CR9966A - Acido 1-(1-(2-etoxietil-3-etil-7-(4-metilpiridin-2-ilamino)-1h-pirazolo[4,3-d]pirimidin-5-il)piperidina-4-carboxilico y las sales del mismo. - Google Patents

Acido 1-(1-(2-etoxietil-3-etil-7-(4-metilpiridin-2-ilamino)-1h-pirazolo[4,3-d]pirimidin-5-il)piperidina-4-carboxilico y las sales del mismo.

Info

Publication number
CR9966A
CR9966A CR9966A CR9966A CR9966A CR 9966 A CR9966 A CR 9966A CR 9966 A CR9966 A CR 9966A CR 9966 A CR9966 A CR 9966A CR 9966 A CR9966 A CR 9966A
Authority
CR
Costa Rica
Prior art keywords
acid
pyrimidin
piperidine
salts
etoxietil
Prior art date
Application number
CR9966A
Other languages
English (en)
Inventor
Brent Tollefson Michael
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of CR9966A publication Critical patent/CR9966A/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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Abstract

La presente invencion comprende el acido 1-(1-(2-etoxietil)-3-etil-7-(4-metilpiridin-2-ilamino)-1H-pirazolo[4,3-d]pirimidin-5-il)piperidina-4-carboxilico y sus sales. La invencion ademas comprende las composiciones framaceuticas, los procedimientos de tratamiento, y los procedimientos de sintesis que se refieren al acido 1-(1-(2-etoxietil9-3-etil-7-(4-metilpiridin-2-ilamino)-1H-pirazolo[4,3-d]pirimidin-5-il)piperidina-4-carboxilico y sus sales.
CR9966A 2005-11-10 2008-05-09 Acido 1-(1-(2-etoxietil-3-etil-7-(4-metilpiridin-2-ilamino)-1h-pirazolo[4,3-d]pirimidin-5-il)piperidina-4-carboxilico y las sales del mismo. CR9966A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73532005P 2005-11-10 2005-11-10

Publications (1)

Publication Number Publication Date
CR9966A true CR9966A (es) 2008-06-16

Family

ID=37685872

Family Applications (1)

Application Number Title Priority Date Filing Date
CR9966A CR9966A (es) 2005-11-10 2008-05-09 Acido 1-(1-(2-etoxietil-3-etil-7-(4-metilpiridin-2-ilamino)-1h-pirazolo[4,3-d]pirimidin-5-il)piperidina-4-carboxilico y las sales del mismo.

Country Status (30)

Country Link
US (2) US20090156618A1 (es)
EP (1) EP1948661B1 (es)
JP (1) JP4208959B1 (es)
KR (1) KR101012592B1 (es)
CN (1) CN101305007B (es)
AP (1) AP2008004437A0 (es)
AR (1) AR057885A1 (es)
AT (1) ATE435865T1 (es)
AU (1) AU2006313486B2 (es)
BR (1) BRPI0618284A2 (es)
CA (1) CA2629339C (es)
CR (1) CR9966A (es)
DE (1) DE602006007728D1 (es)
DK (1) DK1948661T3 (es)
DO (1) DOP2006000248A (es)
EA (1) EA200800920A1 (es)
EC (1) ECSP088441A (es)
ES (1) ES2326919T3 (es)
HK (1) HK1120803A1 (es)
IL (1) IL190456A (es)
MA (1) MA29943B1 (es)
NL (1) NL2000291C2 (es)
NO (1) NO20082593L (es)
PE (1) PE20070764A1 (es)
RS (1) RS20080197A (es)
TN (1) TNSN08209A1 (es)
TW (1) TW200738723A (es)
UY (1) UY29909A1 (es)
WO (1) WO2007054778A1 (es)
ZA (1) ZA200803173B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ590922A (en) * 2008-08-01 2012-09-28 Biocryst Pharm Inc Piperidine derivatives as jak3 inhibitors
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EP2556820A4 (en) * 2010-04-05 2015-01-21 Sk Chemicals Co Ltd COMPOSITION CONTAINING PDE5 INHIBITOR FOR MITIGATION OF SKIN WRINKLES
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