BR112013001634A2 - composto ou sal, medicamento, métodos para a profilaxia ou tratamento da arteriosclerose, da diabete ou obesidade em um mamífero, e, uso do composto ou sal - Google Patents
composto ou sal, medicamento, métodos para a profilaxia ou tratamento da arteriosclerose, da diabete ou obesidade em um mamífero, e, uso do composto ou salInfo
- Publication number
- BR112013001634A2 BR112013001634A2 BR112013001634A BR112013001634A BR112013001634A2 BR 112013001634 A2 BR112013001634 A2 BR 112013001634A2 BR 112013001634 A BR112013001634 A BR 112013001634A BR 112013001634 A BR112013001634 A BR 112013001634A BR 112013001634 A2 BR112013001634 A2 BR 112013001634A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- salt
- prophylaxis
- atherosclerosis
- obesity
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- Health & Medical Sciences (AREA)
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Abstract
composto ou sal, medicamento, métodos para a profilaxia ou tratamento da arteriosclerose, da diabete ou obesidade em um mamífero, e, uso do composto ou sal. é divulgado um composto que tem excelente atividade farmacológica, qualidades fisico-químicas e outras e é útil na prevenção/tratamento de condições relacionadas com eicosanoide incluindo arteriosclerose, osteoartrite e dermatite atópica. o composto é composto representado pela fórmula mencionada abaixo (cada símbolo na fórmula é como descrito no relatório descritivo) ou um sal deste.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
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JP2010166475 | 2010-07-23 | ||
JP2011122796 | 2011-05-31 | ||
PCT/JP2011/066766 WO2012011591A1 (ja) | 2010-07-23 | 2011-07-22 | 縮合複素環化合物およびその用途 |
Publications (1)
Publication Number | Publication Date |
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BR112013001634A2 true BR112013001634A2 (pt) | 2016-05-24 |
Family
ID=45497008
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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BR112013001634A BR112013001634A2 (pt) | 2010-07-23 | 2011-07-22 | composto ou sal, medicamento, métodos para a profilaxia ou tratamento da arteriosclerose, da diabete ou obesidade em um mamífero, e, uso do composto ou sal |
Country Status (8)
Country | Link |
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US (1) | US9023858B2 (pt) |
EP (1) | EP2597095A4 (pt) |
JP (1) | JPWO2012011591A1 (pt) |
CN (1) | CN103119043A (pt) |
BR (1) | BR112013001634A2 (pt) |
CA (1) | CA2806258A1 (pt) |
EA (1) | EA026142B1 (pt) |
WO (1) | WO2012011591A1 (pt) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US11446241B2 (en) | 2013-07-29 | 2022-09-20 | Attillaps Holdings Inc. | Treatment of ophthalmological conditions with acetylcholinesterase inhibitors |
EP3157534B1 (en) | 2014-06-19 | 2022-07-06 | Attillaps Holdings | Acetylcholinesterase inhibitors for treatment of dermatological conditions |
WO2017003723A1 (en) * | 2015-07-01 | 2017-01-05 | Crinetics Pharmaceuticals, Inc. | Somatostatin modulators and uses thereof |
EP3375783A4 (en) * | 2015-11-11 | 2019-03-20 | Sumitomo Chemical Company, Limited | CONDENSED HETEROCYCLIC COMPOUND |
US11028068B2 (en) | 2017-07-25 | 2021-06-08 | Crinetics Pharmaceuticals, Inc. | Somatostatin modulators and uses thereof |
US10639313B2 (en) | 2017-09-01 | 2020-05-05 | Ndsu Research Foundation | Compound for inhibition of delta-5-desaturase (D5D) and treatment of cancer and inflammation |
WO2019217591A1 (en) * | 2018-05-09 | 2019-11-14 | Regeneron Pharmaceuticals, Inc. | Anti-msr1 antibodies and methods of use thereof |
Family Cites Families (37)
Publication number | Priority date | Publication date | Assignee | Title |
