DD202428A5 - Verfahren zur herstellung von prostaglandinsaeurederivaten - Google Patents

Verfahren zur herstellung von prostaglandinsaeurederivaten Download PDF

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Publication number
DD202428A5
DD202428A5 DD81232562A DD23256281A DD202428A5 DD 202428 A5 DD202428 A5 DD 202428A5 DD 81232562 A DD81232562 A DD 81232562A DD 23256281 A DD23256281 A DD 23256281A DD 202428 A5 DD202428 A5 DD 202428A5
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DD
German Democratic Republic
Prior art keywords
hydrogen
derivatives
group
general formula
compound
Prior art date
Application number
DD81232562A
Other languages
German (de)
English (en)
Inventor
Stephan Gero
Jean-Claude Barriere
Jeanine Cleophax
Andre Cier
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of DD202428A5 publication Critical patent/DD202428A5/de

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • C07C405/0008Analogues having the carboxyl group in the side-chains replaced by other functional groups
    • C07C405/0033Analogues having the carboxyl group in the side-chains replaced by other functional groups containing sulfur
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C43/00Ethers; Compounds having groups, groups or groups
    • C07C43/02Ethers
    • C07C43/18Ethers having an ether-oxygen atom bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C43/196Ethers having an ether-oxygen atom bound to a carbon atom of a ring other than a six-membered aromatic ring containing hydroxy or O-metal groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/27Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation
    • C07C45/29Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/56Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds
    • C07C45/57Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom
    • C07C45/60Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom in six-membered rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/65Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by splitting-off hydrogen atoms or functional groups; by hydrogenolysis of functional groups
    • C07C45/66Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by splitting-off hydrogen atoms or functional groups; by hydrogenolysis of functional groups by dehydration
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C47/00Compounds having —CHO groups
    • C07C47/38Unsaturated compounds having —CHO groups bound to carbon atoms of rings other than six—membered aromatic rings
    • C07C47/47Unsaturated compounds having —CHO groups bound to carbon atoms of rings other than six—membered aromatic rings containing ether groups, groups, groups, or groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D319/00Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/041,3-Dioxanes; Hydrogenated 1,3-dioxanes
    • C07D319/061,3-Dioxanes; Hydrogenated 1,3-dioxanes not condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D339/00Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
    • C07D339/02Five-membered rings
    • C07D339/06Five-membered rings having the hetero atoms in positions 1 and 3, e.g. cyclic dithiocarbonates
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/10Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/06Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/10Systems containing only non-condensed rings with a five-membered ring the ring being unsaturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Steroid Compounds (AREA)
DD81232562A 1980-08-12 1981-08-12 Verfahren zur herstellung von prostaglandinsaeurederivaten DD202428A5 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8026240 1980-08-12
GB8113487 1981-05-01

Publications (1)

Publication Number Publication Date
DD202428A5 true DD202428A5 (de) 1983-09-14

Family

ID=26276527

Family Applications (3)

Application Number Title Priority Date Filing Date
DD81232562A DD202428A5 (de) 1980-08-12 1981-08-12 Verfahren zur herstellung von prostaglandinsaeurederivaten
DD81250873A DD213437A5 (de) 1980-08-12 1981-08-12 Verfahren zur herstellung von cyclopentenderivaten
DD83263174A DD223712A5 (de) 1980-08-12 1983-05-12 Verfahren zur herstellung von cyclopentenderivaten

Family Applications After (2)

Application Number Title Priority Date Filing Date
DD81250873A DD213437A5 (de) 1980-08-12 1981-08-12 Verfahren zur herstellung von cyclopentenderivaten
DD83263174A DD223712A5 (de) 1980-08-12 1983-05-12 Verfahren zur herstellung von cyclopentenderivaten

Country Status (27)

