-10-24 | 2021-02-12 | Takeda Pharmaceuticals Co | Compostos de heteroarilo para o tratamento de doenças oftálmicas |
WO2016065326A2 (fr) | 2014-10-24 | 2016-04-28 | Bristol-Myers Squibb Company | Polypeptides fgf-21 modifiés et leurs utilisations |
CA3053091A1 (fr) | 2017-02-08 | 2018-08-16 | Ono Pharmaceutical Co., Ltd. | Compose ayant une activite agoniste du recepteur de la somatostatine et utilisation pharmaceutique associee |
KR102236356B1 (ko) | 2017-11-24 | 2021-04-05 | 주식회사 종근당 | 루푸스의 예방 또는 치료를 위한 조성물 |
KR20190099952A (ko) * | 2018-02-20 | 2019-08-28 | 주식회사 종근당 | 포도막염의 예방 또는 치료를 위한 조성물 |
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JPH06779B2 (ja) | 1985-06-10 | 1994-01-05 | 武田薬品工業株式会社 | チアゾリジオン誘導体およびそれを含んでなる医薬組成物 |
DE3600390A1 (de) | 1986-01-09 | 1987-07-16 | Hoechst Ag | Diarylalkyl-substituierte alkylamine, verfahren zu ihrer herstellung, ihre verwendung sowie sie enthaltende arzneimittel |
DE4206041A1 (de) * | 1992-02-27 | 1993-09-02 | Bayer Ag | Sulfonylbenzyl-substituierte imidazolylpropensaeurederivate |
US5591862A (en) * | 1993-06-11 | 1997-01-07 | Takeda Chemical Industries, Ltd. | Tetrazole derivatives, their production and use |
FR2707641B1 (fr) * | 1993-07-16 | 1995-08-25 | Fournier Ind & Sante | Composés de l'imidazol-5-carboxamide, leur procédé de préparation leurs intermédiaires et leur utilisation en thérapeutique. |
DE19602505A1 (de) | 1996-01-25 | 1997-07-31 | Merck Patent Gmbh | 1-(Pyrazol-4-Indol-3-yl)-Piperidine |
JPH1072434A (ja) | 1996-04-08 | 1998-03-17 | Nissan Chem Ind Ltd | 2,4−置換アニリン誘導体 |
AU742641B2 (en) | 1998-01-28 | 2002-01-10 | Shionogi & Co., Ltd. | Novel tricyclic compound |
EP1428531A1 (fr) | 1998-05-11 | 2004-06-16 | Takeda Chemical Industries, Ltd. | Dérivés d'acide oximinoalcanoique à activité hypoglycémique et hypolipidémique |
US6548529B1 (en) | 1999-04-05 | 2003-04-15 | Bristol-Myers Squibb Company | Heterocyclic containing biphenyl aP2 inhibitors and method |
-
2000
- 2000-11-09 AU AU13031/01A patent/AU780948C/en not_active Ceased
- 2000-11-09 ES ES00974857T patent/ES2225252T3/es not_active Expired - Lifetime
- 2000-11-09 CO CO00085306A patent/CO5261501A1/es not_active Application Discontinuation
- 2000-11-09 PT PT00974857T patent/PT1228067E/pt unknown
- 2000-11-09 CZ CZ20021604A patent/CZ20021604A3/cs unknown
- 2000-11-09 AR ARP000105914A patent/AR026414A1/es not_active Application Discontinuation
- 2000-11-09 KR KR10-2002-7006055A patent/KR100518142B1/ko not_active IP Right Cessation
- 2000-11-09 PE PE2000001199A patent/PE20011021A1/es not_active Application Discontinuation
- 2000-11-09 CA CA002390923A patent/CA2390923A1/fr not_active Abandoned
- 2000-11-09 WO PCT/JP2000/007877 patent/WO2001038325A1/fr active IP Right Grant
- 2000-11-09 NZ NZ519238A patent/NZ519238A/en unknown
- 2000-11-09 EP EP00974857A patent/EP1228067B1/fr not_active Expired - Lifetime
- 2000-11-09 MY MYPI20005273A patent/MY141468A/en unknown
- 2000-11-09 BR BR0015466-0A patent/BR0015466A/pt not_active IP Right Cessation
- 2000-11-09 JP JP2000347462A patent/JP3723071B2/ja not_active Expired - Fee Related
- 2000-11-09 SI SI200030494T patent/SI1228067T1/xx unknown
- 2000-11-09 MX MXPA02004647A patent/MXPA02004647A/es active IP Right Grant
- 2000-11-09 RU RU2002115263/04A patent/RU2252939C2/ru not_active IP Right Cessation
- 2000-11-09 TR TR2004/02512T patent/TR200402512T4/xx unknown
- 2000-11-09 EP EP04076508A patent/EP1457490A1/fr not_active Withdrawn
- 2000-11-09 SK SK643-2002A patent/SK6432002A3/sk unknown
- 2000-11-09 CN CNB008174679A patent/CN1260227C/zh not_active Expired - Fee Related
- 2000-11-09 AT AT00974857T patent/ATE271049T1/de not_active IP Right Cessation
- 2000-11-09 IL IL14949300A patent/IL149493A0/xx unknown
- 2000-11-09 DE DE60012213T patent/DE60012213T2/de not_active Expired - Lifetime
- 2000-11-09 PL PL00356487A patent/PL356487A1/xx not_active Application Discontinuation
- 2000-11-09 DK DK00974857T patent/DK1228067T3/da active
- 2000-11-09 US US10/129,702 patent/US7179823B1/en not_active Expired - Lifetime
- 2000-11-09 HU HU0203165A patent/HUP0203165A3/hu unknown
-
2002
- 2002-05-02 NO NO20022108A patent/NO20022108L/no unknown
- 2002-08-27 HK HK02106297.5A patent/HK1045991B/zh not_active IP Right Cessation
- 2002-10-29 JP JP2002315096A patent/JP4416994B2/ja not_active Expired - Fee Related
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