DE69616956T2 - 3-Amino-2-mercaptobenzoesäure-Derivate und Verfahren zu ihrer Herstellung - Google Patents

3-Amino-2-mercaptobenzoesäure-Derivate und Verfahren zu ihrer Herstellung

Info

Publication number
DE69616956T2
DE69616956T2 DE69616956T DE69616956T DE69616956T2 DE 69616956 T2 DE69616956 T2 DE 69616956T2 DE 69616956 T DE69616956 T DE 69616956T DE 69616956 T DE69616956 T DE 69616956T DE 69616956 T2 DE69616956 T2 DE 69616956T2
Authority
DE
Germany
Prior art keywords
substituted
unsubstituted
compounds
preparation
carbon atoms
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69616956T
Other languages
English (en)
Other versions
DE69616956D1 (de
DE69616956T3 (de
Inventor
Walter Kunz
Beat Jau
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Syngenta Participations AG
Original Assignee
Syngenta Participations AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations AG filed Critical Syngenta Participations AG
Publication of DE69616956D1 publication Critical patent/DE69616956D1/de
Publication of DE69616956T2 publication Critical patent/DE69616956T2/de
Application granted granted Critical
Publication of DE69616956T3 publication Critical patent/DE69616956T3/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/14—Thiadiazoles; Hydrogenated thiadiazoles condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/02—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of thiols
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/02—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of thiols
    • C07C319/12—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of thiols by reactions not involving the formation of mercapto groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/62—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
    • C07C323/63—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C327/00—Thiocarboxylic acids
    • C07C327/20—Esters of monothiocarboxylic acids
    • C07C327/26—Esters of monothiocarboxylic acids having carbon atoms of esterified thiocarboxyl groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C335/04—Derivatives of thiourea
    • C07C335/16—Derivatives of thiourea having nitrogen atoms of thiourea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C335/22—Derivatives of thiourea having nitrogen atoms of thiourea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D277/82—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DE69616956.8T 1995-12-21 1996-12-12 3-Amino-2-mercaptobenzoesäure-Derivate und Verfahren zu ihrer Herstellung Expired - Lifetime DE69616956T3 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH363795 1995-12-21
CH363795 1995-12-21
EP96810865.4A EP0780372B3 (de) 1995-12-21 1996-12-12 3-Amino-2-mercaptobenzoesäure-Derivate und Verfahren zu ihrer Herstellung
US08/770,353 US5770758A (en) 1995-12-21 1996-12-20 3-amino-2-mercaptobenzoic acid derivatives and processes for their preparation

Publications (3)

Publication Number Publication Date
DE69616956D1 DE69616956D1 (de) 2001-12-20
DE69616956T2 true DE69616956T2 (de) 2002-06-20
DE69616956T3 DE69616956T3 (de) 2014-01-30

Family

ID=25693502

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69616956.8T Expired - Lifetime DE69616956T3 (de) 1995-12-21 1996-12-12 3-Amino-2-mercaptobenzoesäure-Derivate und Verfahren zu ihrer Herstellung

Country Status (21)

Country Link
US (1) US5770758A (de)
EP (1) EP0780372B3 (de)
JP (1) JP4217924B2 (de)
KR (1) KR100470887B1 (de)
CN (2) CN1078888C (de)
AT (1) ATE208760T1 (de)
AU (1) AU713526B2 (de)
BR (1) BR9606092A (de)
CA (1) CA2193460C (de)
CZ (1) CZ291857B6 (de)
DE (1) DE69616956T3 (de)
DK (1) DK0780372T3 (de)
ES (1) ES2168121T7 (de)
HU (1) HU221600B (de)
IL (3) IL133900A (de)
MX (2) MX9606665A (de)
PL (1) PL187885B1 (de)
PT (1) PT780372E (de)
RU (1) RU2176241C2 (de)
SK (1) SK283840B6 (de)
ZA (1) ZA9610774B (de)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10313887A1 (de) * 2003-03-27 2004-10-28 Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. Verfahren zum selektiven Gewinnen von Gold aus goldhaltigen Materialien

