BR112013001634A2 - composto ou sal, medicamento, métodos para a profilaxia ou tratamento da arteriosclerose, da diabete ou obesidade em um mamífero, e, uso do composto ou sal - Google Patents

composto ou sal, medicamento, métodos para a profilaxia ou tratamento da arteriosclerose, da diabete ou obesidade em um mamífero, e, uso do composto ou sal

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Publication number
BR112013001634A2
BR112013001634A2 BR112013001634A BR112013001634A BR112013001634A2 BR 112013001634 A2 BR112013001634 A2 BR 112013001634A2 BR 112013001634 A BR112013001634 A BR 112013001634A BR 112013001634 A BR112013001634 A BR 112013001634A BR 112013001634 A2 BR112013001634 A2 BR 112013001634A2
Authority
BR
Brazil
Prior art keywords
compound
salt
prophylaxis
atherosclerosis
obesity
Prior art date
Application number
BR112013001634A
Other languages
English (en)
Inventor
Hideo Suzuki
Hidesaku Tokuhara
Kouhel Asano
Nobuyugi Matsunaga
Rei Okamoto
Takeshi Yamamoto
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of BR112013001634A2 publication Critical patent/BR112013001634A2/pt

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    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
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Abstract

composto ou sal, medicamento, métodos para a profilaxia ou tratamento da arteriosclerose, da diabete ou obesidade em um mamífero, e, uso do composto ou sal. é divulgado um composto que tem excelente atividade farmacológica, qualidades fisico-químicas e outras e é útil na prevenção/tratamento de condições relacionadas com eicosanoide incluindo arteriosclerose, osteoartrite e dermatite atópica. o composto é composto representado pela fórmula mencionada abaixo (cada símbolo na fórmula é como descrito no relatório descritivo) ou um sal deste.
BR112013001634A 2010-07-23 2011-07-22 composto ou sal, medicamento, métodos para a profilaxia ou tratamento da arteriosclerose, da diabete ou obesidade em um mamífero, e, uso do composto ou sal BR112013001634A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2010166475 2010-07-23
JP2011122796 2011-05-31
PCT/JP2011/066766 WO2012011591A1 (ja) 2010-07-23 2011-07-22 縮合複素環化合物およびその用途

Publications (1)

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BR112013001634A2 true BR112013001634A2 (pt) 2016-05-24

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BR112013001634A BR112013001634A2 (pt) 2010-07-23 2011-07-22 composto ou sal, medicamento, métodos para a profilaxia ou tratamento da arteriosclerose, da diabete ou obesidade em um mamífero, e, uso do composto ou sal

Country Status (8)

Country Link
US (1) US9023858B2 (pt)
EP (1) EP2597095A4 (pt)
JP (1) JPWO2012011591A1 (pt)
CN (1) CN103119043A (pt)
BR (1) BR112013001634A2 (pt)
CA (1) CA2806258A1 (pt)
EA (1) EA026142B1 (pt)
WO (1) WO2012011591A1 (pt)

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WO2017003723A1 (en) * 2015-07-01 2017-01-05 Crinetics Pharmaceuticals, Inc. Somatostatin modulators and uses thereof
EP3375783A4 (en) * 2015-11-11 2019-03-20 Sumitomo Chemical Company, Limited CONDENSED HETEROCYCLIC COMPOUND
US11028068B2 (en) 2017-07-25 2021-06-08 Crinetics Pharmaceuticals, Inc. Somatostatin modulators and uses thereof
US10639313B2 (en) 2017-09-01 2020-05-05 Ndsu Research Foundation Compound for inhibition of delta-5-desaturase (D5D) and treatment of cancer and inflammation
WO2019217591A1 (en) * 2018-05-09 2019-11-14 Regeneron Pharmaceuticals, Inc. Anti-msr1 antibodies and methods of use thereof

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US9023858B2 (en) 2015-05-05
CA2806258A1 (en) 2012-01-26
EP2597095A4 (en) 2014-10-01
EP2597095A1 (en) 2013-05-29
CN103119043A (zh) 2013-05-22
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EA026142B1 (ru) 2017-03-31
WO2012011591A1 (ja) 2012-01-26

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