EA201390158A1 - Конденсированное гетероциклическое соединение и его применение - Google Patents

Конденсированное гетероциклическое соединение и его применение

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Publication number
EA201390158A1
EA201390158A1 EA201390158A EA201390158A EA201390158A1 EA 201390158 A1 EA201390158 A1 EA 201390158A1 EA 201390158 A EA201390158 A EA 201390158A EA 201390158 A EA201390158 A EA 201390158A EA 201390158 A1 EA201390158 A1 EA 201390158A1
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EA
Eurasian Patent Office
Prior art keywords
application
heterocyclic compound
condensed heterocyclic
atherosclerosis
relates
Prior art date
Application number
EA201390158A
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English (en)
Other versions
EA026142B1 (ru
Inventor
Нобуюки Мацунага
Хидео Сузуки
Коухей Асано
Хидеказу Токухара
Такеси Ямамото
Реи Окамото
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Такеда Фармасьютикал Компани Лимитед
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Application filed by Такеда Фармасьютикал Компани Лимитед filed Critical Такеда Фармасьютикал Компани Лимитед
Publication of EA201390158A1 publication Critical patent/EA201390158A1/ru
Publication of EA026142B1 publication Critical patent/EA026142B1/ru

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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Abstract

Настоящее изобретение относится к соединению, используемому для профилактики или лечения связанных с эйкозаноидами заболеваний, таких как атеросклероз, атеротромбоз, сахарный диабет, ожирение, астма, лихорадка, боль, рак, ревматизм, остеоартрит, атопический дерматит и тому подобные, и оказывающему более выраженное фармакологическое действие, имеющему более благоприятные физико-химические свойства и тому подобные. Настоящее изобретение относится к соединению, представленному следующей формулойгде каждый символ определен в описании, или к его соли.
EA201390158A 2010-07-23 2011-07-22 Конденсированное гетероциклическое соединение и его применение EA026142B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2010166475 2010-07-23
JP2011122796 2011-05-31
PCT/JP2011/066766 WO2012011591A1 (ja) 2010-07-23 2011-07-22 縮合複素環化合物およびその用途

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EA201390158A1 true EA201390158A1 (ru) 2013-08-30
EA026142B1 EA026142B1 (ru) 2017-03-31

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US (1) US9023858B2 (ru)
EP (1) EP2597095A4 (ru)
JP (1) JPWO2012011591A1 (ru)
CN (1) CN103119043A (ru)
BR (1) BR112013001634A2 (ru)
CA (1) CA2806258A1 (ru)
EA (1) EA026142B1 (ru)
WO (1) WO2012011591A1 (ru)

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RU2781636C2 (ru) * 2016-01-27 2022-10-17 Университет Цюрих Применение модуляторов gabaa-рецептора для лечения зуда

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US11446241B2 (en) 2013-07-29 2022-09-20 Attillaps Holdings Inc. Treatment of ophthalmological conditions with acetylcholinesterase inhibitors
HRP20220854T1 (hr) 2014-06-19 2022-10-14 Attillaps Holdings Inhibitori acetilkolinesteraze za liječenje dermatoloških stanja
WO2017003723A1 (en) * 2015-07-01 2017-01-05 Crinetics Pharmaceuticals, Inc. Somatostatin modulators and uses thereof
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