CZ387492A3 - Analogs of non-aromatic hetero cycles containing nitrogen with a condensed ring, process of their preparation and use - Google Patents

Analogs of non-aromatic hetero cycles containing nitrogen with a condensed ring, process of their preparation and use Download PDF

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Publication number
CZ387492A3
CZ387492A3 CS923874A CS387492A CZ387492A3 CZ 387492 A3 CZ387492 A3 CZ 387492A3 CS 923874 A CS923874 A CS 923874A CS 387492 A CS387492 A CS 387492A CZ 387492 A3 CZ387492 A3 CZ 387492A3
Authority
CZ
Czechia
Prior art keywords
alkyl
group
compound
groups
phenyl
Prior art date
Application number
CS923874A
Other languages
Czech (cs)
English (en)
Inventor
Manoj C Desai
Harry R Howard
Terry J Rosen
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CZ387492A3 publication Critical patent/CZ387492A3/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Polyoxymethylene Polymers And Polymers With Carbon-To-Carbon Bonds (AREA)
  • Eye Examination Apparatus (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Electroluminescent Light Sources (AREA)
CS923874A 1990-09-28 1991-08-20 Analogs of non-aromatic hetero cycles containing nitrogen with a condensed ring, process of their preparation and use CZ387492A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US59042390A 1990-09-28 1990-09-28
PCT/US1991/005776 WO1992006079A1 (en) 1990-09-28 1991-08-20 Fused ring analogs of nitrogen containing nonaromatic heterocycles

Publications (1)

Publication Number Publication Date
CZ387492A3 true CZ387492A3 (en) 1994-02-16

Family

ID=24362216

Family Applications (1)

Application Number Title Priority Date Filing Date
CS923874A CZ387492A3 (en) 1990-09-28 1991-08-20 Analogs of non-aromatic hetero cycles containing nitrogen with a condensed ring, process of their preparation and use

Country Status (22)

Country Link
EP (1) EP0550635B1 (OSRAM)
JP (1) JPH0772175B2 (OSRAM)
CN (1) CN1060285A (OSRAM)
AT (1) ATE121389T1 (OSRAM)
AU (1) AU651145B2 (OSRAM)
BR (1) BR9106905A (OSRAM)
CA (1) CA2089736A1 (OSRAM)
CZ (1) CZ387492A3 (OSRAM)
DE (1) DE69109125T2 (OSRAM)
DK (1) DK0550635T3 (OSRAM)
ES (1) ES2071334T3 (OSRAM)
FI (1) FI931370A7 (OSRAM)
HU (1) HUT68667A (OSRAM)
IE (1) IE66042B1 (OSRAM)
IL (1) IL99525A0 (OSRAM)
MX (1) MX9101274A (OSRAM)
NO (1) NO931151D0 (OSRAM)
PT (1) PT99064A (OSRAM)
TW (1) TW199144B (OSRAM)
WO (1) WO1992006079A1 (OSRAM)
YU (1) YU159291A (OSRAM)
ZA (1) ZA917744B (OSRAM)

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DE69331190T2 (de) * 1992-05-18 2002-04-18 Pfizer Inc., New York Überbrückte azabicyclische derivate als substanz p antagonisten
US5637699A (en) * 1992-06-29 1997-06-10 Merck & Co., Inc. Process for preparing morpholine tachykinin receptor antagonists
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US5719147A (en) * 1992-06-29 1998-02-17 Merck & Co., Inc. Morpholine and thiomorpholine tachykinin receptor antagonists
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ATE194340T1 (de) * 1992-12-10 2000-07-15 Pfizer Aminomethylen substituierte heterocyclische verbindungen und ihre verwendung alssubstanz p antagonisten
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Also Published As

Publication number Publication date
TW199144B (OSRAM) 1993-02-01
AU651145B2 (en) 1994-07-14
IE913396A1 (en) 1992-04-08
EP0550635B1 (en) 1995-04-19
FI931370L (fi) 1993-03-26
HU9300898D0 (en) 1993-06-28
ATE121389T1 (de) 1995-05-15
JPH0772175B2 (ja) 1995-08-02
CN1060285A (zh) 1992-04-15
IE66042B1 (en) 1995-12-13
ES2071334T3 (es) 1995-06-16
IL99525A0 (en) 1992-08-18
NO931151L (no) 1993-03-26
HUT68667A (en) 1995-07-28
FI931370A0 (fi) 1993-03-26
BR9106905A (pt) 1993-08-17
PT99064A (pt) 1992-08-31
EP0550635A1 (en) 1993-07-14
NO931151D0 (no) 1993-03-26
DK0550635T3 (da) 1995-09-04
MX9101274A (es) 1992-05-04
AU8746391A (en) 1992-04-28
JPH06501267A (ja) 1994-02-10
DE69109125D1 (de) 1995-05-24
YU159291A (sh) 1994-01-20
DE69109125T2 (de) 1995-09-28
CA2089736A1 (en) 1992-03-29
WO1992006079A1 (en) 1992-04-16
ZA917744B (en) 1993-03-29
FI931370A7 (fi) 1993-03-26

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