CS248749B2 - Production method of the 6-(subst.)hydroxymethylpenicilan acids - Google Patents

Production method of the 6-(subst.)hydroxymethylpenicilan acids Download PDF

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Publication number
CS248749B2
CS248749B2 CS856935A CS693585A CS248749B2 CS 248749 B2 CS248749 B2 CS 248749B2 CS 856935 A CS856935 A CS 856935A CS 693585 A CS693585 A CS 693585A CS 248749 B2 CS248749 B2 CS 248749B2
Authority
CS
Czechoslovakia
Prior art keywords
group
hydrogen
formula
methyl
carbon atoms
Prior art date
Application number
CS856935A
Other languages
Czech (cs)
English (en)
Inventor
Yuphyng L Chen
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CS248749B2 publication Critical patent/CS248749B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CS856935A 1984-01-30 1985-01-29 Production method of the 6-(subst.)hydroxymethylpenicilan acids CS248749B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US57535484A 1984-01-30 1984-01-30

Publications (1)

Publication Number Publication Date
CS248749B2 true CS248749B2 (en) 1987-02-12

Family

ID=24299979

Family Applications (5)

Application Number Title Priority Date Filing Date
CS85619A CS248733B2 (en) 1984-01-30 1985-01-29 Production method of the 6-(subst.)methlenphenicilan acids
CS856932A CS248746B2 (en) 1984-01-30 1985-01-29 Production method of the 6-(subst.)methylenpenicilan acids
CS856934A CS248748B2 (en) 1984-01-30 1985-01-29 Production method of the 6-(subst.)methylenpenicilan acids
CS856935A CS248749B2 (en) 1984-01-30 1985-01-29 Production method of the 6-(subst.)hydroxymethylpenicilan acids
CS856933A CS248747B2 (en) 1984-01-30 1985-01-29 Production method of the 6-(subst.)hydroxymethylpenicilan acids

Family Applications Before (3)

Application Number Title Priority Date Filing Date
CS85619A CS248733B2 (en) 1984-01-30 1985-01-29 Production method of the 6-(subst.)methlenphenicilan acids
CS856932A CS248746B2 (en) 1984-01-30 1985-01-29 Production method of the 6-(subst.)methylenpenicilan acids
CS856934A CS248748B2 (en) 1984-01-30 1985-01-29 Production method of the 6-(subst.)methylenpenicilan acids

Family Applications After (1)

Application Number Title Priority Date Filing Date
CS856933A CS248747B2 (en) 1984-01-30 1985-01-29 Production method of the 6-(subst.)hydroxymethylpenicilan acids

Country Status (15)

Country Link
JP (1) JPS61109791A (xx)
KR (1) KR880001029B1 (xx)
CS (5) CS248733B2 (xx)
DD (3) DD247678A5 (xx)
EG (1) EG16904A (xx)
ES (5) ES8604972A1 (xx)
FI (1) FI85376C (xx)
HU (2) HU194891B (xx)
IL (1) IL74190A (xx)
NO (1) NO165594C (xx)
PL (5) PL145130B1 (xx)
PT (1) PT79893B (xx)
SU (4) SU1395144A3 (xx)
YU (5) YU44770B (xx)
ZA (1) ZA85682B (xx)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3869630D1 (de) * 1987-01-27 1992-05-07 Pfizer 6-beta(substituierte)-(s)-hydroxymethylpenicillansaeure und deren derivate.
US6156745A (en) 1997-12-29 2000-12-05 Research Corporation Technologies, Inc. 2β-substituted-6-alkylidene penicillanic acid derivatives as β-lactamase inhibitors
US6407091B1 (en) 1999-04-15 2002-06-18 Research Corporation Technologies, Inc. β-lactamase inhibiting compounds
EP1430060B1 (en) 2001-07-24 2006-09-13 Southern Methodist University Foundation for Research 7-alkylidene-3-substituted-3-cephem-4-carboxylates as beta-lactamase inhibitors.
JP2005525399A (ja) 2002-04-04 2005-08-25 アラムクス エルエルシー セリンおよびメタロ−β−ラクタマーゼの阻害剤
GB0711776D0 (en) * 2007-06-18 2007-07-25 Syngenta Participations Ag Substituted aromatic heterocyclic compounds as fungicides
JP6183053B2 (ja) * 2012-08-22 2017-08-23 宇部興産株式会社 テトラヒドロピラニルピリミジン化合物の製造方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4272439A (en) * 1978-06-02 1981-06-09 Schering Corporation 6-(Substituted-hydroxymethylene penams)
DE2927004A1 (de) * 1979-07-04 1981-05-27 Bayer Ag, 5090 Leverkusen Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors

Also Published As

Publication number Publication date
DD247678A5 (de) 1987-07-15
ES8704952A1 (es) 1987-04-16
PL145990B1 (en) 1988-12-31
NO165594C (no) 1991-03-06
SU1396969A3 (ru) 1988-05-15
ES548426A0 (es) 1986-11-16
PL256015A1 (en) 1986-11-18
FI85376B (fi) 1991-12-31
SU1508961A3 (ru) 1989-09-15
IL74190A0 (en) 1985-04-30
ES8705451A1 (es) 1987-05-01
NO850350L (no) 1985-07-31
ES8604972A1 (es) 1986-02-16
KR880001029B1 (ko) 1988-06-15
CS248747B2 (en) 1987-02-12
YU44636B (en) 1990-10-31
CS248733B2 (en) 1987-02-12
CS248748B2 (en) 1987-02-12
PL256013A1 (en) 1986-10-21
PL251750A1 (en) 1985-12-17
CS248746B2 (en) 1987-02-12
KR850005445A (ko) 1985-08-26
SU1503683A3 (ru) 1989-08-23
YU119587A (en) 1988-02-29
HU194567B (en) 1988-02-29
HUT37799A (en) 1986-02-28
ES539890A0 (es) 1986-02-16
YU119787A (en) 1988-04-30
SU1395144A3 (ru) 1988-05-07
HU194891B (en) 1988-03-28
PT79893A (en) 1985-02-01
PL147514B1 (en) 1989-06-30
YU44634B (en) 1990-10-31
FI850375A0 (fi) 1985-01-29
PL149242B1 (en) 1990-01-31
YU44770B (en) 1991-02-28
ES548428A0 (es) 1987-01-16
DD234015A5 (de) 1986-03-19
PL256014A1 (en) 1986-12-02
FI85376C (fi) 1992-04-10
PL145130B1 (en) 1988-08-31
PL149797B1 (en) 1990-03-31
ES548429A0 (es) 1987-04-16
YU44635B (en) 1990-10-31
PL256016A1 (en) 1986-12-02
YU119687A (en) 1988-04-30
ES548427A0 (es) 1987-05-01
YU44805B (en) 1991-02-28
IL74190A (en) 1989-09-28
HUT40443A (en) 1986-12-28
EG16904A (en) 1992-06-30
JPS61109791A (ja) 1986-05-28
ES8702916A1 (es) 1987-01-16
FI850375L (fi) 1985-07-31
YU119487A (en) 1988-02-29
NO165594B (no) 1990-11-26
ZA85682B (en) 1986-09-24
DD247677A5 (de) 1987-07-15
ES8700860A1 (es) 1986-11-16
YU14085A (en) 1987-12-31
PT79893B (en) 1987-02-03

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