CS196282B2 - Method of producing phenylesters of 2-alkoxycarbonyl aminobenzimidazol-5/6/-ylsulphonic acid - Google Patents

Method of producing phenylesters of 2-alkoxycarbonyl aminobenzimidazol-5/6/-ylsulphonic acid Download PDF

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Publication number
CS196282B2
CS196282B2 CS755620A CS562075A CS196282B2 CS 196282 B2 CS196282 B2 CS 196282B2 CS 755620 A CS755620 A CS 755620A CS 562075 A CS562075 A CS 562075A CS 196282 B2 CS196282 B2 CS 196282B2
Authority
CS
Czechoslovakia
Prior art keywords
acid
ester
methoxycarbonylamino
formula
nitro
Prior art date
Application number
CS755620A
Other languages
Czech (cs)
English (en)
Inventor
Heinz Loewe
Josef Urbanietz
Dieter Duewel
Reinhard Kirsch
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Priority to CS787241A priority Critical patent/CS196284B2/cs
Priority to CS787240A priority patent/CS196283B2/cs
Priority to CS787242A priority patent/CS196285B2/cs
Publication of CS196282B2 publication Critical patent/CS196282B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30—Nitrogen atoms not forming part of a nitro radical
    • C07D235/32—Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preventing Corrosion Or Incrustation Of Metals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
CS755620A 1974-08-28 1975-08-15 Method of producing phenylesters of 2-alkoxycarbonyl aminobenzimidazol-5/6/-ylsulphonic acid CS196282B2 (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
CS787241A CS196284B2 (cs) 1974-08-28 1978-11-06 Způsob výroby fenylesterů 2-alkoxykarbonylaminobenzimidazol- -5(B)-ylsulfonové kyseliny
CS787240A CS196283B2 (cs) 1974-08-28 1978-11-06 Způsob výroby fenylesterů 2-alkoxykarbonylamínobenzimidazol- -5(B)-ylsůlfOnové kyseliny
CS787242A CS196285B2 (cs) 1974-08-28 1978-11-06 Způsob výroby íenylesterů 2-alkoxykarbonylaminobenzimidazol- -5(B)-yIsulfonové kyseliny

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2441202A DE2441202C2 (de) 1974-08-28 1974-08-28 2-Carbalkoxyamino-benzimidazolyl-5(6)-sulfonsäure-phenylester, Verfahren zu ihrer Herstellung und diese enthaltende anthelmintische Mittel

Publications (1)

Publication Number Publication Date
CS196282B2 true CS196282B2 (en) 1980-03-31

Family

ID=5924288

Family Applications (1)

Application Number Title Priority Date Filing Date
CS755620A CS196282B2 (en) 1974-08-28 1975-08-15 Method of producing phenylesters of 2-alkoxycarbonyl aminobenzimidazol-5/6/-ylsulphonic acid

Country Status (30)

Country Link
US (2) US3996369A (xx)
JP (1) JPS5910349B2 (xx)
AT (1) AT349461B (xx)
BE (1) BE832858A (xx)
BG (3) BG23900A3 (xx)
CA (1) CA1059136A (xx)
CH (1) CH611606A5 (xx)
CS (1) CS196282B2 (xx)
DD (1) DD122974A5 (xx)
DE (1) DE2441202C2 (xx)
DK (1) DK137533C (xx)
EG (1) EG11811A (xx)
ES (1) ES440385A1 (xx)
FI (1) FI752396A (xx)
FR (1) FR2282880A1 (xx)
GB (2) GB1516508A (xx)
HU (1) HU172144B (xx)
IE (1) IE41655B1 (xx)
IL (1) IL47996A (xx)
IT (1) IT1041927B (xx)
KE (2) KE3089A (xx)
LU (1) LU73256A1 (xx)
MY (2) MY8100222A (xx)
NL (1) NL7509956A (xx)
NO (1) NO140592B (xx)
PL (4) PL100180B1 (xx)
SE (1) SE417508B (xx)
SU (3) SU582760A3 (xx)
ZA (1) ZA755485B (xx)
ZM (1) ZM12675A1 (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3132167A1 (de) * 1981-08-14 1983-03-03 Hoechst Ag, 6000 Frankfurt "5(6)-phenylsulfonyloxy-benzimidazolderivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung gegen leberegel"
DE2608238A1 (de) * 1976-02-28 1977-09-08 Hoechst Ag Substituierte phenylguanidine und verfahren zu ihrer herstellung
DE2653766A1 (de) * 1976-11-26 1978-06-01 Bayer Ag Substituierte benzolsulfonsaeureester, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
DE2836385A1 (de) * 1978-08-19 1980-03-06 Hoechst Ag Monocarboxylate von phenylguanidinsulfonsaeureestern, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
HU182782B (en) * 1979-12-04 1984-03-28 Chinoin Gyogyszer Es Vegyeszet Process for producing alkylthio-benzimidazoles
DE3232959A1 (de) * 1982-09-04 1984-03-08 Hoechst Ag, 6230 Frankfurt Substituierte benzolsulfonsaeureester, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
JPH0320378Y2 (xx) * 1986-11-29 1991-05-01
GB2546967B (en) 2016-01-27 2020-04-15 Thermo Fisher Scient Bremen Gmbh Quadrupole mass spectrometer
GB2552841B (en) 2016-08-12 2020-05-20 Thermo Fisher Scient Bremen Gmbh Method of calibrating a mass spectrometer