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6002013A (en) * 1995-12-21 1999-12-14 Novartis Corporation 3-amino-2-mercaptobenzoic acid derivatives and processes for their preparation
GB9724586D0 (en) * 1997-11-20 1998-01-21 Rhone Poulenc Agriculture New herbicides
ES2405594T3 (es) 2002-09-25 2013-05-31 Memory Pharmaceuticals Corporation Idazoles, benzotiazoles y benzisotiazoles, y preparación y usos de los mismos
DK2368553T3 (en) 2003-04-08 2015-02-09 Progenics Pharm Inc Pharmaceutical preparation comprising methylnaltrexone
WO2005007601A2 (en) * 2003-07-10 2005-01-27 Achillion Pharmaceuticals, Inc. Substituted arylthiourea derivatives useful as inhibitors of viral replication
BRPI0508771A (pt) 2004-03-25 2007-08-14 Memory Pharm Corp indazóis, benzotiazóis, benzoisotiazóis, benzisoxazóis, e a preparação e usos dos mesmos
AR057325A1 (es) 2005-05-25 2007-11-28 Progenics Pharm Inc Sintesis de (s)-n-metilnaltrexona, composiciones farmaceuticas y usos
AR057035A1 (es) 2005-05-25 2007-11-14 Progenics Pharm Inc SíNTESIS DE (R)-N-METILNALTREXONA, COMPOSICIONES FARMACÉUTICAS Y USOS
CN101395161A (zh) 2006-03-02 2009-03-25 马林克罗特公司 噻二唑化合物及其在光疗中的用途
PT2565195E (pt) 2007-03-29 2015-07-28 Wyeth Llc Antagonistas e receptor opióide periférico e respectivas utilizações
ES2765811T5 (es) 2007-03-29 2024-02-27 Progenics Pharm Inc Forma cristalina de bromuro de (R)-n-metilnaltrexona y sus usos
EP3064503A1 (de) 2007-03-29 2016-09-07 Progenics Pharmaceuticals, Inc. Antagonisten der peripheren opioidrezeptoren und ihre verwendung
EP2240489A1 (de) 2008-02-06 2010-10-20 Progenics Pharmaceuticals, Inc. HERSTELLUNG UND VERWENDUNG VON (R), (R)-2,2ýBIS-METHYLNALTREXON
CA2676881C (en) 2008-09-30 2017-04-25 Wyeth Peripheral opioid receptor antagonists and uses thereof
CN101492429B (zh) * 2008-12-10 2010-12-15 上海泰禾(集团)有限公司 一种苯并-[1，2，3]-噻二唑-7-甲酸三氟乙酯的提纯方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4150140A (en) * 1976-12-23 1979-04-17 The Upjohn Company Benzothiazolyl oxanic acids, esters and salts
DE2757924A1 (de) * 1977-12-24 1979-07-05 Hoechst Ag Verfahren zur herstellung von vinylchlorid-polymerisaten
DE3601286A1 (de) * 1986-01-17 1987-07-23 Consiglio Nazionale Ricerche Sammelmittel fuer die selektive flotation von blei- und zinkerzen und verfahren zu deren herstellung
ATE82668T1 (de) 1987-08-21 1992-12-15 Ciba Geigy Ag Benzothiadiazole und ihre verwendung in verfahren und mitteln gegen pflanzenkrankheiten.
EP0384889B1 (de) * 1989-02-21 1993-10-13 Ciba-Geigy Ag Mittel zum Schutz von Pflanzen gegen Krankheiten
EP0529600B1 (de) 1991-08-30 1996-11-06 Hoechst Aktiengesellschaft Verfahren zur Herstellung von 2-Aminobenzthiazolen
JPH0690518A (ja) * 1992-09-09 1994-03-29 Toshiba Corp 地絡継電器
JP3310104B2 (ja) * 1994-04-04 2002-07-29 三新化学工業株式会社 ２−アミノチオフェノール類の製造方法
MX9702787A (es) * 1994-10-17 1997-06-28 Novartis Ag Proceso para la preparacion de 3-aminobenzonitrilos sustituidos.