Country Link
US (1) US4377704A (sv)
AU (2) AU542975B2 (sv)
BG (1) BG36345A3 (sv)
CH (2) CH650251A5 (sv)
DD (3) DD202428A5 (sv)
DE (1) DE3131616A1 (sv)
DK (1) DK356481A (sv)
ES (2) ES8301465A1 (sv)
FI (1) FI812468L (sv)
FR (2) FR2488604A1 (sv)
GR (1) GR74314B (sv)
HU (1) HU191416B (sv)
IL (1) IL63369A (sv)
IS (1) IS1184B6 (sv)
IT (1) IT1214436B (sv)
LU (1) LU83547A1 (sv)
NL (1) NL8103710A (sv)
NO (1) NO812720L (sv)
NZ (1) NZ197729A (sv)
OA (1) OA06879A (sv)
PL (2) PL133879B1 (sv)
PT (1) PT73457B (sv)
RO (2) RO82680B (sv)
SE (2) SE442297B (sv)
SU (1) SU1187716A3 (sv)
YU (2) YU193781A (sv)
ZW (1) ZW17881A1 (sv)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8510277D0 (en) * 1985-04-23 1985-05-30 Glaxo Group Ltd Carbocyclic compounds
AU635065B2 (en) * 1989-09-08 1993-03-11 Emmanouilidis, Theo Mountable washing device
US6711436B1 (en) 1997-08-08 2004-03-23 Duke University Compositions, apparatus and methods for facilitating surgical procedures
AU758370B2 (en) * 1997-08-08 2003-03-20 Duke University Compositions, apparatus and methods for facilitating surgical procedures

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3664502A (en) * 1970-06-26 1972-05-23 Bird Machine Co Slurry screen and process of making it
US4229592A (en) * 1978-02-06 1980-10-21 Kansas University Endowment Association Intermediate for prostaglandins and process for preparing the intermediate
SE7906017L (sv) * 1978-07-11 1980-02-13 Glaxo Group Ltd Prostanoida foreningar

Also Published As

Publication number Publication date
AU3406784A (en) 1985-01-31
FR2488604A1 (fr) 1982-02-19
RO87011A (ro) 1985-05-20
OA06879A (fr) 1983-02-28
YU86183A (en) 1984-04-30
NO812720L (no) 1982-02-15
DE3131616A1 (de) 1982-04-22
ZW17881A1 (en) 1981-10-14
FR2509306A1 (fr) 1983-01-14
PT73457B (en) 1982-10-15
AU542975B2 (en) 1985-03-28
IL63369A (en) 1985-11-29
LU83547A1 (fr) 1981-12-01
IT8123455A0 (it) 1981-08-10
DD223712A5 (de) 1985-06-19
SU1187716A3 (ru) 1985-10-23
SE8104703L (sv) 1982-02-13
AU7400781A (en) 1982-03-04
NZ197729A (en) 1985-03-20
RO82680A (ro) 1984-05-12
HUT34147A (en) 1985-02-28
ES504681A0 (es) 1982-12-01
ES8301465A1 (es) 1982-12-01
FI812468L (fi) 1982-02-13
IT1214436B (it) 1990-01-18
SE8502007D0 (sv) 1985-04-25
PL137212B1 (en) 1986-05-31
RO82680B (ro) 1984-06-30
HU191416B (en) 1987-02-27
PL232567A1 (en) 1983-01-03
US4377704A (en) 1983-03-22
PT73457A (en) 1981-08-01
IS2661A7 (is) 1982-02-13
FR2509306B1 (sv) 1984-04-13
CH650251A5 (fr) 1985-07-15
YU193781A (en) 1984-02-29
DK356481A (da) 1982-02-13
BG36345A3 (en) 1984-10-15
NL8103710A (nl) 1982-03-01
GR74314B (sv) 1984-06-22
SE8502007L (sv) 1985-04-25
ES8305710A1 (es) 1983-04-16
IL63369A0 (en) 1981-10-30
IS1184B6 (is) 1985-05-13
ES514592A0 (es) 1983-04-16
PL133879B1 (en) 1985-07-31
CH655716A5 (fr) 1986-05-15
DD213437A5 (de) 1984-09-12
SE442297B (sv) 1985-12-16
FR2488604B1 (sv) 1984-11-09

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