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JP2000501086A (ja) | 1995-11-24 | 2000-02-02 | ビイク グルデン ロンベルク ヒエーミツシエ フアブリーク ゲゼルシヤフト ミツト ベシユレンクテル ハフツング | ピリドピリミジン |
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AR035016A1 (es) | 1999-08-25 | 2004-04-14 | Takeda Chemical Industries Ltd | Composicion de azol promotor de produccion/secrecion de neurotrofina, compuesto prodroga del mismo, composicion farmaceutica que lo comprende y uso del mismo para preparar esta ultima. |
WO2001025228A1 (fr) | 1999-10-07 | 2001-04-12 | Tadeka Chemical Industries, Ltd. | Derives d'amines |
AR026414A1 (es) | 1999-11-10 | 2003-02-12 | Takeda Pharmaceutical | Compuetos heterociclicos de 5 miembros que contienen nitrogeno |
KR100866820B1 (ko) | 2000-07-13 | 2008-11-04 | 다케다 야쿠힌 고교 가부시키가이샤 | 지질 풍부 플라크 퇴축제 |
CA2416384A1 (en) | 2000-07-17 | 2003-01-16 | Takeda Chemical Industries, Ltd. | Sulfone derivatives, their production and use |
WO2003042204A1 (fr) | 2001-10-19 | 2003-05-22 | Takeda Chemical Industries, Ltd. | Derive d'amine |
WO2003059900A1 (fr) | 2002-01-11 | 2003-07-24 | Takeda Chemical Industries, Ltd. | Derives de coumarine, leur procede de production et d'utilisation |
WO2003106435A1 (en) | 2002-06-18 | 2003-12-24 | Sankyo Company, Limited | Fused-ring pyrimidin-4(3h)-one derivatives, processes for the preparation and uses thereof |
CA2507026A1 (en) | 2002-11-22 | 2004-06-10 | Takeda Pharmaceutical Company Limited | Imidazole derivatives, their production and use |
EP1669352A4 (en) | 2003-09-30 | 2008-12-17 | Takeda Pharmaceutical | THIAZOLINE DERIVATIVE AND ITS USE |
JP4769082B2 (ja) | 2003-12-17 | 2011-09-07 | 武田薬品工業株式会社 | ウレア誘導体、その製造法及び用途 |
CN1918128B (zh) | 2004-02-13 | 2011-01-26 | 万有制药株式会社 | 稠环4-氧代-嘧啶衍生物 |
WO2005091711A2 (en) | 2004-03-24 | 2005-10-06 | Orchid Chemicals & Pharmaceuticals Ltd | Novel condensed pyrimidones |
TWI396686B (zh) | 2004-05-21 | 2013-05-21 | Takeda Pharmaceutical | 環狀醯胺衍生物、以及其製品和用法 |
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DE602006015658D1 (de) | 2005-06-27 | 2010-09-02 | Amgen Inc | Entzündungshemmende arylnitrilverbindungen |
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WO2008089307A2 (en) * | 2007-01-18 | 2008-07-24 | Lexicon Pharmaceuticals, Inc. | Delta 5 desaturase inhibitors for the treatment of pain, inflammation and cancer |
US8922518B2 (en) | 2007-12-20 | 2014-12-30 | Samsung Electronics Co., Ltd. | Mobile terminal having touch screen and function controlling method of the same |
JP5212644B2 (ja) | 2009-01-19 | 2013-06-19 | 日本電気株式会社 | 移動通信ネットワークにおける通信設定方法及び移動通信端末 |
WO2010087467A1 (en) * | 2009-01-27 | 2010-08-05 | Takeda Pharmaceutical Company Limited | Delta-5-desaturase inhibitors |
JP5496631B2 (ja) | 2009-12-14 | 2014-05-21 | 三洋電機株式会社 | 断熱箱体 |
-
2011
- 2011-07-22 CN CN2011800453754A patent/CN103119043A/zh active Pending
- 2011-07-22 EP EP11809761.7A patent/EP2597095A4/en not_active Withdrawn
- 2011-07-22 JP JP2012525456A patent/JPWO2012011591A1/ja active Pending
- 2011-07-22 BR BR112013001634A patent/BR112013001634A2/pt not_active IP Right Cessation
- 2011-07-22 US US13/811,755 patent/US9023858B2/en not_active Expired - Fee Related
- 2011-07-22 CA CA2806258A patent/CA2806258A1/en not_active Abandoned
- 2011-07-22 EA EA201390158A patent/EA026142B1/ru not_active IP Right Cessation
- 2011-07-22 WO PCT/JP2011/066766 patent/WO2012011591A1/ja active Application Filing
Also Published As
Publication number | Publication date |
---|---|
US20130131050A1 (en) | 2013-05-23 |
EA201390158A1 (ru) | 2013-08-30 |
US9023858B2 (en) | 2015-05-05 |
CA2806258A1 (en) | 2012-01-26 |
EP2597095A4 (en) | 2014-10-01 |
EP2597095A1 (en) | 2013-05-29 |
CN103119043A (zh) | 2013-05-22 |
JPWO2012011591A1 (ja) | 2013-09-09 |
EA026142B1 (ru) | 2017-03-31 |
WO2012011591A1 (ja) | 2012-01-26 |
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