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10313887A1 (de) * 2003-03-27 2004-10-28 Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. Verfahren zum selektiven Gewinnen von Gold aus goldhaltigen Materialien

Also Published As

Publication number Publication date
EP0780372A2 (de) 1997-06-25
PT780372E (pt) 2002-04-29
CZ377396A3 (en) 1997-07-16
AU713526C (en) 1997-06-26
MXPA02000515A (es) 2002-09-17
HU221600B (hu) 2002-11-28
JP4217924B2 (ja) 2009-02-04
AU713526B2 (en) 1999-12-02
US5770758A (en) 1998-06-23
PL317601A1 (en) 1997-06-23
IL119819A0 (en) 1997-03-18
CN1163491C (zh) 2004-08-25
HUP9603527A2 (en) 1997-09-29
JPH09235279A (ja) 1997-09-09
IL133900A0 (en) 2001-04-30
ES2168121T7 (es) 2013-09-24
EP0780372B1 (de) 2001-11-14
HU9603527D0 (en) 1997-02-28
BR9606092A (pt) 1998-09-01
IL133900A (en) 2004-07-25
IL119819A (en) 2004-07-25
CA2193460A1 (en) 1997-06-22
ATE208760T1 (de) 2001-11-15
CN1156722A (zh) 1997-08-13
CN1078888C (zh) 2002-02-06
EP0780372B3 (de) 2013-05-22
CA2193460C (en) 2007-03-27
DK0780372T3 (da) 2002-03-11
CN1392144A (zh) 2003-01-22
HUP9603527A3 (en) 1999-04-28
DE69616956D1 (de) 2001-12-20
MX9606665A (es) 1997-06-28
ZA9610774B (en) 1997-06-30
SK283840B6 (sk) 2004-03-02
DE69616956T3 (de) 2014-01-30
ES2168121T3 (es) 2002-06-01
KR100470887B1 (ko) 2005-03-14
RU2176241C2 (ru) 2001-11-27
SK163696A3 (en) 1997-10-08
EP0780372A3 (de) 1997-09-17
PL187885B1 (pl) 2004-10-29
AU7640496A (en) 1997-06-26
CZ291857B6 (cs) 2003-06-18

Similar Documents

Publication Publication Date Title
DE69616956T2 (de) 3-Amino-2-mercaptobenzoesäure-Derivate und Verfahren zu ihrer Herstellung
ATE115952T1 (de) Pyrimidindion-derivate, verfahren zu deren herstellung und diese enthaltende antiarrythmische mittel.
HU9401943D0 (en) Process for producing amide and urea derivatives and compositions containing them
ATE170521T1 (de) 1-methyl-carbapenemderivate, deren herstellung und verwendung als antibiotika
PT85293A (de) Loesungen von oxazaphosphorinen mit verbesserter stabilitaet und verfahren zu deren herstellung
NZ226222A (en) Preparation of n-alkylated alpha-aminodiacids and esters thereof, and use of those compounds in the synthesis of n-heterocyclic dipeptides
MX170732B (es) Composicion de derivados de succinimida y su uso
GR3019711T3 (en) Spiro-indoline-oxazine compounds with photochromatic and photosensitizing characteristics and the process for their preparation
DE3886185T2 (de) 2-Thiazolidinon-Derivate und diese enthaltende pharmazeutische Präparate, Verfahren zu deren Herstellung und deren Verwendung.
DE3686876T2 (de) 4-morpholinyl 1h-indol-derivate, ihre salze, verfahren und zwischenprodukte zur herstellung, verwendung als arzneimittel, sie enthaltende zusammensetzungen.
ATE111904T1 (de) Cyclische aminothioacetalamide, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen.
DE3884518T2 (de) Naphthothiazepin-Derivate und Verfahren zu ihrer Herstellung.
ATE100817T1 (de) Herstellung von optisch aktiven 2-oxoimidazolidin-derivaten.
AR004403A1 (es) Derivados de acido 3-amino-2-mercaptobenzoico, procesos para su preparacion y compuestos intermediarios para su exclusivo uso en los procedimientos correspondientes y procedimiento para preparar los compuestos intermediarios

Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8328 Change in the person/name/address of the agent

Representative=s name: PFENNING MEINIG & PARTNER GBR, 80339 MUENCHEN

8328 Change in the person/name/address of the agent

Representative=s name: MAIWALD PATENTANWALTSGESELLSCHAFT MBH, 80335 MUENC