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH116815A (de) * 1924-06-14 1926-09-16 Ig Farbenindustrie Ag Verfahren zur Darstellung des Phenylesters der 4-Nitro-1-aminobenzol-2-sulfosäure.
US2134642A (en) * 1936-08-12 1938-10-25 Cie Nat Matieres Colorantes Azo dyestuff and process for the manufacture thereof
CH296894A (de) * 1949-07-18 1954-02-28 Ciba Geigy Verfahren zur Herstellung eines aminogruppenhaltigen aromatischen Sulfonsäureesters.
BE666795A (xx) * 1964-08-04 1966-01-13
US3562290A (en) * 1967-11-07 1971-02-09 Du Pont Process for making 2-benzimidazolecarbamic acid alkyl esters
BE793358A (fr) * 1971-12-27 1973-06-27 Hoechst Ag Nouveaux derives de 2-carbalcoxy-amino-benzimidazole presentantune activite anthelmintique et leur procede de preparation
JPS5529110B2 (xx) * 1972-12-25 1980-08-01
US3929824A (en) * 1972-12-29 1975-12-30 Syntex Inc 5(6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity
US3929821A (en) * 1972-12-29 1975-12-30 Syntex Inc 5 (6)-Benzene ring substituted benzimidazole-2-carbamate derivatives
ZA739220B (en) * 1972-12-29 1975-07-30 Syntex Inc 5(6)-benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity
US3929823A (en) * 1973-11-21 1975-12-30 Syntex Inc 5(6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity

Also Published As

Publication number Publication date
PL101537B1 (pl) 1979-01-31
PL101396B1 (pl) 1978-12-30
FR2282880A1 (fr) 1976-03-26
DK137533C (da) 1978-09-04
BE832858A (fr) 1976-03-01
DK384975A (da) 1976-02-29
CA1059136A (en) 1979-07-24
NO140592B (no) 1979-06-25
PL100180B1 (pl) 1978-09-30
LU73256A1 (xx) 1977-04-15
IE41655L (en) 1976-02-28
EG11811A (en) 1979-03-31
ES440385A1 (es) 1977-06-16
HU172144B (hu) 1978-06-28
SE7509441L (sv) 1976-03-01
SU591142A3 (ru) 1978-01-30
BG23900A3 (en) 1977-11-10
PL100496B1 (pl) 1978-10-31
ZM12675A1 (en) 1976-08-23
KE3089A (en) 1980-11-07
IL47996A (en) 1979-01-31
DK137533B (da) 1978-03-20
MY8100222A (en) 1981-12-31
IE41655B1 (en) 1980-02-27
DE2441202C2 (de) 1986-05-28
CH611606A5 (xx) 1979-06-15
US4216161A (en) 1980-08-05
AU8432375A (en) 1977-03-03
SU582760A3 (ru) 1977-11-30
SE417508B (sv) 1981-03-23
US3996369A (en) 1976-12-07
ATA663475A (de) 1978-09-15
GB1516508A (en) 1978-07-05
BG26373A3 (xx) 1979-03-15
JPS5910349B2 (ja) 1984-03-08
SU589912A3 (ru) 1978-01-25
JPS5148664A (en) 1976-04-26
DE2441202A1 (de) 1976-03-11
IT1041927B (it) 1980-01-10
IL47996A0 (en) 1975-11-25
NO752945L (xx) 1976-03-02
AT349461B (de) 1979-04-10
KE3090A (en) 1980-11-07
FI752396A (xx) 1976-02-29
MY8100220A (en) 1981-12-31
FR2282880B1 (xx) 1980-04-30
GB1516509A (en) 1978-07-05
ZA755485B (en) 1976-07-28
DD122974A5 (de) 1976-11-12
NL7509956A (nl) 1976-03-02
BG25222A3 (en) 1978-08-10

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